Azine-substituted phenylacetic acid derivatives and fungicides containing these

ABSTRACT

Compounds of the formula I ##STR1## where X is hydrogen, halogen, alkyl, alkoxy, trifluoromethyl, cyano or nitro, 
     Y is an amino, methylamino or dimethylamino group, 
     Z is a group CHCH 3 , CHOCH 3  or NOCH 3 , 
     R is hydrogen or alkyl, 
     A is hydrogen, alkyl, haloalkyl or cycloalkyl, 
     B is unsubstituted or substituted alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl, heterocyclyl, aryl, heteroaryl, arylalkyl, heteroarylalkyl or the group ##STR2## where W is hydrogen, alkyl, alkoxy, alkylthio, alkylamino or dialkylamino, unsubstituted or substituted aryl or heteroaryl, unsubstituted or substituted aryloxy, arylthio, arylamino or aryl-N-(C 1  -C 6  -alkyl)amino, heteroaryloxy, heteroarylthio, heteroarylamino or heteroaryl-N-(alkyl)amino or 
     A and B, together with the C atom whose substituents they are, are an isocyclic or heterocyclic ring which can also be quinonoid, 
     and fungicides containing these compounds.

The present invention relates to compounds of the formula I ##STR3##where the substituents have the following meanings X is hydrogen, cyano,nitro, trifluoromethyl, halogen, C₁ -C₆ -alkyl or C₁ -C₆ -alkoxy;

Y is methoxy, amino, methylamino or dimethylamino;

Z is CHCH₃, CHOCH₃ or NOCH₃ ;

R is hydrogen or C₁ -C₆ -alkyl;

A is hydrogen, C₁ -C₆ -alkyl, C₁ -C₆ -haloalkyl or C₃ -C₇ -cycloalkyl;

B is unsubstituted or substituted C₁ -C₆ -alkyl, C₂ -C₆ -alkenyl, C₂ -C₆-alkynyl, C₃ -C₇ -cycloalkyl, C₅ -C₇ -cycloalkenyl,

an unsubstituted or substituted, saturated or partially unsaturatedheterocyclyl,

unsubstituted or substituted aryl, which may be fused,

unsubstituted or substituted 5- or 6-membered heteroaryl, which may bebenzo- or hetero-fused,

unsubstituted or substituted aryl-C₁ -C₆ -alkyl or heteroaryl-C₁ -C₆-alkyl, or

C(═O)W;

where

W is hydrogen,

unsubstituted or substituted C₁ -C₆ -alkyl,

C₁ -C₆ -alkoxy, C₁ -C₆ -alkylthio, C₁ -C₆ -alkylamino or di-C₁ -C₆-alkylamino,

unsubstituted or substituted aryl, heteroaryl, aryloxy, arylthio,arylamino, aryl-N-(C₁ -C₆ -alkyl)amino, heteroaryloxy, heteroarylthio,heteroarylamino or heteroaryl-N-(C₁ -C₆ -alkyl)amino;

or

A and B, together with the C atom whose substituents they are, are anunsubstituted or substituted, saturated or unsaturated 3- to 7-memberedisocyclic ring or 5- to 7-membered heterocyclic ring, which may be fusedand which may also be quinonoid.

The invention additionally relates to processes for preparing thesecompounds, compositions containing them, and their use for theproduction of compositions of this type and for the control of pests andharmful fungi.

EP-A-499823 discloses the use of hydrazone-substituted phenylacetic acidderivatives as agrochemical fungicides. Their action, however, isunsatisfactory.

It is an object of the present invention to provide novel compoundshaving improved properties.

We have now found that this object is achieved by the compounds definedat the beginning, processes for their preparation, compositionscontaining them and their use.

The active compounds can be synthesized by general methods for thepreparation of unsymmetrical azines, as are described eg. inHouben/Weyl, "Methoden der organischen Chemie" [Methods of OrganicChemistry] Vol. 10/2, pp.104-111 and Vol. E 14 b, Part 1, pp. 655-673.

For example (see Scheme 1), azines of the formula I can be prepared byreaction of two carbonyl compounds II and III with hydrazine, one of itsacid addition salts or its hydrate in a suitable solvent and ifappropriate in the presence of a catalytically active compound, eg.acetic acid, and the unsymmetrical azine I can be isolated from theadditionally resulting symmetrical azines VI and VII by use of asuitable separation method such as eg. column chromatography, fractionalcrystallization or distillation. The compounds II are accessible bygenerally known methods of organic synthesis or are commerciallyavailable; the preparation of compounds III is described in EP 499823and literature cited there.

It is also possible to bring II and a carbonyl compound VIII to reactionwith hydrazine, one of its acid addition salts or its hydrate, in whichcase an unsymmetrical azine IX mixed with the symmetrical azines VI andX results and can be isolated by the customary separation methods. Thevariable V in the formulae VIII and IX is a group which can be convertedto the group Y--C(═O)--C═Z by standard methods of organic chemistry, forexample as described for similar compounds in EP 463488, pp. 7-8. It maybe advantageous first to synthesize the azines IX and then to preparethe active compound I by conversion of the group V to the groupY--C(═O)--C═Z. The group V is advantageously selected such that itremains unchanged under the conditions of the azine synthesis. It mayalso be advantageous in the starting material of the formula II toemploy a functional substituent in the group B in protected form and todeprotect it after azine formation. The preparation of the carbonylcompounds VIII can be carried out by the methods of organic synthesismentioned for III or generally known.

Furthermore, azines of the formula I or IX can be prepared by convertinga carbonyl compound II to a hydrazone IV by known methods and reactingthis with a carbonyl compound III or VIII in a suitable solvent and ifappropriate in the presence of a catalytically active species [see eg.Liebigs Ann. Chem. 640 (1961), 37]. Also in this process, with theunsymmetrical azine I or IX, the symmetrical azines VI and VII or X canbe formed as by-products which have to be separated off. Instead of thecarbonyl compounds, their Schiff's bases (which can be prepared bygenerally known methods) can also be employed [Liebigs Ann. Chem. 657(1962), 39]; this can be advantageous in relation to the yield andselectivity of the reaction. IX can be converted to I by standardmethods (see above). ##STR4##

It is also possible [Sulfur Lett. 9 (1989), 227], to generate hydrazonesIV by thermolysis of o-ethylsulfamoylbenzoyl hydrazides XII (accessiblefrom N-ethylsaccharin XI, for preparation see eg. J. Pharm. Soc. Jap. 75(1955), 153) in the presence of a carbonyl compound III or VIII and toconvert in situ to the azine I or IX (Scheme 2); the method may beadvantageous for the selective preparation of the unsymmetrical azines.##STR5##

The compounds of the formula I or IX can also be prepared by reaction ofcarbonyl compounds III or VIII, preferably aldehydes (R═H), withphosphazines XIII or metal salts of the phosphonohydrazides XIV in anaza-analogous Wittig reaction [Chem. Ber. 94 (1961), 2477]orHorner-Emmons reaction [Synthesis 1986, 298] (Scheme 3). The synthesisof the starting materials XIII and XIV is described or mentioned in theabove literature. ##STR6##

Azines XVI corresponding to the compounds of the formula I in which Z isa group NOCH₃ and Y is a group NHCH₃, can be prepared either by reactinga carbonyl compound II and hydrazine, one of its acid addition salts orits hydrate or, instead of this starting material combination, ahydrazone IV with an aldehyde or ketone equivalent V (Scheme 4). Thecyclic hemiaminals V are accessible by treating the carbonyl compoundsXV (corresponding to compounds in which R is alkyl, preferably methyl)with methylamine in a suitable solvent, eg. water, methanol ortetrahydrofuran or a mixture of such solvents. Instead of III, V canalso be reacted with XII, XIII or XIV by the methods described inSchemes 2 and 3 to give compounds of the formula XVI. ##STR7##

Compounds of the formula XVI can also be prepared by reacting azines ofthe formula XVII (corresponding to formula I, where Z═NOCH₃ and Y═OR³,R³ being short-chain alkyl, preferably methyl) with methylamine asdescribed above. The starting materials XVII are accessible eg. by theabove methods (see Schemes 1-3).

In the definitions of the symbols given in the above formulae,collective terms were used which are generally representative of thefollowing substituents:

halogen: fluorine, chlorine, bromine and iodine;

alkyl: saturated, straight-chain or branched hydrocarbon radicals having1 to 6 carbon atoms, such as methyl, ethyl, propyl, 1-methylethyl,butyl, 1-methylpropyl, 2-methylpropyl, 1,1-dimethylethyl, pentyl,1-methylbutyl, 2-methylbutyl, 3-methylbutyl, 2,2-dimethylpropyl,1-ethylpropyl, hexyl, 1,1-dimethylpropyl, 1,2-dimethylpropyl,1-methylpentyl, 2-methylpentyl, 3-methylpentyl, 4-methylpentyl,

1,1-dimethylbutyl, 1,2-dimethylbutyl, 1,3-dimethylbutyl,2,2-dimethylbutyl, 2,3-dimethylbutyl, 3,3-dimethylbutyl, 1-ethylbutyl,2-ethylbutyl, 1,1,2-trimethylpropyl, 1,2,2-trimethylpropyl,1-ethyl-1-methylpropyl and 1-ethyl-2-methylpropyl;

alkoxy: straight-chain or branched alkyl groups having 1 to 6 carbonatoms (as mentioned above), which are bonded to the ring system via anoxygen atom (--O--);

alkylthio: straight-chain or branched alkyl groups having 1 to 6 carbonatoms (as mentioned above), which are bonded to the ring system via asulfur atom (--S--);

alkylamino: a straight-chain or branched alkyl group having 1 to 6carbon atoms (as mentioned above), which is bonded to the ring systemvia an amino group (--NH--);

dialkylamino: an amino group which carries two straight-chain orbranched alkyl groups which are independent of one another, each having1 to 6 carbon atoms (as mentioned above);

haloalkyl: straight-chain or branched alkyl groups having 1 to 6,preferably 1 to 4, in particular 1 to 2 carbon atoms (as mentionedabove), it being possible for the hydrogen atoms in these groups to bepartly or completely replaced by halogen atoms as mentioned above, eg.fluoromethyl, difluoromethyl, trifluoromethyl, 1-fluoroethyl,2-fluoroethyl, 1,1-difluoroethyl, 1,2-difluoroethyl, 2,2-difluoroethyl,2,2,2-trifluoroethyl, 1,1,2,2-tetrafluoroethyl, pentafluoroethyl,fluoropropyl, fluorobutyl, fluoropentyl, fluorohexyl, heptafluoropropyl,nonafluorobutyl, chloromethyl, trichloromethyl, 1-chloroethyl,2-chloroethyl, 2,2,2-trichloroethyl, chloropropyl, chlorobutyl,chloropentyl, chlorohexyl, bromomethyl, bromoethyl, dibromoethyl andiodomethyl;

alkenyl: unsaturated, straight-chain or branched hydrocarbon radicalshaving 2 to 6 carbon atoms and a double bond in any desired position,eg. ethenyl, 1-propenyl, 2-propenyl, 1-methylethenyl, 1-butenyl,2-butenyl, 3-butenyl, 1-methyl-1-propenyl, 2-methyl-1-propenyl,1-methyl-2-propenyl, 2-methyl-2-propenyl, 1-pentenyl, 2-pentenyl,3-pentenyl, 4-pentenyl, 1-methyl-1-butenyl, 2-methyl-1-butenyl,3-methyl-1-butenyl, 1-methyl-2-butenyl, 2-methyl-2-butenyl,3-methyl-2-butenyl, 1-methyl-3-butenyl, 2-methyl-3-butenyl,3-methyl-3-butenyl, 1,1-dimethyl-2-propenyl, 1,2-dimethyl-1-propenyl,1,2-dimethyl-2-propenyl, 1-ethyl-1-propenyl, 1-ethyl-2-propenyl,1-hexenyl, 2-hexenyl, 3-hexenyl, 4-hexenyl, 5-hexenyl,1-methyl-1-pentenyl, 2-methyl-1-pentenyl, 3-methyl-1-pentenyl,4-methyl-1-pentenyl, 1-methyl-2-pentenyl, 2-methyl-2-pentenyl,3-methyl-2-pentenyl, 4-methyl-2-pentenyl, 1-methyl-3-pentenyl,2-methyl-3-pentenyl, 3-methyl-3-pentenyl, 4-methyl-3-pentenyl,1-methyl-4-pentenyl, 2-methyl-4-pentenyl, 3-methyl-4-pentenyl,4-methyl-4-pentenyl, 1,1-dimethyl-2-butenyl, 1,1-dimethyl-3-butenyl,1,2-dimethyl-1-butenyl, 1,2-dimethyl-2-butenyl, 1,2-dimethyl-3-butenyl,1,3-dimethyl-1-butenyl, 1,3-dimethyl-2-butenyl, 1,3-dimethyl-3-butenyl,2,2-dimethyl-3-butenyl, 2,3-dimethyl-1-butenyl, 2,3-dimethyl-2-butenyl,2,3-dimethyl-3-butenyl, 3,3-dimethyl-1-butenyl, 3,3-dimethyl-2-butenyl,1-ethyl-1-butenyl, 1-ethyl-2-butenyl, 1-ethyl-3-butenyl,2-ethyl-1-butenyl, 2-ethyl-2-butenyl, 2-ethyl-3-butenyl,1,1,2-trimethyl-2-propenyl, 1-ethyl-1-methyl-2-propenyl,1-ethyl-2-methyl-1-propenyl and -1-ethyl-2-methyl-2-propenyl;

alkynyl: straight-chain or branched hydrocarbon groups having 2 to 6carbon atoms and a triple bond in any desired position, eg. C₂ -C₆-alkynyl such as ethynyl, 1-propynyl, 2-propynyl, 1-butynyl, 2-butynyl,3-butynyl, 1-methyl-2-propynyl, 1-pentynyl, 2-pentynyl, 3-pentynyl,4-pentynyl, 1-methyl-2-butynyl, 1-methyl-3-butynyl, 2-methyl-3-butynyl,3-methyl-1-butynyl, 1,1-dimethyl-2-propynyl, 1-ethyl-2-propynyl,1-hexynyl, 2-hexynyl, 3-hexynyl, 4-hexynyl, 5-hexynyl,1-methyl-2-pentynyl, 1-methyl-3-pentynyl, 1-methyl-4-pentynyl,2-methyl-3-pentynyl, 2-methyl-4-pentynyl, 3-methyl-1-pentynyl,3-methyl-4-pentynyl, 4-methyl-1-pentynyl, 4-methyl-2-pentynyl,1,1-dimethyl-2-butynyl, 1,1-di-methyl-3-butynyl, 1,2-dimethyl-3-butynyl,2,2-dimethyl-3-butynyl, 3,3-dimethyl-1-butynyl, 1-ethyl-2-butynyl,1-ethyl-3-butynyl, 2-ethyl-3-butynyl and 1-ethyl-1-methyl-2-propynyl;

cycloalkyl: monocyclic or bicyclic alkyl groups having 3 to 7 carbonring members, eg. cyclopropyl, cyclobutyl, cyclopentyl, cyclohexyl,cycloheptyl and norbornyl;

cycloalkenyl: monocyclic or bicyclic alkyl groups having 5 to 7 carbonring members, eg. cyclopentenyl, cyclohexenyl, cycloheptenyl andnorbornenyl;

heterocyclyl: saturated or partially unsaturated ring systems which, inaddition to carbon ring members, can also contain 1 to 3 hetero atomsfrom the group consisting of oxygen, sulfur and nitrogen, eg. oxiranyl,oxetanyl, tetrahydrofur-2-yl, tetrahydrofur-3-yl, tetrahydrothien-2-yl,tetrahydrothien-3-yl, pyrrolidin-2-yl, pyrrolidin-3-yl,isoxazolidin-3-yl, isoxazolidin-4-yl, isoxazolidin-5-yl,isothiazolidin-3-yl, isothiazolidin-4-yl, isothiazolidin-5-yl,pyrazolidin-3-yl, pyrazolidin-4-yl, pyrazolidin-5-yl, oxazolidin-2-yl,oxazolidin-4-yl, oxazolidin-5-yl, thiazolidin-2-yl, thiazolidin-4-yl,thiazolidin-5-yl, imidazolidin-2-yl, imidazolidin-4-yl,1,2,4-oxadiazolidinyl, 1,3,4-oxazolidinyl, 1,2,4-thiazolidinyl,1,2,4-triazolidinyl, 1,2,5-triazolidinyl, 2,3-dihydrofuryl,2,5-dihydrofuryl, 2,3-dihydrothienyl, 2,5-dihydrothienyl,2,3-dihydropyrrolyl, 2,5-dihydropyrrolyl, 2,3-dihydroisoxazolyl,2,5-dihydroisoxazolyl, 4,5-dihydroisoxazolyl, 2,3-dihydroisothiazolyl,2,5-dihydroisothiazolyl, 4,5-dihydroisothiazolyl, 2,3-dihydropyrazolyl,2,5-dihydropyrazolyl, 4,5-dihydropyrazolyl, 2,5-dihydrooxazolyl,3,4-dihydrooxazolyl, 2,5-dihydrothiazolyl, 3,4-dihydrothiazolyl,2,5-dihydroimidazolyl, 3,4-dihydroimidazolyl, piperidin-2-yl,piperidin-3-yl, piperidin-4-yl, tetrahydropyridazin-3-yl,tetrahydropyridazin-4-yl, tetrahydropyrimidin-2-yl,tetrahydropyrimidin-4-yl, tetrahydropyrimidin-5-yl,tetrahydropyrazin-2-yl, tetrahydro-1,3,5-triazinyl,tetrahydro-1,2,4-triazinyl, dihydro-1,3-oxazinyl, 1,3-dithian-2-yl,tetrahydropyranyl, 1,3-dioxolan-2-yl, 4H-1,3-thiazin-2-yl,4H-3,1-benzothiazin-2-yl, 2H-1,4-benzothiazin-3-yl,2H-1,4-benzoxazin-3-yl, 1,1-dioxotetrahydrothienyl,dihydro-1,3-oxazin-2-yl, morpholinyl or dihydroquinazolinyl;

aryl, aryloxy, arylthio and arylamino: aromatic, mono- or polycyclichydrocarbons which are bonded to the ring system directly or via anoxygen atom (-oxy), a sulfur atom (-thio) or an amino group (-amino),eg. phenyl, naphthyl, anthryl and phenanthryl or the corresponding oxy,thio or amino groups;

arylalkyl: straight-chain or branched alkyl groups having 1 to 6 carbonatoms (as mentioned above), which can carry one of the above arylradicals in any desired position;

arylalkylamino: alkylamino groups having 1 to 6, preferably 1 to 4, inparticular 1 to 2 carbon atoms (as mentioned above), which carry one ofthe abovementioned aryl radicals on the nitrogen atom;

heteroaryl, heteroaryloxy, -thio and -amino: aromatic, mono- orpolycyclic systems which, in addition to carbon ring members, can alsocontain oxygen, sulfur and/or nitrogen atoms as ring members and whichare bonded to the ring system directly or via an exocyclic oxygen atom(-oxy), sulfur atom (-thio) or an amino group (-amino), eg.

5-membered heteroaryl, containing one to four nitrogen atoms or one tothree nitrogen atoms and a sulfur or oxygen atom: 5-membered ringheteroaryl groups which, in addition to carbon atoms, can contain one tofour nitrogen atoms or one to three nitrogen atoms and a sulfur oroxygen atom as ring members;

benzo-fused 5-membered heteroaryl, containing one to three nitrogenatoms or a nitrogen atom and an oxygen or sulfur atom: 5-membered ringheteroaryl groups which, in addition to carbon atoms, can contain one tofour nitrogen atoms or one to three nitrogen atoms and a sulfur oroxygen atom as ring members, and in which two adjacent carbon ringmembers or a nitrogen and an adjacent carbon ring member can be bridgedby a buta-1,3-dien-1,4-diyl group;

5-membered heteroaryl bonded via nitrogen, containing one to fournitrogen atoms, or benzo-fused 5-membered heteroaryl bonded vianitrogen, containing one to three nitrogen atoms: 5-membered heteroarylgroups which, in addition to carbon atoms, can contain one to fournitrogen atoms or one to three nitrogen atoms as ring members, and inwhich two adjacent carbon ring members or a nitrogen and an adjacentcarbon ring member can be bridged by a buta-1,3-dien-1,4-diyl group,these rings being bonded to the ring system via one of the nitrogen ringmembers;

6-membered heteroaryl, containing one to three or one to four nitrogenatoms: 6-membered heteroaryl groups which, in addition to carbon atoms,can contain one to three or one to four nitrogen atoms as ring members;

benzo-fused 6-membered heteroaryl, containing one to three nitrogenatoms: 6-membered ring heteroaryl groups which, in addition to carbonatoms, can contain one to three nitrogen atoms as ring members, and inwhich two adjacent carbon ring members or a nitrogen and an adjacentcarbon ring member can be bridged by a buta-1,3-dien-1,4-diyl group;

e.g. fur-2-yl, fur-3-yl, thien-2-yl, thien-3-yl, pyrrol-1-yl,pyrrol-2-yl, pyrrol-3-yl, isoxazol-3-yl, isoxazol-4-yl, isoxazol-5-yl,isothiazol-3-yl, isothiazol-4-yl, isothiazol-5-yl, pyrazol-1-yl,pyrazol-3-yl, pyrazol-4-yl, pyrazol-5-yl, oxazol-2-yl, oxazol-4-yl,oxazol-5-yl, thiazol-2-yl, thiazol-4-yl, thiazol-5-yl, imidazol-1-yl,imidazol-2-yl, imidazol-4-yl, imidazol-5-yl, 1,2,4-thiadiazolyl,1,3,4-thiadiazolyl, 1,2,4-oxadiazolyl, t,3,4-oxadiazolyl,1,2,4-triazolyl, tetrazolyl, pyrid-2-yl, pyrid-3-yl, pyrid-4-yl,pyridazin-3-yl, pyridazin-4-yl, pyrimidin-2-yl, pyrimidin-4-yl,pyrimidin-5-yl, pyrazin-2-yl, 1,2,4-triazinyl, 1,3,5-triazinyl and1,2,4,5-tetrazinyl; adjacent substituents of the heteroaromatic can inthis case be fused to an aromatic or heteroaromatic ring such thatheteroaryl is also fused ring systems such as eg. benzofuryl,isobenzofuryl, benzothien-2-yl, benzothien-3-yl, benzothien-4-yl,benzothien-5-yl, benzothien-6-yl, benzothien-7-yl, indol-1-yl,indol-2-yl, indol-3-yl, isoindolyl, benzisoxazolyl, benzisothiazolyl,benzothiazol-2-yl, benzothiazol-4-yl, benzothiazol-5-yl,benzothiazol-6-yl, benzothiazol-7-yl, indazolyl, benzimidazolyl,benzotriazolyl, dibenzofuryl, dibenzothienyl, carbazolyl, acridinyl,phenanthridinyl, quinolin-2-yl, quinolin-3-yl, quinolin-4-yl,quinolin-5-yl, quinolin-6-yl, quinolin-7-yl, quinolin-8-yl,isoquinolin-1-yl, isoquinolin-3-yl, isoquinolin-4-yl, phthalazinyl,quinazolinyl, quinoxalinyl, cinnolinyl, 1,5-naphthyridinyl,1,6-naphthyridinyl, 1,7-naphthyridinyl, 1,8-naphthyridinyl, pteridinyl,pyrrolopyridinyl, pyrrolypyridazinyl, pyrrolopyrimidinyl,pyrrolopyrazinyl, pyrrolo-1,2,4-triazinyl, furopyridinyl,furopyridazinyl, furopyrimidinyl, furopyrazinyl, thienopyridinyl,thienopyridazinyl, thienopyrimidinyl, thienopyrazinyl, imidazopyridinyl,imidazolopyridazinyl, imidazopyrimidinyl, purinyl, imidazopyrazinyl,pyrazolopyridinyl, pyrazolopyridazinyl, pyrazolopyrimidinyl,pyrazolopyrazinyl, isoxazolopyrazinyl, oxazolopyridinyl,oxazolopyrimidinyl, isothiazolopyrimidinyl and triazolopyrimidinyl orthe corresponding oxy, thio and amino groups;

hetarylalkyl: straight-chain or branched alkyl groups having 1 to 6carbon atoms (as mentioned above), which carry one of the aboveheteroaryl radicals in any desired position;

hetarylalkylamino: alkylamino groups having 1 to 6 carbon atoms (asmentioned above), which carry one of the abovementioned heteroarylradicals on the nitrogen atom;

A and B, together with the C atom to which they are bonded, are asaturated or unsaturated, 3- to 7-membered isocyclic or 5- to 7-memberedheterocyclic ring which may be fused or unfused, eg. cyclopropylidene,cyclobutylidene, cyclopentylidene, cyclopentenylidene, cyclohexylidene,cyclohexenylidene, cycloheptylidene, cycloheptenylidene,4-oxohexa-2,5-dien-1-ylidene, tetrahydrothien-3-ylidene,tetrahydropyran-4-ylidene, dihyropyran-4-ylidene,tetrahydrothiopyran-4-ylidene or piperidin-4-ylidene.

In the definition of the compounds I, a few of the substituentsillustrated above were additionally described as unsubstituted orsubstituted. This is understood as meaning that in these radicalshydrogen atoms can be replaced by the groups described in greater detailin the following:

unsubstituted or substituted in relation to alkyl, alkenyl and alkynyl:the substituents can be partially or completely halogenated and/orcarry, for example, one to three, preferably one, of the followinggroups:

cyano, nitro, hydroxyl, mercapto, amino, formyl, carboxyl, formyloxy,aminocarbonyl, hydroxyaminocarbonyl, formamido, aminothiocarbonyl,hydroxysulfinyl, hydroxysulfinyl,

in addition alkyl, alkenyl or alkynyl groups which are bonded to thesubstituents via oxygen (--O--), sulfur (--S--), amino (--NH--),alkylamino [-N(alkyl)-], carbonyl (--CO--), carbonyloxy (--CO--O--),oxycarbonyl (--O--CO--), aminocarbonyl (--NH--CO--), oxyaminocarbonyl(--O--NH--CO--), carbonylamino (--CO--NH--), carbonylalkylamino[--CO--N(alkyl)-], sulfoxyl, sulfinyl, sulfinyl, sulfinyloxy orsulfinyloxy,

in addition cycloalkyl, cycloalkenyl, heterocyclyl, aryl or heteroarylgroups which are bonded to the substituents directly or via oxygen(--O--), sulfur (--S--), amino (--NH--), alkylamino [-N(alkyl)-],carbonyl (--CO--), carbonyloxy (--CO--O--), oxycarbonyl (--O--CO--),aminocarbonyl (--NH--CO--), oxyaminocarbonyl (--O--NH--CO--),carbonylamino (--CO--NH--), carbonylalkylamino [--CO--N(alkyl)-],sulfoxyl, sulfinyl, sulfynyl, sulfynyloxy or sulfinyloxy,

in addition trialkylsilyl (a silyl group with three C₁ -C₄ -alkylradicals which are independent of one another), dialkoxyphosphinyl (aphosphinyl group having two C₁ -C₄ -alkoxy radicals which areindependent of one another) or bis(aryloxy)phosphinyl,

in addition a group --ON═CR'R", where R' is hydrogen, alkyl, alkenyl oralkynyl and R" is hydrogen, alkyl, alkoxy, alkenyl or alkynyl;

unsubstituted or substituted in relation to cycloalkyl, cycloalkenyl andheterocyclyl: the substituents can be partially or completelyhalogenated and/or carry, for example, one to three, preferably one, ofthe following groups:

cyano, nitro, hydroxyl, mercapto, amino, formyl, carboxyl, formyloxy,aminocarbonyl, hydroxyaminocarbonyl, formamido, aminothiocarbonyl,hydroxysulfinyl, hydroxysulfinyl,

in addition alkyl, alkenyl or alkynyl groups which are bonded to thesubstituents directly or via oxygen (--O--), sulfur (--S--), amino(--NH--), alkylamino [-N(alkyl)-], carbonyl (--CO--), carbonyloxy(--CO--O--), oxycarbonyl (--O--CO--), aminocarbonyl (--NH--CO--),oxyaminocarbonyl (--O--NH--CO--), carbonylamino (--CO--NH--),carbonylalkylamino [--CO--N(alkyl)-], sulfoxyl, sulfinyl, sulfinyl,sulfinyloxy or sulfinyloxy,

in addition cycloalkyl, cycloalkenyl, heterocyclyl, aryl or heteroarylgroups which are bonded to the substituents directly or via oxygen(--O--), sulfur (--S--), amino (--NH--), alkylamino [-N(alkyl)-],carbonyl (--CO--), carbonyloxy (--CO--O--), oxycarbonyl (--O--CO--),aminocarbonyl (--NH--CO--), oxyaminocarbonyl (--O--NH--CO--),carbonylamino (--CO--NH--), carbonylalkylamino [--CO--N(alkyl)-],sulfoxyl, sulfinyl, sulfinyl, sulfinyloxy or sulfinyloxy,

in addition trialkylsilyl (a silyl group with three C₁ -C₄ -alkylradicals which are independent of one another), dialkoxyphosphinyl (aphosphinyl group having two C₁ -C₄ -alkoxy radicals which areindependent of one another) or bis(aryloxy)phosphinyl,

in addition a group --ON═CR'R", where R' is hydrogen, alkyl, alkenyl oralkynyl and R" is hydrogen, alkyl, alkoxy, alkenyl or alkynyl;

unsubstituted or substituted in relation to aryl and heteroaryl: thesubstituents can be partially or completely halogenated and/or carry,for example, one to three of the following groups:

cyano, nitro, hydroxyl, mercapto, amino, formyl, carboxyl, formyloxy,aminocarbonyl, hydroxyaminocarbonyl, formamido, aminothiocarbonyl,hydroxysulfinyl, hydroxysulfinyl,

in addition alkyl, alkenyl or alkynyl groups which are bonded to thesubstituents directly or via oxygen (--O--), sulfur (--S--), amino(--NH--), alkylamino [-N(alkyl)-], carbonyl (--CO--), carbonyloxy(--CO--O--), oxycarbonyl (--O--CO--), aminocarbonyl (--NH--CO--),oxyaminocarbonyl (--O--NH--CO--), carbonylamino (--CO--NH--),carbonylalkylamino [--CO--N(alkyl)-], sulfoxyl, sulfinyl, sulfinyl,sulfynyloxy or sulfinyloxy,

in addition cycloalkyl, cycloalkenyl, heterocyclyl, aryl or heteroarylgroups which are bonded to the substituents directly or via oxygen(--O--), sulfur (--S--), amino (--NH--), alkylamino [-N(alkyl)-],carbonyl (--CO--), carbonyloxy (--CO--O--), oxycarbonyl (--O--CO--),aminocarbonyl (--NH--CO--), oxyaminocarbonyl (--O--NH--CO--),carbonylamino (--CO--NH--), carbonylalkylamino [--CO--N(alkyl)-],sulfoxyl, sulfinyl, sulfinyl, sulfinyloxy or sulfinyloxy,

in addition trialkylsilyl (a silyl group with three C₁ -C₄ -alkylradicals which are independent of one another), dialkoxyphosphinyl (aphosphinyl group having two C₁ -C₄ -alkoxy radicals which areindependent of one another) or bis(aryloxy)phosphinyl,

in addition a group --ON═CR'R", where R' is hydrogen, alkyl, alkenyl oralkynyl and R" is hydrogen, alkyl, alkoxy, alkenyl or alkynyl.

The expression "partially or completely halogenated" is intended toexpress that in the corresponding radicals the hydrogen atoms bonded toC atoms are partially or completely replaced by identical or differenthalogen atoms.

In the abovementioned substituents, halogen and the organicsubstructures in each case have the abovementioned meanings. For theirparts, these substituents can again be substituted by one or more of theabovementioned radicals.

The compounds according to the invention can be obtained duringpreparation as stereoisomers (eg. Z/E isomers of C═C or C═N doublebonds, enantiomers or diastereomers), which can be separated by thecustomary methods (chromatography, crystallization, distillation). Boththe individual isomers and their mixtures are suitable as fungicides andare covered by the invention.

With respect to their biological action, compounds I are preferred inwhich X is hydrogen, chlorine, bromine, methyl or methoxy.

In addition, compounds I are preferred in which Y is methoxy and Z ismethoxymethylene.

Additionally, compounds I are preferred in which Y is methoxy and Z ismethoxyimino.

In addition, compounds I are preferred in which Y is methoxy and Z ismethylmethylene.

Additionally, compounds I are preferred in which Y is methoxy ormethylamino.

In addition, compounds I are preferred in which Y is methylamino and Zis methoxyimino.

In addition, compounds I are preferred in which Y is methylamino and Zis methoxymethylene.

In addition, compounds I are preferred in which Y is methylamino and Zis methylmethylene.

In addition, compounds I are preferred in which R is hydrogen or methyl.

In addition, compounds I are preferred in which A is hydrogen,cyclopropyl, C₁ -C₃ -alkyl or C₁ -C₂ -haloalkyl, in particular hydrogen,cyclopropyl, methyl, ethyl, isopropyl or trifluoromethyl.

Additionally, compounds I are preferred in which B is unsubstituted orsubstituted alkyl or cycloalkyl.

In particular, compounds I are preferred in which B is C₁ -C₁₂ -alkyl orC₃ -C₇ -cycloalkyl.

In addition, compounds I are preferred in which B is unsubstituted orsubstituted aryl.

In particular, compounds I are preferred in which B is aryl(particularly phenyl or naphthyl) which is partially or completelyhalogenated and/or carries a group --CR^(a) ═NR^(b) (R^(a) =hydrogen,amino, C₁ -C₄ -alkyl, C₁ -C₄ -alkoxy, C₁ -C₄ -alkylthio or C₁ -C₄-alkylamino; R^(b) =C₁ -C₄ -alkyl or C₁ -C₄ -alkoxy), and/or one tothree of the following groups: cyano, nitro, hydroxyl, mercapto, formyl,carboxyl, aminocarbonyl, cyanomethyl, C₁ -C₆ -alkyl, C₃ -C₆ -cycloalkyl,C₁ -C₄ -haloalkyl, C₂ -C₄ -alkenyl, C₂ -C₄ -alkynyl, C₁ -C₆ -alkoxy, C₃-C₆ -cycloalkoxy, C₁ -C₄ -haloalkoxy, mono- or di-C₁ -C₄ -alkoxy-C₁ -C₂-alkyl, C₁ -C₄ -alkylthio, C₃ -C₆ -cycloalkylthio, C₁ -C₆-alkylcarbonyl, C₁ -C₆ -alkoxycarbonyl, C₁ -C₆ -alkylcarbonyloxy, C₁ -C₄-alkylaminocarbonyl, di-C₁ -C₄ -alkylaminocarbonyl, C₁ -C₄-alkylcarbonylamino, C₁ -C₄ -alkylcarbonyl-C₁ -C₄ -amino, C₁ -C₄-alkylsulfinyl, C₁ -C₄ -alkylsulfoxyl, phenyl or phenoxy, where thephenyl rings for their part can be partially or completely halogenatedand/or can carry one to three of the following groups: cyano, nitro, C₁-C₄ -alkyl, C₃ -C₆ -cycloalkyl, C₁ -C₄ -haloalkyl, C₁ -C₄ -alkoxy, C₃-C₆ -cycloalkoxy and C₁ -C₄ -alkylthio.

In addition, compounds I are preferred in which B is unsubstituted orsubstituted heteroaryl.

Particularly preferred compounds I are those in which B is unsubstitutedor substituted pyridyl, pyridazinyl, pyrimidinyl, pyrazinyl, quinolinyl,isoquinolinyl, cinnolinyl, quinazolinyl, quinoxalinyl, pteridinyl,furyl, thienyl, pyrryl, oxazolyl, thiazolyl, imidazolyl, isoxazolyl,isothiazolyl, pyrazolyl, oxadiazolyl, thiadiazolyl, triazolyl,triazinyl, tetrazinyl, benzofuryl, thionaphthenyl, indolyl,benzoxazolyl, benzothiazolyl, benzimidazolyl, benzisoxazolyl,benzoisothiazolyl, benzopyrazolyl or purinyl.

In particular, compounds I are preferred in which B is heteroaryl whichcan be partially halogenated and/or can carry one to three (preferablyone or two) of the following radicals: nitro, cyanomethyl, C₁ -C₄-alkyl, C₃ -C₆ -cycloalkyl, C₁ -C₄ -haloalkyl, C₁ -C₄ -alkoxy, C₃ -C₆-cycloalkoxy, C₁ -C₄ -haloalkoxy, phenyl or phenoxy, where the phenylrings for their part can be partially or completely halogenated and/orcan carry one to three of the following groups: cyano, nitro, C₁ -C₄-alkyl, C₃ -C₆ -cycloalkyl, C₁ -C₄ -haloalkyl, C₁ -C₄ -alkoxy, C₃ -C₆-cycloalkoxy and C₁ -C₄ -alkylthio.

Additionally, compounds I are preferred in which B is a group -CO-W,where W is hydrogen, C₁ -C₁₂ -alkyl, C₁ -C₆ -alkoxy, C₃ -C₇ -cycloalkyl,phenyl, benzyl, phenoxy, benzyloxy, pyridyl, furyl, thiazolyl orquinolinyl.

In addition, compounds I are preferred in which A and B, together withthe C atom to which they are bonded, are one of the following groups: C₅-C₆ -cycloalkyl, C₅ -C₆ -cycloalkenyl, tetrahydronaphthyl ortetrahydrobenzopyranyl.

Particularly preferred compounds of the formula I are compiled in thefollowing tables 1 to 16.

Table 1

Compounds of the general formula I.1 in which Y is methoxy and Z isCHCH₃ and the combination of the substituents A, R and Q_(m) for acompound in each case corresponds to one line of Table A ##STR8##

Table 2

Compounds of the general formula I.1 in which Y is methoxy and Z isCHOCH₃ and the combination of the substituents A, R and Q_(m) for acompound in each case corresponds to one line of Table A.

Table 3

Compounds of the general formula I.1 in which Y is methoxy and Z isNOCH₃ and the combination of the substituents A, R and Q_(m) for acompound in each case corresponds to one line of Table A.

Table 4

Compounds of the general formula I.1 in which Y is methylamino and Z isCHCH₃ and the combination of the substituents A, R and Q_(m) for acompound in each case corresponds to one line of Table A.

Table 5

Compounds of the general formula I.1 in which Y is methylamino and Z isCHOCH₃ and the combination of the substituents A, R and Q_(m) for acompound in each case corresponds to one line of Table A.

Table 6

Compounds of the general formula I.1 in which Y is methylamino and Z isNOCH₃ and the combination of the substituents A, R and Q_(m) for acompound in each case corresponds to one line of Table A.

Table 7

Compounds of the general formula I.1 in which Y is amino and Z is CHOCH₃and the combination of the substituents A, R and Q_(m) for a compound ineach case corresponds to one line of Table A.

Table 8

Compounds of the general formula I.1 in which Y is dimethylamino and Zis CHOCH₃ and the combination of the substituents A, R and Q_(m) for acompound in each case corresponds to one line of Table A.

Table 9

Compounds of the general formula I.2 in which Y is methoxy and Z isCHCH₃ and the combination of the substituents A, B and R for a compoundin each case corresponds to one line of Table B ##STR9##

Table 10

Compounds of the general formula I.2 in which Y is methoxy and Z isCHOCH₃ and the combination of the substituents A, B and R for a compoundin each case corresponds to one line of Table B.

Table 11

Compounds of the general formula I.2 in which Y is methoxy and Z isNOCH₃ and the combination of the substituents A, B and R for a compoundin each case corresponds to one line of Table B.

Table 12

Compounds of the general formula I.2 in which Y is methylamino and Z isCHCH₃ and the combination of the substituents A, B and R for a compoundin each case corresponds to one line of Table B.

Table 13

Compounds of the general formula I.2 in which Y is methylamino and Z isCHOCH₃ and the combination of the substituents A, B and R for a compoundin each case corresponds to one line of Table B.

Table 14

Compounds of the general formula I.2 in which Y is methylamino and Z isNOCH₃ and the combination of the substituents A, B and R for a compoundin each case corresponds to one line of Table B.

Table 15

Compounds of the general formula I.2 in which Y is amino and Z is CHOCH₃and the combination of the substituents A, B and R for a compound ineach case corresponds to one line of Table B.

Table 16

Compounds of the general formula I.2 in which Y is dimethylamino and Zis CHOCH₃ and the combination of the substituents A, B and R for acompound in each case corresponds to one line of Table B.

                  TABLE A                                                         ______________________________________                                        R         A           Q.sub.m                                                 ______________________________________                                        H         H           H                                                       H         H           2-F                                                     H         H           3-F                                                     H         H           4-F                                                     H         H           2,3-F.sub.2                                             H         H           2,4-F.sub.2                                             H         H           2,5-F.sub.2                                             H         H           2,6-F.sub.2                                             H         H           3,4-F.sub.2                                             H         H           3,5-F.sub.2                                             H         H           2-Cl                                                    H         H           3-Cl                                                    H         H           4-Cl                                                    H         H           2,4-Cl.sub.2                                            H         H           2,5-Cl.sub.2                                            H         H           3,4-Cl.sub.2                                            H         H           3,5-Cl.sub.2                                            H         H           2-Br                                                    H         H           3-Br                                                    H         H           4-Br                                                    H         H           2,4-Br.sub.2                                            H         H           3,4-Br.sub.2                                            H         H           3,5-Br.sub.2                                            H         H           2-I                                                     H         H           3-I                                                     H         H           4-I                                                     H         H           2-F, 4-Cl                                               H         H           2-F, 5-Cl                                               H         H           2-F, 4-Br                                               H         H           2-F, 5-Br                                               H         H           2-Cl, 4-Br                                              H         H           2-Cl, 5-Br                                              H         H           3-F, 4-Cl                                               H         H           3-F, 5-Cl                                               H         H           3-F, 4-Br                                               H         H           3-F, 5-Br                                               H         H           3-Cl, 4-Br                                              H         H           3-Cl, 5-Br                                              H         H           3-Cl, 4-F                                               H         H           3-Br, 4-F                                               H         H           3-Br, 4-Cl                                              H         H           2-NO.sub.2                                              H         H           3-NO.sub.2                                              H         H           4-NO.sub.2                                              H         H           2-CN                                                    H         H           3-CN                                                    H         H           4-CN                                                    H         H           2-CH.sub.3                                              H         H           3-CH.sub.3                                              H         H           4-CH.sub.3                                              H         H           2,3-(CH.sub.3).sub.2                                    H         H           2,4-(CH.sub.3).sub.2                                    H         H           2,5-(CH.sub.3).sub.2                                    H         H           2,6-(CH.sub.3).sub.2                                    H         R           3,4-(CH.sub.3).sub.2                                    H         H           3,5-(CH.sub.3).sub.2                                    H         H           2,4,5-(CH.sub.3).sub.3                                  H         H           2,4,6-(CH.sub.3).sub.3                                  H         H           3,4,5-(CH.sub.3).sub.3                                  H         H           2-C.sub.2 H.sub.5                                       H         H           3-C.sub.2 H.sub.5                                       H         H           4-C.sub.2 H.sub.5                                       H         H           3,4-(C.sub.2 H.sub.5).sub.2                             H         H           3,5-(C.sub.2 H.sub.5).sub.2                             H         H           3-n-C.sub.3 H.sub.7                                     H         H           4-n-C.sub.3 H.sub.7                                     H         H           3,4-(n-C.sub.3 H.sub.7).sub.2                           H         H           3,5-(n-C.sub.3 H.sub.7).sub.2                           H         H           3-i-C.sub.3 H.sub.7                                     H         H           4-i-C.sub.3 H.sub.7                                     H         H           3,4-(i-C.sub.3 H.sub.7).sub.2                           H         H           3,5-(i-C.sub.3 H.sub.7).sub.2                           H         H           3-Cyclopropyl                                           H         H           4-Cyclopropyl                                           H         H           3-n-C.sub.4 H.sub.9                                     H         H           4-n-C.sub.4 H.sub.9                                     H         H           3,4-(n-C.sub.4 H.sub.9).sub.2                           H         H           3,5-(n-C.sub.4 H.sub.9).sub.2                           H         H           3-s-C.sub.4 H.sub.9                                     H         H           4-s-C.sub.4 H.sub.9                                     H         H           3-i-C.sub.4 H.sub.9                                     H         H           4-i-C.sub.4 H.sub.9                                     H         H           3-t-C.sub.4 H.sub.9                                     H         H           4-t-C.sub.4 H.sub.9                                     H         H           3,4-(t-C.sub.4 H.sub.9).sub.2                           H         H           3,5-(t-C.sub.4 H.sub.9).sub.2                           H         H           3-n-C.sub.5 H.sub.11                                    H         H           4-n-C.sub.5 H.sub.11                                    H         H           3-n-C.sub.6 H.sub.13                                    H         H           4-n-C.sub.6 H.sub.13                                    H         H           3-Cyclohexyl                                            H         H           4-Cyclohexyl                                            H         H           3-Phenyl                                                H         H           4-Phenyl                                                H         H           3-Vinyl                                                 H         H           4-Vinyl                                                 H         H           3-Allyl                                                 H         H           4-Allyl                                                 H         H           3-Propargyl                                             H         H           4-Propargyl                                             H         H           3-(Propen-2-yl)                                         H         H           4-(Propen-2-yl)                                         H         H           2-CH.sub.3, 4-C.sub.2 H.sub.5                           H         H           2-CH.sub.3, 5-C.sub.2 H.sub.5                           H         H           2-CH.sub.3 --, 4-n-C.sub.3 H.sub.7                      H         H           2-CH.sub.3, 5-n-C.sub.3 H.sub.7                         H         H           2-CH.sub.3, 4-i-C.sub.3 H.sub.7                         H         H           2-CH.sub.3, 5-i-C.sub.3 H.sub.7                         H         H           2-CH.sub.3, 4-n-C.sub.4 H.sub.9                         H         H           2-CH.sub.3, 4-s-C.sub.4 H.sub.9                         H         H           2-CH.sub.3, 4-i-C.sub.4 H.sub.9                         H         H           2-CH.sub.3, 4-t-C.sub.4 H.sub.9                         H         H           2-CH.sub.3, 4-phenyl                                    H         H           2-CH.sub.3, 5-phenyl                                    H         H           2-CH.sub.3, 4-vinyl                                     H         H           2-CH.sub.3, 4-allyl                                     H         H           2-CH.sub.3, 4-propargyl                                 H         H           2-CH.sub.3, 4-(propen-2-yl)                             H         H           3-CH.sub.3, 4-C.sub.2 H.sub.5                           H         H           3-CH.sub.3, 5-C.sub.2 H.sub.5                           H         H           3-CH.sub.3, 4-n-C.sub.3 H.sub.7                         H         H           3-CH.sub.3, 5-n-C.sub.3 H.sub.7                         H         H           3-CH.sub.3, 4-i-C.sub.3 H.sub.7                         H         H           3-CH.sub.3, 5-i-C.sub.3 H.sub.7                         H         H           3-CH.sub.3, 4-cyclopropyl                               H         H           3-CH.sub.3, 4-t-C.sub.4 H.sub.9                         H         H           3-CH.sub.3, 5-t-C.sub.4 H.sub.9                         H         H           3-CH.sub.3, 4-phenyl                                    H         H           3-CH.sub.3, 5-phenyl                                    H         H           3-CH.sub.3, 4-vinyl                                     H         H           3-CH.sub.3, 4-allyl                                     H         H           3-CH.sub.3, 4-propargyl                                 H         H           3-CH.sub.3, 4-propen-2-yl                               H         H           3-C.sub.2 H.sub.5, 4-CH.sub.3                           H         H           3-i-C.sub.3 H.sub.7, 4-CH.sub.3                         H         H           3-t-C.sub.4 H.sub.9, 4-CH.sub.3                         H         H           3-Phenyl, 4-CH.sub.3                                    H         H           2-OH                                                    H         H           3-OH                                                    H         H           4-OH                                                    H         H           2-OCH.sub.3                                             H         H           3-OCH.sub.3                                             H         H           4-OCH.sub.3                                             H         H           2,3-(OCH.sub.3).sub.2                                   H         H           2,4-(OCH.sub.3).sub.2                                   H         H           2,5-(OCH.sub.3).sub.2                                   H         H           3,4-(OCH.sub.3).sub.2                                   H         H           3,5-(OCH.sub.3).sub.2                                   H         H           3,4,5-(OCH.sub.3).sub.3                                 H         H           3-OC.sub.2 H.sub.5                                      H         H           4-OC.sub.2 H.sub.5                                      H         H           3,4-(OC.sub.2 H.sub.5).sub.2                            H         H           3,5-(OC.sub.2 H.sub.5).sub.2                            H         H           3-O-n-C.sub.3 H.sub.7                                   H         H           4-O-n-C.sub.3 H.sub.7                                   H         H           3-O-i-C.sub.3 H.sub.7                                   H         H           4-O-i-C.sub.3 H.sub.7                                   H         H           3-O-Cyclopropyl                                         H         H           4-O-Cyclopropyl                                         H         H           3-O-n-C.sub.4 H.sub.9                                   H         H           4-O-n-C.sub.4 H.sub.9                                   H         H           3-O-s-C.sub.4 H.sub.9                                   H         H           4-O-s-C.sub.4 H.sub.9                                   H         H           3-O-i-C.sub.4 H.sub.9                                   H         H           4-O-i-C.sub.4 H.sub.9                                   H         H           3-O-t-C.sub.4 H.sub.9                                   H         H           4-O-t-C.sub.4 H.sub.9                                   H         H           3-O-n-C.sub.5 H.sub.11                                  H         H           4-O-n-C.sub.5 H.sub.11                                  H         H           3-O-n-C.sub.6 H.sub.13                                  H         H           4-O-n-C.sub.6 H.sub.13                                  H         H           3-O-Cyclohexyl                                          H         H           4-O-Cyclohexyl                                          H         H           3-O-Phenyl                                              H         H           4-O-Phenyl                                              H         H           3-O-Allyl                                               H         H           4-O-Allyl                                               H         H           2-CF.sub.3                                              H         H           3-CF.sub.3                                              H         H           4-CF.sub.3                                              H         H           2,4-(CF.sub.3).sub.2                                    H         H           3,5-(CF.sub.3).sub.2                                    H         H           3-CF.sub.2 Cl                                           H         H           4-CF.sub.2 Cl                                           H         H           3-CFCl.sub.2                                            H         H           4-CFCl.sub.2                                            H         H           3-CCl.sub.3                                             H         H           4-CCl.sub.3                                             H         H           3-CH.sub.2 CH.sub.2 F                                   H         H           4-CH.sub.2 CH.sub.2 F                                   H         H           3-CH.sub.2 CF.sub.3                                     H         H           4-CH.sub.2 CF.sub.3                                     H         H           3-C.sub.2 F.sub.5                                       H         H           4-C.sub.2 F.sub.5                                       H         H           3-CHCl.sub.2                                            H         H           4-CHCl.sub.2                                            H         H           3-CH.sub.2 Cl                                           H         H           4-CH.sub.2 Cl                                           H         H           3-CF.sub.2 CHF.sub.2                                    H         H           4-CF.sub.2 CHF.sub.2                                    H         H           3-CF.sub.2 CH.sub.2 Cl                                  H         H           4-CF.sub.2 CH.sub.2 Cl                                  H         H           2-OCF.sub.3                                             H         H           3-OCF.sub.3                                             H         H           4-OCF.sub.3                                             H         H           3-OCHF.sub.2                                            H         H           4-OCHF.sub.2                                            H         H           3-OC.sub.2 F.sub.5                                      H         H           4-OC.sub.2 F.sub.5                                      H         H           3-OCF.sub.2 CHF.sub.2                                   H         H           4-OCF.sub.2 CHF.sub.2                                   H         H           3-CH.sub.2 OCH.sub.3                                    H         H           4-CH.sub.2 OCH.sub.3                                    H         H           3-CH.sub.2 O-t-C.sub.4 H.sub.9                          H         H           4-CH.sub.2 O-t-C.sub.4 H.sub.9                          H         H           3-C(CH.sub.3)(OCH.sub.3).sub.2                          H         H           4-C(CH.sub.3)(OCH.sub.3).sub.2                          H         H           3-CH(OCH.sub.3).sub.2                                   H         H           4-CH(OCH.sub.3).sub.2                                   H         H           3-CH.sub.2 CN                                           H         H           4-CH.sub.2 CN                                           H         H           3-CHO                                                   H         H           4-CHO                                                   H         H           3-CO--CH.sub.3                                          H         H           4-CO--CH.sub.3                                          H         H           3-CO--C.sub.2 H.sub.5                                   H         H           4-CO--C.sub.2 H.sub.5                                   H         H           2-COOH                                                  H         H           3-COOH                                                  H         H           4-COOH                                                  H         H           3-COOCH.sub.3                                           H         H           4-COOCH.sub.3                                           H         H           3-COOC.sub.2 H.sub.5                                    H         H           4-COOC.sub.2 H.sub.5                                    H         H           3-COO-n-C.sub.3 H.sub.7                                 H         H           4-COO-n-C.sub.3 H.sub.7                                 H         H           3-COO-i-C.sub.3 H.sub.7                                 H         H           4-COO-i-C.sub.3 H.sub.7                                 H         H           3-COO-n-C.sub.4 H.sub.9                                 H         H           4-COO-n-C.sub.4 H.sub.9                                 H         H           3-COO-s-C.sub.4 H.sub.9                                 H         H           4-COO-s-C.sub.4 H.sub.9                                 H         H           3-COO-i-C.sub.4 H.sub.9                                 H         H           4-COO-i-C.sub.4 H.sub.9                                 H         H           3-COO-t-C.sub.4 H.sub.9                                 H         H           4-COO-t-C.sub.4 H.sub.9                                 H         H           3-COO-n-C.sub.5 H.sub.11                                H         H           4-COO-n-C.sub.5 H.sub.11                                H         H           3-COO-n-C.sub.6 H.sub.13                                H         H           4-COO-n-C.sub.6 H.sub.13                                H         H           2-CONH.sub.2                                            H         H           3-CONH.sub.2                                            H         H           4-CONH.sub.2                                            H         H           3-CONHCH.sub.3                                          H         H           4-CONHCH.sub.3                                          H         H           3-CON(CH.sub.3).sub.2                                   H         H           4-CON(CH.sub.3).sub.2                                   H         H           3-CON(C.sub.2 H.sub.5).sub.2                            H         H           4-CON(C.sub.2 H.sub.5).sub.2                            H         H           2-CSNH.sub.2                                            H         H           3-CSNH.sub.2                                            H         H           4-CSNH.sub.2                                            H         H           2-NH.sub.2                                              H         H           3-NH.sub.2                                              H         H           4-NH.sub.2                                              H         H           3-NHCH.sub.3                                            H         H           4-NHCH.sub.3                                            H         H           3-N(CH.sub.3).sub.2                                     H         H           4-N(CH.sub.3).sub.2                                     H         H           3-NHCO--CH.sub.3                                        H         H           4-NHCO--CH.sub.3                                        H         H           3-NCH.sub.3 --CO--CH.sub.3                              H         H           4-NCH.sub.3 --CO--CH.sub.3                              H         H           3-NHCOOCH.sub.3                                         H         H           4-NHCOOCH.sub.3                                         H         H           3-NCH.sub.3 --COOCH.sub.3                               H         H           4-NCH.sub.3 --COOCH.sub.3                               H         H           3-OCO--CH.sub.3                                         H         H           4-OCO--CH.sub.3                                         H         H           3-OCO-t-C.sub.4 H.sub.9                                 H         H           4-OCO-t-C.sub.4 H.sub.9                                 H         H           3-SH                                                    H         H           4-SH                                                    H         H           3-SCH.sub.3                                             H         H           4-SCH.sub.3                                             H         H           3-S-t-C.sub.4 H.sub.9                                   H         H           4-S-t-C.sub.4 H.sub.9                                   H         H           3-SO--CH.sub.3                                          H         H           4-SO--CH.sub.3                                          H         H           3-SO.sub.2 CH.sub.3                                     H         H           4-SO.sub.2 CH.sub.3                                     H         H           3-CH═NCH.sub.3                                      H         H           4-CH═NCH.sub.3                                      H         H           3-C(CH.sub.3)═NCH.sub.3                             H         H           4-C(CH.sub.3)═NCH.sub.3                             H         H           3-C(SCH.sub.3)═NOCH.sub.3                           H         H           4-C(SCH.sub.3)═NOCH.sub.3                           H         H           3-C(OCH.sub.3)═NOCH.sub.3                           H         H           4-C(OCH.sub.3)═NOCH.sub.3                           H         H           3-C(NH.sub.2)═NOCH.sub.3                            H         H           4-C(NH.sub.2)═NOCH.sub.3                            H         H           3-C(NHCH.sub.3)═NOCH.sub.3                          H         H           4-C(NHCH.sub.3)═NOCH.sub.3                          H         H           3-CH═NOCH.sub.3                                     H         H           4-CH═NOCH.sub.3                                     H         H           3-C(CH.sub.3)═NOCH.sub.3                            H         H           4-C(CH.sub.3)═NOCH.sub.3                            H         H           3-C(CH.sub.3)═NOC.sub.2 H.sub.5                     H         H           4-C(CH.sub.3)═NOC.sub.2 H.sub.5                     H         H           3-C(CH.sub.3)═NO-n-C.sub.3 H.sub.7                  H         H           4-C(CH.sub.3)═NO-n-C.sub.3 H.sub.7                  H         H           3-C(CH.sub.3)═NO-i-C.sub.3 H.sub.7                  H         H           4-C(CH.sub.3)═NO-i-C.sub.3 H.sub.7                  H         H           3-C(CH.sub.3)═NO-n-C.sub.4 H.sub.9                  H         H           4-C(CH.sub.3)═NO-n-C.sub.4 H.sub.9                  H         H           3-C(CH.sub.3)═NO-s-C.sub.4 H.sub.9                  H         H           4-C(CH.sub.3)═NO-s-C.sub.4 H.sub.9                  H         H           3-C(CH.sub.3)═NO-i-C.sub.4 H.sub.9                  H         H           4-C(CH.sub.3)═NO-i-C.sub.4 H.sub.9                  H         H           3-C(CH.sub.3)═NO-t-C.sub.4 H.sub.9                  H         H           4-C(CH.sub.3)═NO-t-C.sub.4 H.sub.9                  H         H           3-C(CH.sub.3)═NO-n-C.sub.5 H.sub.11                 H         H           4-C(CH.sub.3)═NO-n-C.sub.5 H.sub.11                 H         H           3-C(CH.sub.3)═NO-n-C.sub.6 H.sub.13                 H         H           4-C(CH.sub.3)═NO-n-C.sub.6 H.sub.13                 H         H           2-Cl, 4-CH.sub.3                                        H         H           2-Cl, 5-CH.sub.3                                        H         H           3-Cl, 4-CH.sub.3                                        H         H           3-Cl, 5-CH.sub.3                                        H         H           2-CH.sub.3, 4-Cl                                        H         H           2-CH.sub.3, 5-Cl                                        H         H           3-CH.sub.3, 4-Cl                                        H         H           3-Cl, 5-t-C.sub.4 H.sub.9                               H         H           2-Cl, 4-t-C.sub.4 H.sub.9                               H         H           2-F, 4-CH.sub.3                                         H         H           3-F, 4-CH.sub.3                                         H         H           3-F, 5-CH.sub.3                                         H         H           2-CH.sub.3, 4-F                                         H         H           3-CH.sub.3, 4-F                                         H         H           2-F, 4-t-C.sub.4 H.sub.9                                H         H           3-F, 4-t-C.sub.4 H.sub.9                                H         H           2-F, 4-OCH.sub.3                                        H         H           2-Br, 4-CH.sub.3                                        H         H           3-Br, 4-CH.sub.3                                        H         H           3-Br, 5-CH.sub.3                                        H         H           2-CH.sub.3, 4-Br                                        H         H           3-CH.sub.3, 4-Br                                        H         H           2-Br, 4-t-C.sub.4 H.sub.9                               H         H           2-Cl, 4-NO.sub.2                                        H         H           3-Cl, 4-NO.sub.2                                        H         H           3-Cl, 5-NO.sub.2                                        H         H           3-NO.sub.2, 4-Cl                                        H         H           3-Cl, 4-OCH                                             H         H           3-OCH.sub.3, 4-Cl                                       H         H           2-Cl, 5-CF.sub.3                                        H         H           3-Cl, 4-CF.sub.3                                        H         H           3-Cl, 5-CF.sub.3                                        H         H           3-CF.sub.3, 4-Cl                                        H         H           3-Cl, 5-OCF.sub.3                                       H         H           3-F, 5-CF.sub.3                                         H         H           2-CH.sub.3, 4-CN                                        H         H           3-NO.sub.2, 4-CH.sub.3                                  H         H           2-CH.sub.3, 4-OCH.sub.3                                 H         H           3-CH.sub.3, 4-OCH.sub.3                                 H         H           3-CH.sub.3, 5-OCH.sub.3                                 H         H           3-OCH.sub.3, 4-CH.sub.3                                 H         H           2-CH.sub.3, 4-O-i-C.sub.3 H.sub.7                       H         H           3-CH.sub.3, 4-O-i-C.sub.3 H.sub.7                       H         H           3-O-i-C.sub.3 H.sub.7, 4-CH.sub.3                       H         H           2-CH.sub.3, 4-CF.sub.3                                  H         H           2-CH.sub.3, 5-CF.sub.3                                  H         H           3-CH.sub.3, 4-CF.sub.3                                  H         H           3-CH.sub.3, 5-CF.sub.3                                  H         H           3-CF.sub.3, 4-CH.sub.3                                  H         H           3-CF.sub.3, 4-OCH.sub.3                                 H         H           3-OCH.sub.3, 4-CF.sub.3                                 H         H           2-CH.sub.3, 4-C(CH.sub.3)═NOCH.sub.3                H         H           3-CH.sub.3, 4-C(CH.sub.3)═NOCH.sub.3                H         H           2-OH, 5-CH.sub.3                                        H         H           3-CH.sub.3, 4-OC.sub.2 H.sub.5                          H         H           3-CH.sub.3, 4-O-t-C.sub.4 H.sub.9                       H         H           3-OC.sub.2 H.sub.5, 4-CH.sub.3                          H         H           3-O-t-C.sub.4 H.sub.9, 4-CH.sub.3                       H         H           2-C(COOCH.sub.3)═NOCH.sub.3                         H         H           2,3-Butadienyl                                          H         H           3,4-Butadienyl                                          CH.sub.3  H           H                                                       CH.sub.3  H           2-F                                                     CH.sub.3  H           3-F                                                     CH.sub.3  H           4-F                                                     CH.sub.3  H           2,4-F.sub.2                                             CH.sub.3  H           3,4-F.sub.2                                             CH.sub.3  H           3,5-F.sub.2                                             CH.sub.3  H           2-Cl                                                    CH.sub.3  H           3-Cl                                                    CH.sub.3  H           4-Cl                                                    CH.sub.3  H           2,4-Cl.sub.2                                            CH.sub.3  H           3,4-Cl.sub.2                                            CH.sub.3  H           3,5-Cl.sub.2                                            CH.sub.3  H           2-Br                                                    CH.sub.3  H           3-Br                                                    CH.sub.3  H           4-Br                                                    CH.sub.3  H           3,5-Br.sub.2                                            CH.sub.3  H           3-I                                                     CH.sub.3  H           4-I                                                     CH.sub.3  H           3-F, 5-Cl                                               CH.sub.3  H           3-F, 5-Br                                               CH.sub.3  H           3-Cl, 5-Br                                              CH.sub.3  H           3-Br, 4-F                                               CH.sub.3  H           2-NO.sub.2                                              CH.sub.3  H           3-NO.sub.2                                              CH.sub.3  H           4-NO.sub.2                                              CH.sub.3  H           2-CN                                                    CH.sub.3  H           3-CN                                                    CH.sub.3  H           4-CN                                                    CH.sub.3  H           2-CH.sub.3                                              CH.sub.3  H           3-CH.sub.3                                              CH.sub.3  H           4-CH.sub.3                                              CH.sub.3  H           2,4-(CH.sub.3).sub.2                                    CH.sub.3  H           2,5-(CH.sub.3).sub.2                                    CH.sub.3  H           3,4-(CH.sub.3).sub.2                                    CH.sub.3  H           3,5-(CH.sub.3).sub.2                                    CH.sub.3  H           2,4,5-(CH.sub.3).sub.3                                  CH.sub.3  H           2,4,6-(CH.sub.3).sub.3                                  CH.sub.3  H           3-C.sub.2 H.sub.5                                       CH.sub.3  H           4-C.sub.2 H.sub.5                                       CH.sub.3  H           3,4-(C.sub.2 H.sub.5).sub.2                             CH.sub.3  H           3,5-(C.sub.2 H.sub.5).sub.2                             CH.sub.3  H           3-n-C.sub.3 H.sub.7                                     CH.sub.3  H           4-n-C.sub.3 H.sub.7                                     CH.sub.3  H           3-i-C.sub.3 H.sub.7                                     CH.sub.3  H           4-i-C.sub.3 H.sub.7                                     CH.sub.3  H           3-Cyclopropyl                                           CH.sub.3  H           4-Cyclopropyl                                           CH.sub.3  H           3-n-C.sub.4 H.sub.9                                     CH.sub.3  H           4-n-C.sub.4 H.sub.9                                     CH.sub.3  H           3-t-C.sub.4 H.sub.9                                     CH.sub.3  H           4-t-C.sub.4 H.sub.9                                     CH.sub.3  H           3-n-C.sub.6 H.sub.13                                    CH.sub.3  H           4-n-C.sub.6 H.sub.13                                    CH.sub.3  H           3-Cyclohexyl                                            CH.sub.3  H           4-Cyclohexyl                                            CH.sub.3  H           3-Phenyl                                                CH.sub.3  H           4-Phenyl                                                CH.sub.3  H           4-Allyl                                                 CH.sub.3  H           4-Propargyl                                             CH.sub.3  H           2-CH.sub.3, 4-C.sub.2 H.sub.5                           CH.sub.3  H           2-CH.sub.3, 4-i-C.sub.3 H.sub.7                         CH.sub.3  H           2-CH.sub.3, 4-t-C.sub.4 H.sub.9                         CH.sub.3  H           2-CH.sub.3, 4-phenyl                                    CH.sub.3  H           3-CH.sub.3, 4-phenyl                                    CH.sub.3  H           3-OH                                                    CH.sub.3  H           4-OH                                                    CH.sub.3  H           3-OCH.sub.3                                             CH.sub.3  H           4-OCH.sub.3                                             CH.sub.3  H           3,4-(OCH.sub.3).sub.2                                   CH.sub.3  H           3,5-(OCH.sub.3).sub.2                                   CH.sub.3  H           3,4,5-(OCH.sub.3).sub.3                                 CH.sub.3  H           4-OC.sub.2 H.sub.5                                      CH.sub.3  H           4-O-i-C.sub.3 H.sub.7                                   CH.sub.3  H           3-O-t-C.sub.4 H.sub.9                                   CH.sub.3  H           4-O-t-C.sub.4 H.sub.9                                   CH.sub.3  H           4-O-n-C.sub.6 H.sub.13                                  CH.sub.3  H           3-O-Phenyl                                              CH.sub.3  H           4-O-Phenyl                                              CH.sub.3  H           4-O-Allyl                                               CH.sub.3  H           2-CF.sub.3                                              CH.sub.3  H           3-CF.sub.3                                              CH.sub.3  H           4-CF.sub.3                                              CH.sub.3  H           3,5-(CF.sub.3).sub.2                                    CH.sub.3  H           4-CH.sub.2 CF.sub.3                                     CH.sub.3  H           4-C.sub.2 F.sub.5                                       CH.sub.3  H           4-CF.sub.2 CHF.sub.2                                    CH.sub.3  H           3-OCF.sub.3                                             CH.sub.3  H           4-OCF.sub.3                                             CH.sub.3  H           4-OCH.sub.2 CF.sub.3                                    CH.sub.3  H           4-OC.sub.2 F.sub.5                                      CH.sub.3  H           4-OCF.sub.2 CHF.sub.2                                   CH.sub.3  H           3-CH.sub.2 OCH.sub.3                                    CH.sub.3  H           4-CH.sub.2 OCH.sub.3                                    CH.sub.3  H           4-CH.sub.2 --O-t-C.sub.4 H.sub.9                        CH.sub.3  H           4-CH(OCH.sub.3).sub.2                                   CH.sub.3  H           4-CH.sub.2 CN                                           CH.sub.3  H           3-CHO                                                   CH.sub.3  H           4-CHO                                                   CH.sub.3  H           3-CO--CH.sub.3                                          CH.sub.3  H           4-CO--CH.sub.3                                          CH.sub.3  H           3-COOH                                                  CH.sub.3  H           4-COOH                                                  CH.sub.3  H           3-COOCH.sub.3                                           CH.sub.3  H           4-COOCH.sub.3                                           CH.sub.3  H           3-COOC.sub.2 H.sub.5                                    CH.sub.3  H           4-COOC.sub.2 H.sub.5                                    CH.sub.3  H           3-COO-i-C.sub.3 H.sub.7                                 CH.sub.3  H           4-COO-i-C.sub.3 H.sub.7                                 CH.sub.3  H           3-COO-t-C.sub.4 H.sub.9                                 CH.sub.3  H           4-COO-t-C.sub.4 H.sub.9                                 CH.sub.3  H           3-COO-n-C.sub.6 H.sub.13                                CH.sub.3  H           4-COO-n-C.sub.6 H.sub.13                                CH.sub.3  H           3-CONH.sub.2                                            CH.sub.3  H           4-CONH.sub.2                                            CH.sub.3  H           3-CONHCH.sub.3                                          CH.sub.3  H           4-CONHCH.sub.3                                          CH.sub.3  H           3-CON(CH.sub.3).sub.2                                   CH.sub.3  H           4-CON(CH.sub.3).sub.2                                   CH.sub.3  H           3-CSNH.sub.2                                            CH.sub.3  H           4-CSNH.sub.2                                            CH.sub.3  H           3-NH.sub.2                                              CH.sub.3  H           4-NH.sub.2                                              CH.sub.3  H           4-NHCH.sub.3                                            CH.sub.3  H           4-N(CH.sub.3).sub.2                                     CH.sub.3  H           3-NHCO--CH.sub.3                                        CH.sub.3  H           4-NHCO--CH.sub.3                                        CH.sub.3  H           4-NCH.sub.3 --CO--CH.sub.3                              CH.sub.3  H           4-NHCOOCH.sub.3                                         CH.sub.3  H           4-NCH.sub.3 --COOCH.sub.3                               CH.sub.3  H           3-OCO--CH.sub.3                                         CH.sub.3  H           4-OCO--CH.sub.3                                         CH.sub.3  H           4-OCO-t-C.sub.4 H.sub.9                                 CH.sub.3  H           4-SH                                                    CH.sub.3  H           4-SCH.sub.3                                             CH.sub.3  H           4-S-t-C.sub.4 H.sub.9                                   CH.sub.3  H           4-SO--CH.sub.3                                          CH.sub.3  H           4-SO.sub.2 --CH.sub.3                                   CH.sub.3  H           4-C(CH.sub.3)═NCH.sub.3                             CH.sub.3  H           4-C(SCH.sub.3)═NOCH.sub.3                           CH.sub.3  H           4-C(OCH.sub.3)═NOCH.sub.3                           CH.sub.3  H           3-CH═NOCH.sub.3                                     CH.sub.3  H           4-CH═NOCH.sub.3                                     CH.sub.3  H           3-C(CH.sub.3)═NOCH.sub.3                            CH.sub.3  H           4-C(CH.sub.3)═NOCH.sub.3                            CH.sub.3  H           4-C(CH.sub.3)═NOC.sub.2 H.sub.5                     CH.sub.3  H           4-C(CH.sub.3)═NO-n-C.sub.3 H.sub.7                  CH.sub.3  H           4-C(CH.sub.3)═NO-i-C.sub.3 H.sub.7                  CH.sub.3  H           4-C(CH.sub.3)═NO-n-C.sub.4 H.sub.9                  CH.sub.3  H           4-C(CH.sub.3)═NO-t-C.sub.4 H.sub.9                  CH.sub.3  H           4-C(CH.sub.3)═NO-n-C.sub.5 H.sub.11                 CH.sub.3  H           4-C(CH.sub.3)═NO-n-C.sub.6 H.sub.13                 CH.sub.3  H           2-Cl, 4-CH.sub.3                                        CH.sub.3  H           3-Cl, 5-CH.sub.3                                        CH.sub.3  H           2-CH.sub.3, 4-Cl                                        CH.sub.3  H           3-CH.sub.3, 4-Cl                                        CH.sub.3  H           3-F, 5-CH.sub.3                                         CH.sub.3  H           3-Br, 5-CH.sub.3                                        CH.sub.3  H           3-Cl, 5-NO.sub.2                                        CH.sub.3  H           3-NO.sub.2, 4-Cl                                        CH.sub.3  H           3-Cl, 4-OCH.sub.3                                       CH.sub.3  H           3-OCH.sub.3, 4-Cl                                       CH.sub.3  H           3-Cl, 5-CF.sub.3                                        CH.sub.3  H           3-Cl, 5-OCF.sub.3                                       CH.sub.3  H           3-F, 5-CF.sub.3                                         CH.sub.3  H           2-CH.sub.3, 4-CN                                        CH.sub.3  H           2-CH.sub.3, 4-OCH.sub.3                                 CH.sub.3  H           2-CH.sub.3, 4-CF.sub.3                                  CH.sub.3  H           2-CH.sub.3, 4-C(CH.sub.3)═NOCH.sub.3                CH.sub.3  H           3-CH.sub.3, 4-C(CH.sub.3)═NOCH.sub.3                CH.sub.3  H           2-OH, 5-CH.sub.3                                        CH.sub.3  H           3-CH.sub.3, 4-O-t-C.sub.4 H.sub.9                       CH.sub.3  H           2-C(COOCH.sub.3)═NOCH.sub.3                         CH.sub.3  H           2,3-Butadienyl                                          CH.sub.3  H           3,4-Butadienyl                                          H         CH.sub.3    H                                                       H         CH.sub.3    2-F                                                     H         CH.sub.3    3-F                                                     H         CH.sub.3    4-F                                                     H         CH.sub.3    2,3-F.sub.2                                             H         CH.sub.3    2,4-F.sub.2                                             H         CH.sub.3    2,5-F.sub.2                                             H         CH.sub.3    2,6-F.sub.2                                             H         CH.sub.3    3,4-F.sub.2                                             H         CH.sub.3    3,5-F.sub.2                                             H         CH.sub.3    2-Cl                                                    H         CH.sub.3    3-Cl                                                    H         CH.sub.3    4-Cl                                                    H         CH.sub.3    2,4-Cl.sub.2                                            H         CH.sub.3    2,5-Cl.sub.2                                            H         CH.sub.3    3,4-Cl.sub.2                                            H         CH.sub.3    3,5-Cl.sub.2                                            H         CH.sub.3    2-Br                                                    H         CH.sub.3    3-Br                                                    H         CH.sub.3    4-Br                                                    H         CH.sub.3    2,4-Br.sub.2                                            H         CH.sub.3    3,4-Br.sub.2                                            H         CH.sub.3    3,5-Br.sub.2                                            H         CH.sub.3    2-I                                                     H         CH.sub.3    3-I                                                     H         CH.sub.3    4-I                                                     H         CH.sub.3    2-F, 4-Cl                                               H         CH.sub.3    2-F, 5-Cl                                               H         CH.sub.3    2-F, 4-Br                                               H         CH.sub.3    2-F, 5-Br                                               H         CH.sub.3    2-Cl, 4-Br                                              H         CH.sub.3    2-Cl, 5-Br                                              H         CH.sub.3    3-F, 4-Cl                                               H         CH.sub.3    3-F, 5-Cl                                               H         CH.sub.3    3-F, 4-Br                                               H         CH.sub.3    3-F, 5-Br                                               H         CH.sub.3    3-Cl, 4-Br                                              H         CH.sub.3    3-Cl, 5-Br                                              H         CH.sub.3    3-Cl, 4-F                                               H         CH.sub.3    3-Br, 4-F                                               H         CH.sub.3    3-Br, 4-Cl                                              H         CH.sub.3    2-NO.sub.2                                              H         CH.sub.3    3-NO.sub.2                                              H         CH.sub.3    4-NO.sub.2                                              H         CH.sub.3    2-CN                                                    H         CH.sub.3    3-CN                                                    H         CH.sub.3    4-CN                                                    H         CH.sub.3    2-CH.sub.3                                              H         CH.sub.3    3-CH.sub.3                                              H         CH.sub.3    4-CH.sub.3                                              H         CH.sub.3    2,3-(CH.sub.3).sub.2                                    H         CH.sub.3    2,4-(CH.sub.3).sub.2                                    H         CH.sub.3    2,5-(CH.sub.3).sub.2                                    H         CH.sub.3    2,6-(CH.sub.3).sub.2                                    H         CH.sub.3    3,4-(CH.sub.3).sub.2                                    H         CH.sub.3    3,5-(CH.sub.3).sub.2                                    H         CH.sub.3    2,4,5-(CH.sub.3).sub.3                                  H         CH.sub.3    2,4,6-(CH.sub.3).sub.3                                  H         CH.sub.3    3,4,5-(CH.sub.3).sub.3                                  H         CH.sub.3    2-C.sub.2 H.sub.5                                       H         CH.sub.3    3-C.sub.2 H.sub.5                                       H         CH.sub.3    4-C.sub.2 H.sub.5                                       H         CH.sub.3    3,4-(C.sub.2 H.sub.5).sub.2                             H         CH.sub.3    3,5-(C.sub.2 H.sub.5).sub.2                             H         CH.sub.3    3-n-C.sub.3 H.sub.7                                     H         CH.sub.3    4-n-C.sub.3 H.sub.7                                     H         CH.sub.3    3,4-(n-C.sub.3 H.sub.7).sub.2                           H         CH.sub.3    3,5-(n-C.sub.3 H.sub.7).sub.2                           H         CH.sub.3    3-i-C.sub.3 H.sub.7                                     H         CH.sub.3    4-i-C.sub.3 H.sub.7                                     H         CH.sub.3    3,4-(i-C.sub.3 H.sub.7).sub.2                           H         CH.sub.3    3,5-(i-C.sub.3 H.sub.7).sub.2                           H         CH.sub.3    3-Cyclopropyl                                           H         CH.sub.3    4-Cyclopropyl                                           H         CH.sub.3    3-n-C.sub.4 H.sub.9                                     H         CH.sub.3    4-n-C.sub.4 H.sub.9                                     H         CH.sub.3    3,4-(n-C.sub.4 H.sub.9).sub.2                           H         CH.sub.3    3,5-(n-C.sub.4 H.sub.9).sub.2                           H         CH.sub.3    3-s-C.sub.4 H.sub.9                                     H         CH.sub.3    4-s-C.sub.4 H.sub.9                                     H         CH.sub.3    3-i-C.sub.4 H.sub.9                                     H         CH.sub.3    4-i-C.sub.4 H.sub.9                                     H         CH.sub.3    3-t-C.sub.4 H.sub.9                                     H         CH.sub.3    4-t-C.sub.4 H.sub.9                                     H         CH.sub.3    3,4-(t-C.sub.4 H.sub.9).sub.2                           H         CH.sub.3    3,5-(t-C.sub.4 H.sub.9).sub.2                           H         CH.sub.3    3-n-C.sub.5 H.sub.11                                    H         CH.sub.3    4-n-C.sub.5 H.sub.11                                    H         CH.sub.3    3-n-C.sub.6 H.sub.13                                    H         CH.sub.3    4-n-C.sub.6 H.sub.13                                    H         CH.sub.3    3-Cyclohexyl                                            H         CH.sub.3    4-Cyclohexyl                                            H         CH.sub.3    3-Phenyl                                                H         CH.sub.3    4-Phenyl                                                H         CH.sub.3    3-Vinyl                                                 H         CH.sub.3    4-Vinyl                                                 H         CH.sub.3    3-Allyl                                                 H         CH.sub.3    4-Allyl                                                 H         CH.sub.3    3-Propargyl                                             H         CH.sub.3    4-Propargyl                                             H         CH.sub.3    3-(Propen-2-yl)                                         H         CH.sub.3    4-(Propen-2-yl)                                         H         CH.sub.3    2-CH.sub.3, 4-C.sub.2 H.sub.5                           H         CH.sub.3    2-CH.sub.3, 5-C.sub.2 H.sub.5                           H         CH.sub.3    2-CH.sub.3 --, 4-n-C.sub.3 H.sub.7                      H         CH.sub.3    2-CH.sub.3, 5-n-C.sub.3 H.sub.7                         H         CH.sub.3    2-CH.sub.3, 4-i-C.sub.3 H.sub.7                         H         CH.sub.3    2-CH.sub.3, 5-i-C.sub.3 H.sub.7                         H         CH.sub.3    2-CH.sub.3, 4-n-C.sub.4 H.sub.9                         H         CH.sub.3    2-CH.sub.3, 4-s-C.sub.4 H.sub.9                         H         CH.sub.3    2-CH.sub.3, 4-i-C.sub.4 H.sub.9                         H         CH.sub.3    2-CH.sub.3, 4-t-C.sub.4 H.sub.9                         H         CH.sub.3    2-CH.sub.3, 4-phenyl                                    H         CH.sub.3    2-CH.sub.3, 5-phenyl                                    H         CH.sub.3    2-CH.sub.3, 4-vinyl                                     H         CH.sub.3    2-CH.sub.3, 4-allyl                                     H         CH.sub.3    2-CH.sub.3, 4-propargyl                                 H         CH.sub.3    2-CH.sub.3, 4-(propen-2-yl)                             H         CH.sub.3    3-CH.sub.3, 4-C.sub.2 H.sub.5                           H         CH.sub.3    3-CH.sub.3, 5-C.sub.2 H.sub.5                           H         CH.sub.3    3-CH.sub.3, 4-n-C.sub.3 H.sub.7                         H         CH.sub.3    3-CH.sub.3, 5-n-C.sub.3 H.sub.7                         H         CH.sub.3    3-CH.sub.3, 4-i-C.sub.3 H.sub.7                         H         CH.sub.3    3-CH.sub.3, 5-i-C.sub.3 H.sub.7                         H         CH.sub.3    3-CH.sub.3, 4-cyclopropyl                               H         CH.sub.3    3-CH.sub.3, 4-t-C.sub.4 H.sub.9                         H         CH.sub.3    3-CH.sub.3, 5-t-C.sub.4 H.sub.9                         H         CH.sub.3    3-CH.sub.3, 4-phenyl                                    H         CH.sub.3    3-CH.sub.3, 5-phenyl                                    H         CH.sub.3    3-CH.sub.3, 4-vinyl                                     H         CH.sub.3    3-CH.sub.3, 4-allyl                                     H         CH.sub.3    3-CH.sub.3, 4-propargyl                                 H         CH.sub.3    3-CH.sub.3, 4-propen-2-yl                               H         CH.sub.3    3-C.sub.2 H.sub.5, 4-CH.sub.3                           H         CH.sub.3    3-i-C.sub.3 H.sub.7, 4-CH.sub.3                         H         CH.sub.3    3-t-C.sub.4 H.sub.9, 4-CH.sub.3                         H         CH.sub.3    3-Phenyl, 4-CH.sub.3                                    H         CH.sub.3    2-OH                                                    H         CH.sub.3    3-OH                                                    H         CH.sub.3    4-OH                                                    H         CH.sub.3    2-OCH.sub.3                                             H         CH.sub.3    3-OCH.sub.3                                             H         CH.sub.3    4-OCH.sub.3                                             H         CH.sub.3    2,3-(OCH.sub.3).sub.2                                   H         CH.sub.3    2,4-(OCH.sub.3).sub.2                                   H         CH.sub.3    2,5-(OCH.sub.3).sub.2                                   H         CH.sub.3    3,4-(OCH.sub.3).sub.2                                   H         CH.sub.3    3,5-(OCH.sub.3).sub.2                                   H         CH.sub.3    3,4,5-(OCH.sub.3).sub.3                                 H         CH.sub.3    3-OC.sub.2 H.sub.5                                      H         CH.sub.3    4-OC.sub.2 H.sub.5                                      H         CH.sub.3    3,4-(OC.sub.2 H.sub.5).sub.2                            H         CH.sub.3    3,5-(OC.sub.2 H.sub.5).sub.2                            H         CH.sub.3    3-O-n-C.sub.3 H.sub.7                                   H         CH.sub.3    4-O-n-C.sub.3 H.sub.7                                   H         CH.sub.3    3-O-i-C.sub.3 H.sub.7                                   H         CH.sub.3    4-O-i-C.sub.3 H.sub.7                                   H         CH.sub.3    3-O-Cyclopropyl                                         H         CH.sub.3    4-O-Cyclopropyl                                         H         CH.sub.3    3-O-n-C.sub.4 H.sub.9                                   H         CH.sub.3    4-O-n-C.sub.4 H.sub.9                                   H         CH.sub.3    3-O-s-C.sub.4 H.sub.9                                   H         CH.sub.3    4-O-s-C.sub.4 H.sub.9                                   H         CH.sub.3    3-O-i-C.sub.4 H.sub.9                                   H         CH.sub.3    4-O-i-C.sub.4 H.sub.9                                   H         CH.sub.3    3-O-t-C.sub.4 H.sub.9                                   H         CH.sub.3    4-O-t-C.sub.4 H.sub.9                                   H         CH.sub.3    3-O-n-C.sub.5 H.sub.11                                  H         CH.sub.3    4-O-n-C.sub.5 H.sub.11                                  H         CH.sub.3    3-O-n-C.sub.6 H.sub.13                                  H         CH.sub.3    4-O-n-C.sub.6 H.sub.13                                  H         CH.sub.3    3-O-Cyclohexyl                                          H         CH.sub.3    4-O-Cyclohexyl                                          H         CH.sub.3    3-O-Phenyl                                              H         CH.sub.3    4-O-Phenyl                                              H         CH.sub.3    3-O-Allyl                                               H         CH.sub.3    4-O-Allyl                                               H         CH.sub.3    2-CF.sub.3                                              H         CH.sub.3    3-CF.sub.3                                              H         CH.sub.3    4-CF.sub.3                                              H         CH.sub.3    2,4-(CF.sub.3).sub.2                                    H         CH.sub.3    3,5-(CF.sub.3).sub.2                                    H         CH.sub.3    3-CF.sub.2 Cl                                           H         CH.sub.3    4-CF.sub.2 Cl                                           H         CH.sub.3    3-CFCl.sub.2                                            H         CH.sub.3    4-CFCl.sub.2                                            H         CH.sub.3    3-CCl.sub.3                                             H         CH.sub.3    4-CCl.sub.3                                             H         CH.sub.3    3-CH.sub.2 CH.sub.2 F                                   H         CH.sub.3    4-CH.sub.2 CH.sub.2 F                                   H         CH.sub.3    3-CH.sub.2 CF.sub.3                                     H         CH.sub.3    4-CH.sub.2 CF.sub.3                                     H         CH.sub.3    3-C.sub.2 F.sub.5                                       H         CH.sub.3    4-C.sub.2 F.sub.5                                       H         CH.sub.3    3-CHCl.sub.2                                            H         CH.sub.3    4-CHCl.sub.2                                            H         CH.sub.3    3-CH.sub.2 Cl                                           H         CH.sub.3    4-CH.sub.2 Cl                                           H         CH.sub.3    3-CF.sub.2 CHF.sub.2                                    H         CH.sub.3    4-CF.sub.2 CHF.sub.2                                    H         CH.sub.3    3-CH.sub.2 CH.sub.2 Cl                                  H         CH.sub.3    4-CH.sub.2 CH.sub.2 Cl                                  H         CH.sub.3    2-OCF.sub.3                                             H         CH.sub.3    3-OCF.sub.3                                             H         CH.sub.3    4-OCF.sub.3                                             H         CH.sub.3    3-OCHF.sub.2                                            H         CH.sub.3    4-OCHF.sub.2                                            H         CH.sub.3    3-OC.sub.2 F.sub.5                                      H         CH.sub.3    4-OC.sub.2 F.sub.5                                      H         CH.sub.3    3-OCF.sub.2 CHF.sub.2                                   H         CH.sub.3    4-OCF.sub.2 CHF.sub.2                                   H         CH.sub.3    3-CH.sub.2 OCH.sub.3                                    H         CH.sub.3    4-CH.sub.2 OCH.sub.3                                    H         CH.sub.3    3-CH.sub.2 O-t-C.sub.4 H.sub.9                          H         CH.sub.3    4-CH.sub.2 O-t-C.sub.4 H.sub.9                          H         CH.sub.3    3-C(CH.sub.3)(OCH.sub.3).sub.2                          H         CH.sub.3    4-C(CH.sub.3)(OCH.sub.3).sub.2                          H         CH.sub.3    3-CH(OCH.sub.3).sub.2                                   H         CH.sub.3    4-CH(OCH.sub.3).sub.2                                   H         CH.sub.3    3-CH.sub.2 CN                                           H         CH.sub.3    4-CH.sub.2 CN                                           H         CH.sub.3    3-CHO                                                   H         CH.sub.3    4-CHO                                                   H         CH.sub.3    3-CO--CH.sub.3                                          H         CH.sub.3    4-CO--CH.sub.3                                          H         CH.sub.3    3-CO--C.sub.2 H.sub.5                                   H         CH.sub.3    4-CO--C.sub.2 H.sub.5                                   H         CH.sub.3    2-COOH                                                  H         CH.sub.3    3-COOH                                                  H         CH.sub.3    4-COOH                                                  H         CH.sub.3    3-COOCH.sub.3                                           H         CH.sub.3    4-COOCH.sub.3                                           H         CH.sub.3    3-COOC.sub.2 H.sub.5                                    H         CH.sub.3    4-COOC.sub.2 H.sub.5                                    H         CH.sub.3    3-COO-n-C.sub.3 H.sub.7                                 H         CH.sub.3    4-COO-n-C.sub.3 H.sub.7                                 H         CH.sub.3    3-COO-i-C.sub.3 H.sub.7                                 H         CH.sub.3    4-COO-i-C.sub.3 H.sub.7                                 H         CH.sub.3    3-COO-n-C.sub.4 H.sub.9                                 H         CH.sub.3    4-COO-n-C.sub.4 H.sub.9                                 H         CH.sub.3    3-COO-s-C.sub.4 H.sub.9                                 H         CH.sub.3    4-COO-s-C.sub.4 H.sub.9                                 H         CH.sub.3    3-COO-i-C.sub.4 H.sub.9                                 H         CH.sub.3    4-COO-i-C.sub.4 H.sub.9                                 H         CH.sub.3    3-COO-t-C.sub.4 H.sub.9                                 H         CH.sub.3    4-COO-t-C.sub.4 H.sub.9                                 H         CH.sub.3    3-COO-n-C.sub.5 H.sub.11                                H         CH.sub.3    4-COO-n-C.sub.5 H.sub.11                                H         CH.sub.3    3-COO-n-C.sub.6 H.sub.13                                H         CH.sub.3    4-COO-n-C.sub.6 H.sub.13                                H         CH.sub.3    2-CONH.sub.2                                            H         CH.sub.3    3-CONH.sub.2                                            H         CH.sub.3    4-CONH.sub.2                                            H         CH.sub.3    3-CONHCH.sub.3                                          H         CH.sub.3    4-CONHCH.sub.3                                          H         CH.sub.3    3-CON(CH.sub.3).sub.2                                   H         CH.sub.3    4-CON(CH.sub.3).sub.2                                   H         CH.sub.3    3-CON(C.sub.2 H.sub.5).sub.2                            H         CH.sub.3    4-CON(C.sub.2 H.sub.5).sub.2                            H         CH.sub.3    2-CSNH.sub.2                                            H         CH.sub.3    3-CSNH.sub.2                                            H         CH.sub.3    4-CSNH.sub.2                                            H         CH.sub.3    2-NH.sub.2                                              H         CH.sub.3    3-NH.sub.2                                              H         CH.sub.3    4-NH.sub.2                                              H         CH.sub.3    3-NHCH.sub.3                                            H         CH.sub.3    4-NHCH.sub.3                                            H         CH.sub.3    3-N(CH.sub.3).sub.2                                     H         CH.sub.3    4-N(CH.sub.3).sub.2                                     H         CH.sub.3    3-NHCO--CH.sub.3                                        H         CH.sub.3    4-NHCO--CH.sub.3                                        H         CH.sub.3    3-NCH.sub.3 --CO--CH.sub.3                              H         CH.sub.3    4-NCH.sub.3 --CO--CH.sub.3                              H         CH.sub.3    3-NHCOOCH.sub.3                                         H         CH.sub.3    4-NHCOOCH.sub.3                                         H         CH.sub.3    3-NCH.sub.3 --COOCH.sub.3                               H         CH.sub.3    4-NCH.sub.3 --COOCH.sub.3                               H         CH.sub.3    3-OCO--CH.sub.3                                         H         CH.sub.3    4-OCO--CH.sub.3                                         H         CH.sub.3    3-OCO-t-C.sub.4 H.sub.9                                 H         CH.sub.3    4-OCO-t-C.sub.4 H.sub.9                                 H         CH.sub.3    3-SH                                                    H         CH.sub.3    4-SH                                                    H         CH.sub.3    3-SCH.sub.3                                             H         CH.sub.3    4-SCH.sub.3                                             H         CH.sub.3    3-S-t-C.sub.4 H.sub.9                                   H         CH.sub.3    4-S-t-C.sub.4 H.sub.9                                   H         CH.sub.3    3-SO--CH.sub.3                                          H         CH.sub.3    4-SO--CH.sub.3                                          H         CH.sub.3    3-SO.sub.2 CH.sub.3                                     H         CH.sub.3    4-SO.sub.2 CH.sub.3                                     H         CH.sub.3    3-CH═NCH.sub.3                                      H         CH.sub.3    4-CH═NCH.sub.3                                      H         CH.sub.3    3-C(CH.sub.3)═NCH.sub.3                             H         CH.sub.3    4-C(CH.sub.3)═NCH.sub.3                             H         CH.sub.3    3-C(SCH.sub.3)═NOCH.sub.3                           H         CH.sub.3    4-C(SCH.sub.3)═NOCH.sub.3                           H         CH.sub.3    3-C(OCH.sub.3)═NOCH.sub.3                           H         CH.sub.3    4-C(OCH.sub.3)═NOCH.sub.3                           H         CH.sub.3    3-C(NH.sub.2)═NOCH.sub.3                            H         CH.sub.3    4-C(NH.sub.2)═NOCH.sub.3                            H         CH.sub.3    3-C(NHCH.sub.3)═NOCH.sub.3                          H         CH.sub.3    4-C(NHCH.sub.3)═NOCH.sub.3                          H         CH.sub.3    3-CH═NOCH.sub.3                                     H         CH.sub.3    4-CH═NOCH.sub.3                                     H         CH.sub.3    3-C(CH.sub.3)═NOCH.sub.3                            H         CH.sub.3    4-C(CH.sub.3)═NOCH.sub.3                            H         CH.sub.3    3-C(CH.sub.3)═NOC.sub.2 H.sub.5                     H         CH.sub.3    4-C(CH.sub.3)═NOC.sub.2 H.sub.5                     H         CH.sub.3    3-C(CH.sub.3)═NO-n-C.sub.3 H.sub.7                  H         CH.sub.3    4-C(CH.sub.3)═NO-n-C.sub.3 H.sub.7                  H         CH.sub.3    3-C(CH.sub.3)═NO-i-C.sub.3 H.sub.7                  H         CH.sub.3    4-C(CH.sub.3)═NO-i-C.sub.3 H.sub.7                  H         CH.sub.3    3-C(CH.sub.3)═NO-n-C.sub.4 H.sub.9                  H         CH.sub.3    4-C(CH.sub.3)═NO-n-C.sub.4 H.sub.9                  H         CH.sub.3    3-C(CH.sub.3)═NO-s-C.sub.4 H.sub.9                  H         CH.sub.3    4-C(CH.sub.3)═NO-s-C.sub.4 H.sub.9                  H         CH.sub.3    3-C(CH.sub.3)═NO-i-C.sub.4 H.sub.9                  H         CH.sub.3    4-C(CH.sub.3)═NO-i-C.sub.4 H.sub.9                  H         CH.sub.3    3-C(CH.sub.3)═NO-t-C.sub.4 H.sub.9                  H         CH.sub.3    4-C(CH.sub.3)═NO-t-C.sub.4 H.sub.9                  H         CH.sub.3    3-C(CH.sub.3)═NO-n-C.sub.5 H.sub.11                 H         CH.sub.3    4-C(CH.sub.3)═NO-n-C.sub.5 H.sub.11                 H         CH.sub.3    3-C(CH.sub.3)═NO-n-C.sub.6 H.sub.13                 H         CH.sub.3    4-C(CH.sub.3)═NO-n-C.sub.6 H.sub.13                 H         CH.sub.3    2-Cl, 4-CH.sub.3                                        H         CH.sub.3    2-Cl, 5-CH.sub.3                                        H         CH.sub.3    3-Cl, 4-CH.sub.3                                        H         CH.sub.3    3-Cl, 5-CH.sub.3                                        H         CH.sub.3    2-CH.sub.3, 4-Cl                                        H         CH.sub.3    2-CH.sub.3, 5-Cl                                        H         CH.sub.3    3-CH.sub.3, 4-Cl                                        H         CH.sub.3    3-Cl, 5-t-C.sub.4 H.sub.9                               H         CH.sub.3    2-Cl, 4-t-C.sub.4 H.sub.9                               H         CH.sub.3    2-F, 4-CH.sub.3                                         H         CH.sub.3    3-F, 4-CH.sub.3                                         H         CH.sub.3    3-F, 5-CH.sub.3                                         H         CH.sub.3    2-CH.sub.3, 4-F                                         H         CH.sub.3    3-CH.sub.3, 4-F                                         H         CH.sub.3    2-F, 4-t-C.sub.4 H.sub.9                                H         CH.sub.3    3-F, 4-t-C.sub.4 H.sub.9                                H         CH.sub.3    2-F, 4-OCH.sub.3                                        H         CH.sub.3    2-Br, 4-CH.sub.3                                        H         CH.sub.3    3-Br, 4-CH.sub.3                                        H         CH.sub.3    3-Br, 5-CH.sub.3                                        H         CH.sub.3    2-CH.sub.3, 4-Br                                        H         CH.sub.3    3-CH.sub.3, 4-Br                                        H         CH.sub.3    2-Br, 4-t-C.sub.4 H.sub.9                               H         CH.sub.3    2-Cl, 4-NO.sub.2                                        H         CH.sub.3    3-Cl, 4-NO.sub.2                                        H         CH.sub.3    3-Cl, 5-NO.sub.2                                        H         CH.sub.3    3-NO.sub.2, 4-Cl                                        H         CH.sub.3    3-Cl, 4-OCH                                             H         CH.sub.3    3-OCH.sub.3, 4-Cl                                       H         CH.sub.3    2-Cl, 5-CF.sub.3                                        H         CH.sub.3    3-Cl, 4-CF.sub.3                                        H         CH.sub.3    3-Cl, 5-CF.sub.3                                        H         CH.sub.3    3-CF.sub.3, 4-Cl                                        H         CH.sub.3    3-Cl, 5-OCF.sub.3                                       H         CH.sub.3    3-F, 5-CF.sub.3                                         H         CH.sub.3    2-CH.sub.3, 4-CN                                        H         CH.sub.3    3-NO.sub.2, 4-CH.sub.3                                  H         CH.sub.3    2-CH.sub.3, 4-OCH.sub.3                                 H         CH.sub.3    3-CH.sub.3, 4-OCH.sub.3                                 H         CH.sub.3    3-CH.sub.3, 5-OCH.sub.3                                 H         CH.sub.3    3-OCH.sub.3, 4-CH.sub.3                                 H         CH.sub.3    2-CH.sub.3, 4-O-i-C.sub.3 H.sub.7                       H         CH.sub.3    3-CH.sub.3, 4-O-i-C.sub.3 H.sub.7                       H         CH.sub.3    3-O-i-C.sub.3 H.sub.7, 4-CH.sub.3                       H         CH.sub.3    2-CH.sub.3, 4-CF.sub.3                                  H         CH.sub.3    2-CH.sub.3, 5-CF.sub.3                                  H         CH.sub.3    3-CH.sub.3, 4-CF.sub.3                                  H         CH.sub.3    3-CH.sub.3, 5-CF.sub.3                                  H         CH.sub.3    3-CF.sub.3, 4-CH.sub.3                                  H         CH.sub.3    3-CF.sub.3, 4-OCH.sub.3                                 H         CH.sub.3    3-OCH.sub.3, 4-CF.sub.3                                 H         CH.sub.3    2-CH.sub.3, 4-C(CH.sub.3)═NOCH.sub.3                H         CH.sub.3    3-CH.sub.3, 4-C(CH.sub.3)═NOCH.sub.3                H         CH.sub.3    2-OH, 5-CH.sub.3                                        H         CH.sub.3    3-CH.sub.3, 4-OC.sub.2 H.sub.5                          H         CH.sub.3    3-CH.sub.3, 4-O-t-C.sub.4 H.sub.9                       H         CH.sub.3    3-OC.sub.2 H.sub.5, 4-CH.sub.3                          H         CH.sub.3    3-O-t-C.sub.4 H.sub.9, 4-CH.sub.3                       H         CH.sub.3    2-C(COOCH.sub.3)═NOCH.sub.3                         H         CH.sub.3    2,3-Butadienyl                                          H         CH.sub.3    3,4-Butadienyl                                          CH.sub.3  CH.sub.3    H                                                       CH.sub.3  CH.sub.3    2-F                                                     CH.sub.3  CH.sub.3    3-F                                                     CH.sub.3  CH.sub.3    4-F                                                     CH.sub.3  CH.sub.3    2,4-F.sub.2                                             CH.sub.3  CH.sub.3    3,4-F.sub.2                                             CH.sub.3  CH.sub.3    3,5-F.sub.2                                             CH.sub.3  CH.sub.3    2-Cl                                                    CH.sub.3  CH.sub.3    3-Cl                                                    CH.sub.3  CH.sub.3    4-Cl                                                    CH.sub.3  CH.sub.3    2,4-Cl.sub.2                                            CH.sub.3  CH.sub.3    3,4-Cl.sub.2                                            CH.sub.3  CH.sub.3    3,5-Cl.sub.2                                            CH.sub.3  CH.sub.3    2-Br                                                    CH.sub.3  CH.sub.3    3-Br                                                    CH.sub.3  CH.sub.3    4-Br                                                    CH.sub.3  CH.sub.3    3,5-Br.sub.2                                            CH.sub.3  CH.sub.3    3-I                                                     CH.sub.3  CH.sub.3    4-I                                                     CH.sub.3  CH.sub.3    3-F, 5-Cl                                               CH.sub.3  CH.sub.3    3-F, 5-Br                                               CH.sub.3  CH.sub.3    3-Cl, 5-Br                                              CH.sub.3  CH.sub.3    3-Br, 4-F                                               CH.sub.3  CH.sub.3    2-NO.sub.2                                              CH.sub.3  CH.sub.3    3-NO.sub.2                                              CH.sub.3  CH.sub.3    4-NO.sub.2                                              CH.sub.3  CH.sub.3    2-CN                                                    CH.sub.3  CH.sub.3    3-CN                                                    CH.sub.3  CH.sub.3    4-CN                                                    CH.sub.3  CH.sub.3    2-CH.sub.3                                              CH.sub.3  CH.sub.3    3-CH.sub.3                                              CH.sub.3  CH.sub.3    4-CH.sub.3                                              CH.sub.3  CH.sub.3    2,4-(CH.sub.3).sub.2                                    CH.sub.3  CH.sub.3    2,5-(CH.sub.3).sub.2                                    CH.sub.3  CH.sub.3    3,4-(CH.sub.3).sub.2                                    CH.sub.3  CH.sub.3    3,5-(CH.sub.3).sub.2                                    CH.sub.3  CH.sub.3    2,4,5-(CH.sub.3).sub.3                                  CH.sub.3  CH.sub.3    2,4,6-(CH.sub.3).sub.3                                  CH.sub.3  CH.sub.3    3-C.sub.2 H.sub.5                                       CH.sub.3  CH.sub.3    4-C.sub.2 H.sub.5                                       CH.sub.3  CH.sub.3    3,4-(C.sub.2 H.sub.5).sub.2                             CH.sub.3  CH.sub.3    3,5-(C.sub.2 H.sub.5).sub.2                             CH.sub.3  CH.sub.3    3-n-C.sub.3 H.sub.7                                     CH.sub.3  CH.sub.3    4-n-C.sub.3 H.sub.7                                     CH.sub.3  CH.sub.3    3-i-C.sub.3 H.sub.7                                     CH.sub.3  CH.sub.3    4-i-C.sub.3 H.sub.7                                     CH.sub.3  CH.sub.3    3-Cyclopropyl                                           CH.sub.3  CH.sub.3    4-Cyclopropyl                                           CH.sub.3  CH.sub.3    3-n-C.sub.4 H.sub.9                                     CH.sub.3  CH.sub.3    4-n-C.sub.4 H.sub.9                                     CH.sub.3  CH.sub.3    3-t-C.sub.4 H.sub.9                                     CH.sub.3  CH.sub.3    4-t-C.sub.4 H.sub.9                                     CH.sub.3  CH.sub.3    3-n-C.sub.6 H.sub.13                                    CH.sub.3  CH.sub.3    4-n-C.sub.6 H.sub.13                                    CH.sub.3  CH.sub.3    3-Cyclohexyl                                            CH.sub.3  CH.sub.3    4-Cyclohexyl                                            CH.sub.3  CH.sub.3    3-Phenyl                                                CH.sub.3  CH.sub.3    4-Phenyl                                                CH.sub.3  CH.sub.3    4-Allyl                                                 CH.sub.3  CH.sub.3    4-Propargyl                                             CH.sub.3  CH.sub.3    2-CH.sub.3, 4-C.sub.2 H.sub.5                           CH.sub.3  CH.sub.3    2-CH.sub.3, 4-i-C.sub.3 H.sub.7                         CH.sub.3  CH.sub.3    2-CH.sub.3, 4-t-C.sub.4 H.sub.9                         CH.sub.3  CH.sub.3    2-CH.sub.3, 4-phenyl                                    CH.sub.3  CH.sub.3    3-CH.sub.3, 4-phenyl                                    CH.sub.3  CH.sub.3    3-OH                                                    CH.sub.3  CH.sub.3    4-OH                                                    CH.sub.3  CH.sub.3    3-OCH.sub.3                                             CH.sub.3  CH.sub.3    4-OCH.sub.3                                             CH.sub.3  CH.sub.3    3,4-(OCH.sub.3).sub.2                                   CH.sub.3  CH.sub.3    3,5-(OCH.sub.3).sub.2                                   CH.sub.3  CH.sub.3    3,4,5-(OCH.sub.3).sub.3                                 CH.sub.3  CH.sub.3    4-OC.sub.2 H.sub.5                                      CH.sub.3  CH.sub.3    4-O-i-C.sub.3 H.sub.7                                   CH.sub.3  CH.sub.3    3-O-t-C.sub.4 H.sub.9                                   CH.sub.3  CH.sub.3    4-O-t-C.sub.4 H.sub.9                                   CH.sub.3  CH.sub.3    4-O-n-C.sub.6 H.sub.13                                  CH.sub.3  CH.sub.3    3-O-Phenyl                                              CH.sub.3  CH.sub.3    4-O-Phenyl                                              CH.sub.3  CH.sub.3    4-O-Allyl                                               CH.sub.3  CH.sub.3    2-CF.sub.3                                              CH.sub.3  CH.sub.3    3-CF.sub.3                                              CH.sub.3  CH.sub.3    4-CF.sub.3                                              CH.sub.3  CH.sub.3    3,5-(CF.sub.3).sub.2                                    CH.sub.3  CH.sub.3    4-CH.sub.2 CF.sub.3                                     CH.sub.3  CH.sub.3    4-C.sub.2 F.sub.5                                       CH.sub.3  CH.sub.3    4-CF.sub.2 CHF.sub.2                                    CH.sub.3  CH.sub.3    3-OCF.sub.3                                             CH.sub.3  CH.sub.3    4-OCF.sub.3                                             CH.sub.3  CH.sub.3    4-OCH.sub.2 CF.sub.3                                    CH.sub.3  CH.sub.3    4-OC.sub.2 F.sub.5                                      CH.sub.3  CH.sub.3    4-OCF.sub.2 CHF.sub.2                                   CH.sub.3  CH.sub.3    3-CH.sub.2 OCH.sub.3                                    CH.sub.3  CH.sub.3    4-CH.sub.2 OCH.sub.3                                    CH.sub.3  CH.sub.3    4-CH.sub.2 --O-t-C.sub.4 H.sub.9                        CH.sub.3  CH.sub.3    4-CH(OCH.sub.3).sub.2                                   CH.sub.3  CH.sub.3    4-CH.sub.2 CN                                           CH.sub.3  CH.sub.3    3-CHO                                                   CH.sub.3  CH.sub.3    4-CHO                                                   CH.sub.3  CH.sub.3    3-CO--CH.sub.3                                          CH.sub.3  CH.sub.3    4-CO--CH.sub.3                                          CH.sub.3  CH.sub.3    3-COOH                                                  CH.sub.3  CH.sub.3    4-COOH                                                  CH.sub.3  CH.sub.3    3-COOCH.sub.3                                           CH.sub.3  CH.sub.3    4-COOCH.sub.3                                           CH.sub.3  CH.sub.3    3-COOC.sub.2 H.sub.5                                    CH.sub.3  CH.sub.3    4-COOC.sub.2 H.sub.5                                    CH.sub.3  CH.sub.3    3-COO-i-C.sub.3 H.sub.7                                 CH.sub.3  CH.sub.3    4-COO-i-C.sub.3 H.sub.7                                 CH.sub.3  CH.sub.3    3-COO-t-C.sub.4 H.sub.9                                 CH.sub.3  CH.sub.3    4-COO-t-C.sub.4 H.sub.9                                 CH.sub.3  CH.sub.3    3-COO-n-C.sub.6 H.sub.13                                CH.sub.3  CH.sub.3    4-COO-n-C.sub.6 H.sub.13                                CH.sub.3  CH.sub.3    3-CONH.sub.2                                            CH.sub.3  CH.sub.3    4-CONH.sub.2                                            CH.sub.3  CH.sub.3    3-CONHCH.sub.3                                          CH.sub.3  CH.sub.3    4-CONHCH.sub.3                                          CH.sub.3  CH.sub.3    3-CON(CH.sub.3).sub.2                                   CH.sub.3  CH.sub.3    4-CON(CH.sub.3).sub.2                                   CH.sub.3  CH.sub.3    3-CSNH.sub.2                                            CH.sub.3  CH.sub.3    4-CSNH.sub.2                                            CH.sub.3  CH.sub.3    3-NH.sub.2                                              CH.sub.3  CH.sub.3    4-NH.sub.2                                              CH.sub.3  CH.sub.3    4-NHCH.sub.3                                            CH.sub.3  CH.sub.3    4-N(CH.sub.3).sub.2                                     CH.sub.3  CH.sub.3    3-NHCO--CH.sub.3                                        CH.sub.3  CH.sub.3    4-NHCO--CH.sub.3                                        CH.sub.3  CH.sub.3    4-NCH.sub.3 --CO--CH.sub.3                              CH.sub.3  CH.sub.3    4-NHCOOCH.sub.3                                         CH.sub.3  CH.sub.3    4-NCH.sub.3 --COOCH.sub.3                               CH.sub.3  CH.sub.3    3-OCO--CH.sub.3                                         CH.sub.3  CH.sub.3    4-OCO--CH.sub.3                                         CH.sub.3  CH.sub.3    4-OCO-t-C.sub.4 H.sub.9                                 CH.sub.3  CH.sub.3    4-SH                                                    CH.sub.3  CH.sub.3    4-SCH.sub.3                                             CH.sub.3  CH.sub.3    4-S-t-C.sub.4 H.sub.9                                   CH.sub.3  CH.sub.3    4-SO--CH.sub.3                                          CH.sub.3  CH.sub.3    4-SO.sub.2 --CH.sub.3                                   CH.sub.3  CH.sub.3    4-C(CH.sub.3)═NCH.sub.3                             CH.sub.3  CH.sub.3    4-C(SCH.sub.3)═NOCH.sub.3                           CH.sub.3  CH.sub.3    4-C(OCH.sub.3)═NOCH.sub.3                           CH.sub.3  CH.sub.3    3-CH═NOCH.sub.3                                     CH.sub.3  CH.sub.3    4-CH═NOCH.sub.3                                     CH.sub.3  CH.sub.3    3-C(CH.sub.3)═NOCH.sub.3                            CH.sub.3  CH.sub.3    4-C(CH.sub.3)═NOCH.sub.3                            CH.sub.3  CH.sub.3    4-C(CH.sub.3)═NOC.sub.2 H.sub.5                     CH.sub.3  CH.sub.3    4-C(CH.sub.3)═NO-n-C.sub.3 H.sub.7                  CH.sub.3  CH.sub.3    4-C(CH.sub.3)═NO-i-C.sub.3 H.sub.7                  CH.sub.3  CH.sub.3    4-C(CH.sub.3)═NO-n-C.sub.4 H.sub.9                  CH.sub.3  CH.sub.3    4-C(CH.sub.3)═NO-t-C.sub.4 H.sub.9                  CH.sub.3  CH.sub.3    4-C(CH.sub.3)═NO-n-C.sub.5 H.sub.11                 CH.sub.3  CH.sub.3    4-C(CH.sub.3)═NO-n-C.sub.6 H.sub.13                 CH.sub.3  CH.sub.3    2-Cl, 4-CH.sub.3                                        CH.sub.3  CH.sub.3    3-Cl, 5-CH.sub.3                                        CH.sub.3  CH.sub.3    2-CH.sub.3, 4-Cl                                        CH.sub.3  CH.sub.3    3-CH.sub.3, 4-Cl                                        CH.sub.3  CH.sub.3    3-F, 5-CH.sub.3                                         CH.sub.3  CH.sub.3    3-Br, 5-CH.sub.3                                        CH.sub.3  CH.sub.3    3-Cl, 5-NO.sub.2                                        CH.sub.3  CH.sub.3    3-NO.sub.2, 4-Cl                                        CH.sub.3  CH.sub.3    3-Cl, 4-OCH.sub.3                                       CH.sub.3  CH.sub.3    3-OCH.sub.3, 4-Cl                                       CH.sub.3  CH.sub.3    3-Cl, 5-CF.sub.3                                        CH.sub.3  CH.sub.3    3-Cl, 5-OCF.sub.3                                       CH.sub.3  CH.sub.3    3-F, 5-CF.sub.3                                         CH.sub.3  CH.sub.3    2-CH.sub.3, 4-CN                                        CH.sub.3  CH.sub.3    2-CH.sub.3, 4-OCH.sub.3                                 CH.sub.3  CH.sub.3    2-CH.sub.3, 4-CF.sub.3                                  CH.sub.3  CH.sub.3    2-CH.sub.3, 4-C(CH.sub.3)═NOCH.sub.3                CH.sub.3  CH.sub.3    3-CH.sub.3, 4-C(CH.sub.3)═NOCH.sub.3                CH.sub.3  CH.sub.3    2-OH, 5-CH.sub.3                                        CH.sub.3  CH.sub.3    3-CH.sub.3, 4-O-t-C.sub.4 H.sub.9                       CH.sub.3  CH.sub.3    2-C(COOCH.sub.3)═NOCH.sub.3                         CH.sub.3  CH.sub.3    2,3-Butadienyl                                          CH.sub.3  CH.sub.3    3,4-Butadienyl                                          H         Cyclopropyl H                                                       H         Cyclopropyl 2-F                                                     H         Cyclopropyl 3-F                                                     H         Cyclopropyl 4-F                                                     H         Cyclopropyl 2,3-F.sub.2                                             H         Cyclopropyl 2,4-F.sub.2                                             H         Cyclopropyl 2,5-F.sub.2                                             H         Cyclopropyl 2,6-F.sub.2                                             H         Cyclopropyl 3,4-F.sub.2                                             H         Cyclopropyl 3,5-F.sub.2                                             H         Cyclopropyl 2-Cl                                                    H         Cyclopropyl 3-Cl                                                    H         Cyclopropyl 4-Cl                                                    H         Cyclopropyl 2,4-Cl.sub.2                                            H         Cyclopropyl 2,5-Cl.sub.2                                            H         Cyclopropyl 3,4-Cl.sub.2                                            H         Cyclopropyl 3,5-Cl.sub.2                                            H         Cyclopropyl 2-Br                                                    H         Cyclopropyl 3-Br                                                    H         Cyclopropyl 4-Br                                                    H         Cyclopropyl 2,4-Br.sub.2                                            H         Cyclopropyl 3,4-Br.sub.2                                            H         Cyclopropyl 3,5-Br.sub.2                                            H         Cyclopropyl 2-I                                                     H         Cyclopropyl 3-I                                                     H         Cyclopropyl 4-I                                                     H         Cyclopropyl 2-F, 4-Cl                                               H         Cyclopropyl 2-F, 5-Cl                                               H         Cyclopropyl 2-F, 4-Br                                               H         Cyclopropyl 2-F, 5-Br                                               H         Cyclopropyl 2-Cl, 4-Br                                              H         Cyclopropyl 2-Cl, 5-Br                                              H         Cyclopropyl 3-F, 4-Cl                                               H         Cyclopropyl 3-F, 5-Cl                                               H         Cyclopropyl 3-F, 4-Br                                               H         Cyclopropyl 3-F, 5-Br                                               H         Cyclopropyl 3-Cl, 4-Br                                              H         Cyclopropyl 3-Cl, 5-Br                                              H         Cyclopropyl 3-Cl, 4-F                                               H         Cyclopropyl 3-Br, 4-F                                               H         Cyclopropyl 3-Br, 4-Cl                                              H         Cyclopropyl 2-NO.sub.2                                              H         Cyclopropyl 3-NO.sub.2                                              H         Cyclopropyl 4-NO.sub.2                                              H         Cyclopropyl 2-CN                                                    H         Cyclopropyl 3-CN                                                    H         Cyclopropyl 4-CN                                                    H         Cyclopropyl 2-CH.sub.3                                              H         Cyclopropyl 3-CH.sub.3                                              H         Cyclopropyl 4-CH.sub.3                                              H         Cyclopropyl 2,3-(CH.sub.3).sub.2                                    H         Cyclopropyl 2,4-(CH.sub.3).sub.2                                    H         Cyclopropyl 2,5-(CH.sub.3).sub.2                                    H         Cyclopropyl 2,6-(CH.sub.3).sub.2                                    H         Cyclopropyl 3,4-(CH.sub.3).sub.2                                    H         Cyclopropyl 3,5-(CH.sub.3).sub.2                                    H         Cyclopropyl 2,4,5-(CH.sub.3).sub.3                                  H         Cyclopropyl 2,4,6-(CH.sub.3).sub.3                                  H         Cyclopropyl 3,4,5-(CH.sub.3).sub.3                                  H         Cyclopropyl 2-C.sub.2 H.sub.5                                       H         Cyclopropyl 3-C.sub.2 H.sub.5                                       H         Cyclopropyl 4-C.sub.2 H.sub.5                                       H         Cyclopropyl 3,4-(C.sub.2 H.sub.5).sub.2                             H         Cyclopropyl 3,5-(C.sub.2 H.sub.5).sub.2                             H         Cyclopropyl 3-n-C.sub.3 H.sub.7                                     H         Cyclopropyl 4-n-C.sub.3 H.sub.7                                     H         Cyclopropyl 3,4-(n-C.sub.3 H.sub.7).sub.2                           H         Cyclopropyl 3,5-(n-C.sub.3 H.sub.7).sub.2                           H         Cyclopropyl 3-i-C.sub.3 H.sub.7                                     H         Cyclopropyl 4-i-C.sub.3 H.sub.7                                     H         Cyclopropyl 3,4-(i-C.sub.3 H.sub.7).sub.2                           H         Cyclopropyl 3,5-(i-C.sub.3 H.sub.7).sub.2                           H         Cyclopropyl 3-Cyclopropyl                                           H         Cyclopropyl 4-Cyclopropyl                                           H         Cyclopropyl 3-n-C.sub.4 H.sub.9                                     H         Cyclopropyl 4-n-C.sub.4 H.sub.9                                     H         Cyclopropyl 3,4-(n-C.sub.4 H.sub.9).sub.2                           H         Cyclopropyl 3,5-(n-C.sub.4 H.sub.9).sub.2                           H         Cyclopropyl 3-s-C.sub.4 H.sub.9                                     H         Cyclopropyl 4-s-C.sub.4 H.sub.9                                     H         Cyclopropyl 3-i-C.sub.4 H.sub.9                                     H         Cyclopropyl 4-i-C.sub.4 H.sub.9                                     H         Cyclopropyl 3-t-C.sub.4 H.sub.9                                     H         Cyclopropyl 4-t-C.sub.4 H.sub.9                                     H         Cyclopropyl 3,4-(t-C.sub.4 H.sub.9).sub.2                           H         Cyclopropyl 3,5-(t-C.sub.4 H.sub.9).sub.2                           H         Cyclopropyl 3-n-C.sub.5 H.sub.11                                    H         Cyclopropyl 4-n-C.sub.5 H.sub.11                                    H         Cyclopropyl 3-n-C.sub.6 H.sub.13                                    H         Cyclopropyl 4-n-C.sub.6 H.sub.13                                    H         Cyclopropyl 3-Cyclohexyl                                            H         Cyclopropyl 4-Cyclohexyl                                            H         Cyclopropyl 3-Phenyl                                                H         Cyclopropyl 4-Phenyl                                                H         Cyclopropyl 3-Vinyl                                                 H         Cyclopropyl 4-Vinyl                                                 H         Cyclopropyl 3-Allyl                                                 H         Cyclopropyl 4-Allyl                                                 H         Cyclopropyl 3-Propargyl                                             H         Cyclopropyl 4-Propargyl                                             H         Cyclopropyl 3-(Propen-2-yl)                                         H         Cyclopropyl 4-(Propen-2-yl)                                         H         Cyclopropyl 2-CH.sub.3, 4-C.sub.2 H.sub.5                           H         Cyclopropyl 2-CH.sub.3, 5-C.sub.2 H.sub.5                           H         Cyclopropyl 2-CH.sub.3 --, 4-n-C.sub.3 H.sub.7                      H         Cyclopropyl 2-CH.sub.3, 5-n-C.sub.3 H.sub.7                         H         Cyclopropyl 2-CH.sub.3, 4-i-C.sub.3 H.sub.7                         H         Cyclopropyl 2-CH.sub.3, 5-i-C.sub.3 H.sub.7                         H         Cyclopropyl 2-CH.sub.3, 4-n-C.sub.4 H.sub.9                         H         Cyclopropyl 2-CH.sub.3, 4-s-C.sub.4 H.sub.9                         H         Cyclopropyl 2-CH.sub.3, 4-i-C.sub.4 H.sub.9                         H         Cyclopropyl 2-CH.sub.3, 4-t-C.sub.4 H.sub.9                         H         Cyclopropyl 2-CH.sub.3, 4-phenyl                                    H         Cyclopropyl 2-CH.sub.3, 5-phenyl                                    H         Cyclopropyl 2-CH.sub.3, 4-vinyl                                     H         Cyclopropyl 2-CH.sub.3, 4-allyl                                     H         Cyclopropyl 2-CH.sub.3, 4-propargyl                                 H         Cyclopropyl 2-CH.sub.3, 4-(propen-2-yl)                             H         Cyclopropyl 3-CH.sub.3, 4-C.sub.2 H.sub.5                           H         Cyclopropyl 3-CH.sub.3, 5-C.sub.2 H.sub.5                           H         Cyclopropyl 3-CH.sub.3, 4-n-C.sub.3 H.sub.7                         H         Cyclopropyl 3-CH.sub.3, 5-n-C.sub.3 H.sub.7                         H         Cyclopropyl 3-CH.sub.3, 4-i-C.sub.3 H.sub.7                         H         Cyclopropyl 3-CH.sub.3, 5-i-C.sub.3 H.sub.7                         H         Cyclopropyl 3-CH.sub.3, 4-cyclopropyl                               H         Cyclopropyl 3-CH.sub.3, 4-t-C.sub.4 H.sub.9                         H         Cyclopropyl 3-CH.sub.3, 5-t-C.sub.4 H.sub.9                         H         Cyclopropyl 3-CH.sub.3, 4-phenyl                                    H         Cyclopropyl 3-CH.sub.3, 5-Phenyl                                    H         Cyclopropyl 3-CH.sub.3, 4-vinyl                                     H         Cyclopropyl 3-CH.sub.3, 4-allyl                                     H         Cyclopropyl 3-CH.sub.3, 4-propargyl                                 H         Cyclopropyl 3-CH.sub.3, 4-propen-2-yl                               H         Cyclopropyl 3-C.sub.2 H.sub.5, 4-CH.sub.3                           H         Cyclopropyl 3-i-C.sub.3 H.sub.7, 4-CH.sub.3                         H         Cyclopropyl 3-t-C.sub.4 H.sub.9, 4-CH.sub.3                         H         Cyclopropyl 3-Phenyl, 4-CH.sub.3                                    H         Cyclopropyl 2-OH                                                    H         Cyclopropyl 3-OH                                                    H         Cyclopropyl 4-OH                                                    H         Cyclopropyl 2-OCH.sub.3                                             H         Cyclopropyl 3-OCH.sub.3                                             H         Cyclopropyl 4-OCH.sub.3                                             H         Cyclopropyl 2,3-(OCH.sub.3).sub.2                                   H         Cyclopropyl 2,4-(OCH.sub.3).sub.2                                   H         Cyclopropyl 2,5-(OCH.sub.3).sub.2                                   H         Cyclopropyl 3,4-(OCH.sub.3).sub.2                                   H         Cyclopropyl 3,5-(OCH.sub.3).sub.2                                   H         Cyclopropyl 3,4,5-(OCH.sub.3).sub.3                                 H         Cyclopropyl 3-OC.sub.2 H.sub.5                                      H         Cyclopropyl 4-OC.sub.2 H.sub.5                                      H         Cyclopropyl 3,4-(OC.sub.2 H.sub.5).sub.2                            H         Cyclopropyl 3,5-(OC.sub.2 H.sub.5).sub.2                            H         Cyclopropyl 3-O-n-C.sub.3 H.sub.7                                   H         Cyclopropyl 4-O-n-C.sub.3 H.sub.7                                   H         Cyclopropyl 3-O-i-C.sub.3 H.sub.7                                   H         Cyclopropyl 4-O-i-C.sub.3 H.sub.7                                   H         Cyclopropyl 3-O-Cyclopropyl                                         H         Cyclopropyl 4-O-Cyclopropyl                                         H         Cyclopropyl 3-O-n-C.sub.4 H.sub.9                                   H         Cyclopropyl 4-O-n-C.sub.4 H.sub.9                                   H         Cyclopropyl 3-O-s-C.sub.4 H.sub.9                                   H         Cyclopropyl 4-O-s-C.sub.4 H.sub.9                                   H         Cyclopropyl 3-O-i-C.sub.4 H.sub.9                                   H         Cyclopropyl 4-O-i-C.sub.4 H.sub.9                                   H         Cyclopropyl 3-O-t-C.sub.4 H.sub.9                                   H         Cyclopropyl 4-O-t-C.sub.4 H.sub.9                                   H         Cyclopropyl 3-O-n-C.sub.5 H.sub.11                                  H         Cyclopropyl 4-O-n-C.sub.5 H.sub.11                                  H         Cyclopropyl 3-O-n-C.sub.6 H.sub.13                                  H         Cyclopropyl 4-O-n-C.sub.6 H.sub.13                                  H         Cyclopropyl 3-O-Cyclohexyl                                          H         Cyclopropyl 4-O-Cyclohexyl                                          H         Cyclopropyl 3-O-Phenyl                                              H         Cyclopropyl 4-O-Phenyl                                              H         Cyclopropyl 3-O-Allyl                                               H         Cyclopropyl 4-O-Allyl                                               H         Cyclopropyl 2-CF.sub.3                                              H         Cyclopropyl 3-CF.sub.3                                              H         Cyclopropyl 4-CF.sub.3                                              H         Cyclopropyl 2,4-(CF.sub.3).sub.2                                    H         Cyclopropyl 3,5-(CF.sub.3).sub.2                                    H         Cyclopropyl 3-CF.sub.2 Cl                                           H         Cyclopropyl 4-CF.sub.2 Cl                                           H         Cyclopropyl 3-CFCl.sub.2                                            H         Cyclopropyl 4-CFCl.sub.2                                            H         Cyclopropyl 3-CCl.sub.3                                             H         Cyclopropyl 4-CCl.sub.3                                             H         Cyclopropyl 3-CH.sub.2 CH.sub.2 F                                   H         Cyclopropyl 4-CH.sub.2 CH.sub.2 F                                   H         Cyclopropyl 3-CH.sub.2 CF.sub.3                                     H         Cyclopropyl 4-CH.sub.2 CF.sub.3                                     H         Cyclopropyl 3-C.sub.2 F.sub.5                                       H         Cyclopropyl 4-C.sub.2 F.sub.5                                       H         Cyclopropyl 3-CHCl.sub.2                                            H         Cyclopropyl 4-CHCl.sub.2                                            H         Cyclopropyl 3-CH.sub.2 Cl                                           H         Cyclopropyl 4-CH.sub.2 Cl                                           H         Cyclopropyl 3-CF.sub.2 CHF.sub.2                                    H         Cyclopropyl 4-CF.sub.2 CHF.sub.2                                    H         Cyclopropyl 3-CH.sub.2 CH.sub.2 Cl                                  H         Cyclopropyl 4-CH.sub.2 CH.sub.2 Cl                                  H         Cyclopropyl 2-OCF.sub.3                                             H         Cyclopropyl 3-OCF.sub.3                                             H         Cyclopropyl 4-OCF.sub.3                                             H         Cyclopropyl 3-OCHF.sub.2                                            H         Cyclopropyl 4-OCHF.sub.2                                            H         Cyclopropyl 3-OC.sub.2 F.sub.5                                      H         Cyclopropyl 4-OC.sub.2 F.sub.5                                      H         Cyclopropyl 3-OCF.sub.2 CHF.sub.2                                   H         Cyclopropyl 4-OCF.sub.2 CHF.sub.2                                   H         Cyclopropyl 3-CH.sub.2 OCH.sub.3                                    H         Cyclopropyl 4-CH.sub.2 OCH.sub.3                                    H         Cyclopropyl 3-CH.sub.2 O-t-C.sub.4 H.sub.9                          H         Cyclopropyl 4-CH.sub.2 O-t-C.sub.4 H.sub.9                          H         Cyclopropyl 3-C(CH.sub.3)(OCH.sub.3).sub.2                          H         Cyclopropyl 4-C(CH.sub.3)(OCH.sub.3).sub.2                          H         Cyclopropyl 3-CH(OCH.sub.3).sub.2                                   H         Cyclopropyl 4-CH(OCH.sub.3).sub.2                                   H         Cyclopropyl 3-CH.sub.2 CN                                           H         Cyclopropyl 4-CH.sub.2 CN                                           H         Cyclopropyl 3-CHO                                                   H         Cyclopropyl 4-CHO                                                   H         Cyclopropyl 3-CO--CH.sub.3                                          H         Cyclopropyl 4-CO--CH.sub.3                                          H         Cyclopropyl 3-CO--C.sub.2 H.sub.5                                   H         Cyclopropyl 4-CO--C.sub.2 H.sub.5                                   H         Cyclopropyl 2-COOH                                                  H         Cyclopropyl 3-COOH                                                  H         Cyclopropyl 4-COOH                                                  H         Cyclopropyl 3-COOCH.sub.3                                           H         Cyclopropyl 4-COOCH.sub.3                                           H         Cyclopropyl 3-COOC.sub.2 H.sub.5                                    H         Cyclopropyl 4-COOC.sub.2 H.sub.5                                    H         Cyclopropyl 3-COO-n-C.sub.3 H.sub.7                                 H         Cyclopropyl 4-COO-n-C.sub.3 H.sub.7                                 H         Cyclopropyl 3-COO-i-C.sub.3 H.sub.7                                 H         Cyclopropyl 4-COO-i-C.sub.3 H.sub.7                                 H         Cyclopropyl 3-COO-n-C.sub.4 H.sub.9                                 H         Cyclopropyl 4-COO-n-C.sub.4 H.sub.9                                 H         Cyclopropyl 3-COO-s-C.sub.4 H.sub.9                                 H         Cyclopropyl 4-COO-s-C.sub.4 H.sub.9                                 H         Cyclopropyl 3-COO-i-C.sub.4 H.sub.9                                 H         Cyclopropyl 4-COO-i-C.sub.4 H.sub.9                                 H         Cyclopropyl 3-COO-t-C.sub.4 H.sub.9                                 H         Cyclopropyl 4-COO-t-C.sub.4 H.sub.9                                 H         Cyclopropyl 3-COO-n-C.sub.5 H.sub.11                                H         Cyclopropyl 4-COO-n-C.sub.5 H.sub.11                                H         Cyclopropyl 3-COO-n-C.sub.6 H.sub.13                                H         Cyclopropyl 4-COO-n-C.sub.6 H.sub.13                                H         Cyclopropyl 2-CONH.sub.2                                            H         Cyclopropyl 3-CONH.sub.2                                            H         Cyclopropyl 4-CONH.sub.2                                            H         Cyclopropyl 3-CONHCH.sub.3                                          H         Cyclopropyl 4-CONHCH.sub.3                                          H         Cyclopropyl 3-CON(CH.sub.3).sub.2                                   H         Cyclopropyl 4-CON(CH.sub.3).sub.2                                   H         Cyclopropyl 3-CON(C.sub.2 H.sub.5).sub.2                            H         Cyclopropyl 4-CON(C.sub.2 H.sub.5).sub.2                            H         Cyclopropyl 2-CSNH.sub.2                                            H         Cyclopropyl 3-CSNH.sub.2                                            H         Cyclopropyl 4-CSNH.sub.2                                            H         Cyclopropyl 2-NH.sub.2                                              H         Cyclopropyl 3-NH.sub.2                                              H         Cyclopropyl 4-NH.sub.2                                              H         Cyclopropyl 3-NHCH.sub.3                                            H         Cyclopropyl 4-NHCH.sub.3                                            H         Cyclopropyl 3-N(CH.sub.3).sub.2                                     H         Cyclopropyl 4-N(CH.sub.3).sub.2                                     H         Cyclopropyl 3-NHCO--CH.sub.3                                        H         Cyclopropyl 4-NHCO--CH.sub.3                                        H         Cyclopropyl 3-NCH.sub.3 --CO--CH.sub.3                              H         Cyclopropyl 4-NCH.sub.3 --CO--CH.sub.3                              H         Cyclopropyl 3-NHCOOCH.sub.3                                         H         Cyclopropyl 4-NHCOOCH.sub.3                                         H         Cyclopropyl 3-NCH.sub.3 --COOCH.sub.3                               H         Cyclopropyl 4-NCH.sub.3 --COOCH.sub.3                               H         Cyclopropyl 3-OCO--CH.sub.3                                         H         Cyclopropyl 4-OCO--CH.sub.3                                         H         Cyclopropyl 3-OCO-t-C.sub.4 H.sub.9                                 H         Cyclopropyl 4-OCO-t-C.sub.4 H.sub.9                                 H         Cyclopropyl 3-SH                                                    H         Cyclopropyl 4-SH                                                    H         Cyclopropyl 3-SCH.sub.3                                             H         Cyclopropyl 4-SCH.sub.3                                             H         Cyclopropyl 3-S-t-C.sub.4 H.sub.9                                   H         Cyclopropyl 4-S-t-C.sub.4 H.sub.9                                   H         Cyclopropyl 3-SO--CH.sub.3                                          H         Cyclopropyl 4-SO--CH.sub.3                                          H         Cyclopropyl 3-SO.sub.2 CH.sub.3                                     H         Cyclopropyl 4-SO.sub.2 CH.sub.3                                     H         Cyclopropyl 3-CH═NCH.sub.3                                      H         Cyclopropyl 4-CH═NCH.sub.3                                      H         Cyclopropyl 3-C(CH.sub.3)═NCH.sub.3                             H         Cyclopropyl 4-C(CH.sub.3)═NCH.sub.3                             H         Cyclopropyl 3-C(SCH.sub.3)═NOCH.sub.3                           H         Cyclopropyl 4-C(SCH.sub.3)═NOCH.sub.3                           H         Cyclopropyl 3-C(OCH.sub.3)═NOCH.sub.3                           H         Cyclopropyl 4-C(OCH.sub.3)═NOCH.sub.3                           H         Cyclopropyl 3-C(NH.sub.2)═NOCH.sub.3                            H         Cyclopropyl 4-C(NH.sub.2)═NOCH.sub.3                            H         Cyclopropyl 3-C(NHCH.sub.3)═NOCH.sub.3                          H         Cyclopropyl 4-C(NHCH.sub.3)═NOCH.sub.3                          H         Cyclopropyl 3-CH═NOCH.sub.3                                     H         Cyclopropyl 4-CH═NOCH.sub.3                                     H         Cyclopropyl 3-C(CH.sub.3)═NOCH.sub.3                            H         Cyclopropyl 4-C(CH.sub.3)═NOCH.sub.3                            H         Cyclopropyl 3-C(CH.sub.3)═NOC.sub.2 H.sub.5                     H         Cyclopropyl 4-C(CH.sub.3)═NOC.sub.2 H.sub.5                     H         Cyclopropyl 3-C(CH.sub.3)═NO-n-C.sub.3 H.sub.7                  H         Cyclopropyl 4-C(CH.sub.3)═NO-n-C.sub.3 H.sub.7                  H         Cyclopropyl 3-C(CH.sub.3)═NO-i-C.sub.3 H.sub.7                  H         Cyclopropyl 4-C(CH.sub.3)═NO-i-C.sub.3 H.sub.7                  H         Cyclopropyl 3-C(CH.sub.3)═NO-n-C.sub.4 H.sub.9                  H         Cyclopropyl 4-C(CH.sub.3)═NO-n-C.sub.4 H.sub.9                  H         Cyclopropyl 3-C(CH.sub.3)═NO-s-C.sub.4 H.sub.9                  H         Cyclopropyl 4-C(CH.sub.3)═NO-s-C.sub.4 H.sub.9                  H         Cyclopropyl 3-C(CH.sub.3)═NO-i-C.sub.4 H.sub.9                  H         Cyclopropyl 4-C(CH.sub.3)═NO-t-C.sub.4 H.sub.9                  H         Cyclopropyl 3-C(CH.sub.3)═NO-t-C.sub.4 H.sub.9                  H         Cyclopropyl 4-C(CH.sub.3)═NO-t-C.sub.4 H.sub.9                  H         Cyclopropyl 3-C(CH.sub.3)═NO-n-C.sub.5 H.sub.11                 H         Cyclopropyl 4-C(CH.sub.3)═NO-n-C.sub.5 H.sub.11                 H         Cyclopropyl 3-C(CH.sub.3)═NO-n-C.sub.6 H.sub.13                 H         Cyclopropyl 4-C(CH.sub.3)═NO-n-C.sub.6 H.sub.13                 H         Cyclopropyl 2-Cl, 4-CH.sub.3                                        H         Cyclopropyl 2-Cl, 5-CH.sub.3                                        H         Cyclopropyl 3-Cl, 4-CH.sub.3                                        H         Cyclopropyl 3-Cl, 5-CH.sub.3                                        H         Cyclopropyl 2-CH.sub.3, 4-Cl                                        H         Cyclopropyl 2-CH.sub.3, 5-Cl                                        H         Cyclopropyl 3-CH.sub.3, 4-Cl                                        H         Cyclopropyl 3-Cl, 5-t-C.sub.4 H.sub.9                               H         Cyclopropyl 2-Cl, 4-t-C.sub.4 H.sub.9                               H         Cyclopropyl 2-F, 4-CH.sub.3                                         H         Cyclopropyl 3-F, 4-CH.sub.3                                         H         Cyclopropyl 3-F, 5-CH.sub.3                                         H         Cyclopropyl 2-CH.sub.3, 4-F                                         H         Cyclopropyl 3-CH.sub.3, 4-F                                         H         Cyclopropyl 2-F, 4-t-C.sub.4 H.sub.9                                H         Cyclopropyl 3-F, 4-t-C.sub.4 H.sub.9                                H         Cyclopropyl 2-F, 4-OCH.sub.3                                        H         Cyclopropyl 2-Br, 4-CH.sub.3                                        H         Cyclopropyl 3-Br, 4-CH.sub.3                                        H         Cyclopropyl 3-Br, 5-CH.sub.3                                        H         Cyclopropyl 2-CH.sub.3, 4-Br                                        H         Cyclopropyl 3-CH.sub.3, 4-Br                                        H         Cyclopropyl 2-Br, 4-t-C.sub.4 H.sub.9                               H         Cyclopropyl 2-Cl, 4-NO.sub.2                                        H         Cyclopropyl 3-Cl, 4-NO.sub.2                                        H         Cyclopropyl 3-Cl, 5-NO.sub.2                                        H         Cyclopropyl 3-NO.sub.2, 4-Cl                                        H         Cyclopropyl 3-Cl, 4-OCH.sub.3                                       H         Cyclopropyl 3-OCH.sub.3, 4-Cl                                       H         Cyclopropyl 2-Cl, 5-CF.sub.3                                        H         Cyclopropyl 3-Cl, 4-CF.sub.3                                        H         Cyclopropyl 3-Cl, 5-CF.sub.3                                        H         Cyclopropyl 3-CF.sub.3, 4-Cl                                        H         Cyclopropyl 3-Cl, 5-OCF.sub.3                                       H         Cyclopropyl 3-F, 5-CF.sub.3                                         H         Cyclopropyl 2-CH.sub.3, 4-CN                                        H         Cyclopropyl 3-NO.sub.2, 4-CH.sub.3                                  H         Cyclopropyl 2-CH.sub.3, 4-OCH.sub.3                                 H         Cyclopropyl 3-CH.sub.3, 4-OCH.sub.3                                 H         Cyclopropyl 3-CH.sub.3, 5-OCH.sub.3                                 H         Cyclopropyl 3-OCH.sub.3, 4-CH.sub.3                                 H         Cyclopropyl 2-CH.sub.3, 4-O-i-C.sub.3 H.sub.7                       H         Cyclopropyl 3-CH.sub.3, 4-O-i-C.sub.3 H.sub.7                       H         Cyclopropyl 3-O-i-C.sub.3 H.sub.7, 4-CH.sub.3                       H         Cyclopropyl 2-CH.sub.3, 4-CF.sub.3                                  H         Cyclopropyl 2-CH.sub.3, 5-CF.sub.3                                  H         Cyclopropyl 3-CH.sub.3, 4-CF.sub.3                                  H         Cyclopropyl 3-CH.sub.3, 5-CF.sub.3                                  H         Cyclopropyl 3-CF.sub.3, 4-CH.sub.3                                  H         Cyclopropyl 3-CF.sub.3, 4-OCH.sub.3                                 H         Cyclopropyl 3-OCH.sub.3, 4-CF.sub.3                                 H         Cyclopropyl 2-CH.sub.3, 4-C(CH.sub.3)═NOCH.sub.3                H         Cyclopropyl 3-CH.sub.3, 4-C(CH.sub.3)═NOCH.sub.3                H         Cyclopropyl 2-OH, 5-CH.sub.3                                        H         Cyclopropyl 3-CH.sub.3, 4-OC.sub.2 H.sub.5                          H         Cyclopropyl 3-CH.sub.3, 4-O-t-C.sub.4 H.sub.9                       H         Cyclopropyl 3-OC.sub.2 H.sub.5, 4-CH.sub.3                          H         Cyclopropyl 3-O-t-C.sub.4 H.sub.9, 4-CH.sub.3                       H         Cyclopropyl 2-C(COOCH.sub.3)═NOCH.sub.3                         H         Cyclopropyl 2,3-Butadienyl                                          H         Cyclopropyl 3,4-Butadienyl                                          CH.sub.3  Cyclopropyl H                                                       CH.sub.3  Cyclopropyl 2-F                                                     CH.sub.3  Cyclopropyl 3-F                                                     CH.sub.3  Cyclopropyl 4-F                                                     CH.sub.3  Cyclopropyl 2,4-F.sub.2                                             CH.sub.3  Cyclopropyl 3,4-F.sub.2                                             CH.sub.3  Cyclopropyl 3,5-F.sub.2                                             CH.sub.3  Cyclopropyl 2-Cl                                                    CH.sub.3  Cyclopropyl 3-Cl                                                    CH.sub.3  Cyclopropyl 4-Cl                                                    CH.sub.3  Cyclopropyl 2,4-Cl.sub.2                                            CH.sub.3  Cyclopropyl 3,4-Cl.sub.2                                            CH.sub.3  Cyclopropyl 3,5-Cl.sub.2                                            CH.sub.3  Cyclopropyl 2-Br                                                    CH.sub.3  Cyclopropyl 3-Br                                                    CH.sub.3  Cyclopropyl 4-Br                                                    CH.sub.3  Cyclopropyl 3,5-Br.sub.2                                            CH.sub.3  Cyclopropyl 3-I                                                     CH.sub.3  Cyclopropyl 4-I                                                     CH.sub.3  Cyclopropyl 3-F, 5-Cl                                               CH.sub.3  Cyclopropyl 3-F, 5-Br                                               CH.sub.3  Cyclopropyl 3-Cl, 5-Br                                              CH.sub.3  Cyclopropyl 3-Br, 4-F                                               CH.sub.3  Cyclopropyl 2-NO.sub.2                                              CH.sub.3  Cyclopropyl 3-NO.sub.2                                              CH.sub.3  Cyclopropyl 4-NO.sub.2                                              CH.sub.3  Cyclopropyl 2-CN                                                    CH.sub.3  Cyclopropyl 3-CN                                                    CH.sub.3  Cyclopropyl 4-CN                                                    CH.sub.3  Cyclopropyl 2-CH.sub.3                                              CH.sub.3  Cyclopropyl 3-CH.sub.3                                              CH.sub.3  Cyclopropyl 4-CH.sub.3                                              CH.sub.3  Cyclopropyl 2,4-(CH.sub.3).sub.2                                    CH.sub.3  Cyclopropyl 2,5-(CH.sub.3).sub.2                                    CH.sub.3  Cyclopropyl 3,4-(CH.sub.3).sub.2                                    CH.sub.3  Cyclopropyl 3,5-(CH.sub.3).sub.2                                    CH.sub.3  Cyclopropyl 2,4,5-(CH.sub.3).sub.3                                  CH.sub.3  Cyclopropyl 2,4,6-(CH.sub.3).sub.3                                  CH.sub.3  Cyclopropyl 3-C.sub.2 H.sub.5                                       CH.sub.3  Cyclopropyl 4-C.sub.2 H.sub.5                                       CH.sub.3  Cyclopropyl 3,4-(C.sub.2 H.sub.5).sub.2                             CH.sub.3  Cyclopropyl 3,5-(C.sub.2 H.sub.5).sub.2                             CH.sub.3  Cyclopropyl 3-n-C.sub.3 H.sub.7                                     CH.sub.3  Cyclopropyl 4-n-C.sub.3 H.sub.7                                     CH.sub.3  Cyclopropyl 3-i-C.sub.3 H.sub.7                                     CH.sub.3  Cyclopropyl 4-i-C.sub.3 H.sub.7                                     CH.sub.3  Cyclopropyl 3-Cyclopropyl                                           CH.sub.3  Cyclopropyl 4-Cyclopropyl                                           CH.sub.3  Cyclopropyl 3-n-C.sub.4 H.sub.9                                     CH.sub.3  Cyclopropyl 4-n-C.sub.4 H.sub.9                                     CH.sub.3  Cyclopropyl 3-t-C.sub.4 H.sub.9                                     CH.sub.3  Cyclopropyl 4-t-C.sub.4 H.sub.9                                     CH.sub.3  Cyclopropyl 3-n-C.sub.6 H.sub.13                                    CH.sub.3  Cyclopropyl 4-n-C.sub.6 H.sub.13                                    CH.sub.3  Cyclopropyl 3-Cyclohexyl                                            CH.sub.3  Cyclopropyl 4-Cyclohexyl                                            CH.sub.3  Cyclopropyl 3-Phenyl                                                CH.sub.3  Cyclopropyl 4-Phenyl                                                CH.sub.3  Cyclopropyl 4-Allyl                                                 CH.sub.3  Cyclopropyl 4-Propargyl                                             CH.sub.3  Cyclopropyl 2-CH.sub.3, 4-C.sub.2 H.sub.5                           CH.sub.3  Cyclopropyl 2-CH.sub.3, 4-i-C.sub.3 H.sub.7                         CH.sub.3  Cyclopropyl 2-CH.sub.3, 4-t-C.sub.4 H.sub.9                         CH.sub.3  Cyclopropyl 2-CH.sub.3, 4-phenyl                                    CH.sub.3  Cyclopropyl 3-CH.sub.3, 4-phenyl                                    CH.sub.3  Cyclopropyl 3-OH                                                    CH.sub.3  Cyclopropyl 4-OH                                                    CH.sub.3  Cyclopropyl 3-OCH.sub.3                                             CH.sub.3  Cyclopropyl 4-OCH.sub.3                                             CH.sub.3  Cyclopropyl 3,4-(OCH.sub.3).sub.2                                   CH.sub.3  Cyclopropyl 3,5-(OCH.sub.3).sub.2                                   CH.sub.3  Cyclopropyl 3,4,5-(OCH.sub.3).sub.3                                 CH.sub.3  Cyclopropyl 4-OC.sub.2 H.sub.5                                      CH.sub.3  Cyclopropyl 4-O-i-C.sub.3 H.sub.7                                   CH.sub.3  Cyclopropyl 3-O-t-C.sub.4 H.sub.9                                   CH.sub.3  Cyclopropyl 4-O-t-C.sub.4 H.sub.9                                   CH.sub.3  Cyclopropyl 4-O-n-C.sub.6 H.sub.13                                  CH.sub.3  Cyclopropyl 3-O-Phenyl                                              CH.sub.3  Cyclopropyl 4-O-Phenyl                                              CH.sub.3  Cyclopropyl 4-O-Allyl                                               CH.sub.3  Cyclopropyl 2-CF.sub.3                                              CH.sub.3  Cyclopropyl 3-CF.sub.3                                              CH.sub.3  Cyclopropyl 4-CF.sub.3                                              CH.sub.3  Cyclopropyl 3,5-(CF.sub.3).sub.2                                    CH.sub.3  Cyclopropyl 4-CH.sub.2 CF.sub.3                                     CH.sub.3  Cyclopropyl 4-C.sub.2 F.sub.5                                       CH.sub.3  Cyclopropyl 4-CF.sub.2 CHF.sub.2                                    CH.sub.3  Cyclopropyl 3-OCF.sub.3                                             CH.sub.3  Cyclopropyl 4-OCF.sub.3                                             CH.sub.3  Cyclopropyl 4-OCH.sub.2 CF.sub.3                                    CH.sub.3  Cyclopropyl 4-OC.sub.2 F.sub.5                                      CH.sub.3  Cyclopropyl 4-OCF.sub.2 CHF.sub.2                                   CH.sub.3  Cyclopropyl 3-CH.sub.2 OCH.sub.3                                    CH.sub.3  Cyclopropyl 4-CH.sub.2 OCH.sub.3                                    CH.sub.3  Cyclopropyl 4-CH.sub.2 --O-t-C.sub.4 H.sub.9                        CH.sub.3  Cyclopropyl 4-CH(OCH.sub.3).sub.2                                   CH.sub.3  Cyclopropyl 4-CH.sub.2 CN                                           CH.sub.3  Cyclopropyl 3-CHO                                                   CH.sub.3  Cyclopropyl 4-CHO                                                   CH.sub.3  Cyclopropyl 3-CO--CH.sub.3                                          CH.sub.3  Cyclopropyl 4-CO--CH.sub.3                                          CH.sub.3  Cyclopropyl 3-COOH                                                  CH.sub.3  Cyclopropyl 4-COOH                                                  CH.sub.3  Cyclopropyl 3-COOCH.sub.3                                           CH.sub.3  Cyclopropyl 4-COOCH.sub.3                                           CH.sub.3  Cyclopropyl 3-COOC.sub.2 H.sub.5                                    CH.sub.3  Cyclopropyl 4-COOC.sub.2 H.sub.5                                    CH.sub.3  Cyclopropyl 3-COO-i-C.sub.3 H.sub.7                                 CH.sub.3  Cyclopropyl 4-COO-i-C.sub.3 H.sub.7                                 CH.sub.3  Cyclopropyl 3-COO-t-C.sub.4 H.sub.9                                 CH.sub.3  Cyclopropyl 4-COO-t-C.sub.4 H.sub.9                                 CH.sub.3  Cyclopropyl 3-COO-n-C.sub.6 H.sub.13                                CH.sub.3  Cyclopropyl 4-COO-n-C.sub.6 H.sub.13                                CH.sub.3  Cyclopropyl 3-CONH.sub.2                                            CH.sub.3  Cyclopropyl 4-CONH.sub.2                                            CH.sub.3  Cyclopropyl 3-CONHCH.sub.3                                          CH.sub.3  Cyclopropyl 4-CONHCH.sub.3                                          CH.sub.3  Cyclopropyl 3-CON(CH.sub.3).sub.2                                   CH.sub.3  Cyclopropyl 4-CON(CH.sub.3).sub.2                                   CH.sub.3  Cyclopropyl 3-CSNH.sub.2                                            CH.sub.3  Cyclopropyl 4-CSNH.sub.2                                            CH.sub.3  Cyclopropyl 3-NH.sub.2                                              CH.sub.3  Cyclopropyl 4-NH.sub.2                                              CH.sub.3  Cyclopropyl 4-NHCH.sub.3                                            CH.sub.3  Cyclopropyl 4-N(CH.sub.3).sub.2                                     CH.sub.3  Cyclopropyl 3-NHCO--CH.sub.3                                        CH.sub.3  Cyclopropyl 4-NHCO--CH.sub.3                                        CH.sub.3  Cyclopropyl 4-NCH.sub.3 --CO--CH.sub.3                              CH.sub.3  Cyclopropyl 4-NHCOOCH.sub.3                                         CH.sub.3  Cyclopropyl 4-NCH.sub.3 --COOCH.sub.3                               CH.sub.3  Cyclopropyl 3-OCO--CH.sub.3                                         CH.sub.3  Cyclopropyl 4-OCO--CH.sub.3                                         CH.sub.3  Cyclopropyl 4-OCO-t-C.sub.4 H.sub.9                                 CH.sub.3  Cyclopropyl 4-SH                                                    CH.sub.3  Cyclopropyl 4-SCH.sub.3                                             CH.sub.3  Cyclopropyl 4-S-t-C.sub.4 H.sub.9                                   CH.sub.3  Cyclopropyl 4-SO--CH.sub.3                                          CH.sub.3  Cyclopropyl 4-SO.sub.2 --CH.sub.3                                   CH.sub.3  Cyclopropyl 4-C(CH.sub.3)═NCH.sub.3                             CH.sub.3  Cyclopropyl 4-C(SCH.sub.3)═NOCH.sub.3                           CH.sub.3  Cyclopropyl 4-C(OCH.sub.3)═NOCH.sub.3                           CH.sub.3  Cyclopropyl 3-CH═NOCH.sub.3                                     CH.sub.3  Cyclopropyl 4-CH═NOCH.sub.3                                     CH.sub.3  Cyclopropyl 3-C(CH.sub.3)═NOCH.sub.3                            CH.sub.3  Cyclopropyl 4-C(CH.sub.3)═NOCH.sub.3                            CH.sub.3  Cyclopropyl 4-C(CH.sub.3)═NOC.sub.2 H.sub.5                     CH.sub.3  Cyclopropyl 4-C(CH.sub.3)═NO-n-C.sub.3 H.sub.7                  CH.sub.3  Cyclopropyl 4-C(CH.sub.3)═NO-i-C.sub.3 H.sub.7                  CH.sub.3  Cyclopropyl 4-C(CH.sub.3)═NO-n-C.sub.4 H.sub.9                  CH.sub.3  Cyclopropyl 4-C(CH.sub.3)═NO-t-C.sub.4 H.sub.9                  CH.sub.3  Cyclopropyl 4-C(CH.sub.3)═NO-n-C.sub.5 H.sub.11                 CH.sub.3  Cyclopropyl 4-C(CH.sub.3)═NO-n-C.sub.6 H.sub.13                 CH.sub.3  Cyclopropyl 2-Cl, 4-CH.sub.3                                        CH.sub.3  Cyclopropyl 3-Cl, 5-CH.sub.3                                        CH.sub.3  Cyclopropyl 2-CH.sub.3, 4-Cl                                        CH.sub.3  Cyclopropyl 3-CH.sub.3, 4-Cl                                        CH.sub.3  Cyclopropyl 3-F, 5-CH.sub.3                                         CH.sub.3  Cyclopropyl 3-Br, 5-CH.sub.3                                        CH.sub.3  Cyclopropyl 3-Cl, 5-NO.sub.2                                        CH.sub.3  Cyclopropyl 3-NO.sub.2, 4-Cl                                        CH.sub.3  Cyclopropyl 3-Cl, 4-OCH.sub.3                                       CH.sub.3  Cyclopropyl 3-OCH.sub.3, 4-Cl                                       CH.sub.3  Cyclopropyl 3-Cl, 5-CF.sub.3                                        CH.sub.3  Cyclopropyl 3-Cl, 5-OCF.sub.3                                       CH.sub.3  Cyclopropyl 3-F, 5-CF.sub.3                                         CH.sub.3  Cyclopropyl 2-CH.sub.3, 4-CN                                        CH.sub.3  Cyclopropyl 2-CH.sub.3, 4-OCH.sub.3                                 CH.sub.3  Cyclopropyl 2-CH.sub.3, 4-CF.sub.3                                  CH.sub.3  Cyclopropyl 2-CH.sub.3, 4-C(CH.sub.3)═NOCH.sub.3                CH.sub.3  Cyclopropyl 3-CH.sub.3, 4-C(CH.sub.3)═NOCH.sub.3                CH.sub.3  Cyclopropyl 2-OH, 5-CH.sub.3                                        CH.sub.3  Cyclopropyl 3-CH.sub.3, 4-O-t-C.sub.4 H.sub.9                       CH.sub.3  Cyclopropyl 2-C(COOCH.sub.3)═NOCH.sub.3                         CH.sub.3  Cyclopropyl                                                         CH.sub.3  Cyclopropyl                                                         H         C.sub.2 H.sub.5                                                                           H                                                       H         C.sub.2 H.sub.5                                                                           2-F                                                     H         C.sub.2 H.sub.5                                                                           3-F                                                     H         C.sub.2 H.sub.5                                                                           4-F                                                     H         C.sub.2 H.sub.5                                                                           2,3-F.sub.2                                             H         C.sub.2 H.sub.5                                                                           2,4-F.sub.2                                             H         C.sub.2 H.sub.5                                                                           2,5-F.sub.2                                             H         C.sub.2 H.sub.5                                                                           2,6-F.sub.2                                             H         C.sub.2 H.sub.5                                                                           3,4-F.sub.2                                             H         C.sub.2 H.sub.5                                                                           3,5-F.sub.2                                             H         C.sub.2 H.sub.5                                                                           2-Cl                                                    H         C.sub.2 H.sub.5                                                                           3-Cl                                                    H         C.sub.2 H.sub.5                                                                           4-Cl                                                    H         C.sub.2 H.sub.5                                                                           2,4-Cl.sub.2                                            H         C.sub.2 H.sub.5                                                                           2,5-Cl.sub.2                                            H         C.sub.2 H.sub.5                                                                           3,4-Cl.sub.2                                            H         C.sub.2 H.sub.5                                                                           3,5-Cl.sub.2                                            H         C.sub.2 H.sub.5                                                                           2-Br                                                    H         C.sub.2 H.sub.5                                                                           3-Br                                                    H         C.sub.2 H.sub.5                                                                           4-Br                                                    H         C.sub.2 H.sub.5                                                                           2,4-Br.sub.2                                            H         C.sub.2 H.sub.5                                                                           3,4-Br.sub.2                                            H         C.sub.2 H.sub.5                                                                           3,5-Br.sub.2                                            H         C.sub.2 H.sub.5                                                                           2-I                                                     H         C.sub.2 H.sub.5                                                                           3-I                                                     H         C.sub.2 H.sub.5                                                                           4-I                                                     H         C.sub.2 H.sub.5                                                                           2-F, 4-Cl                                               H         C.sub.2 H.sub.5                                                                           2-F, 5-Cl                                               H         C.sub.2 H.sub.5                                                                           2-F, 4-Br                                               H         C.sub.2 H.sub.5                                                                           2-F, 5-Br                                               H         C.sub.2 H.sub.5                                                                           2-Cl, 4-Br                                              H         C.sub.2 H.sub.5                                                                           2-Cl, 5-Br                                              H         C.sub.2 H.sub.5                                                                           3-F, 4-Cl                                               H         C.sub.2 H.sub.5                                                                           3-F, 5-Cl                                               H         C.sub.2 H.sub.5                                                                           3-F, 4-Br                                               H         C.sub.2 H.sub.5                                                                           3-F, 5-Br                                               H         C.sub.2 H.sub.5                                                                           3-Cl, 4-Br                                              H         C.sub.2 H.sub.5                                                                           3-Cl, 5-Br                                              H         C.sub.2 H.sub.5                                                                           3-Cl, 4-F                                               H         C.sub.2 H.sub.5                                                                           3-Br, 4-F                                               H         C.sub.2 H.sub.5                                                                           3-Br, 4-Cl                                              H         C.sub.2 H.sub.5                                                                           2-NO.sub.2                                              H         C.sub.2 H.sub.5                                                                           3-NO.sub.2                                              H         C.sub.2 H.sub.5                                                                           4-NO.sub.2                                              H         C.sub.2 H.sub.5                                                                           2-CN                                                    H         C.sub.2 H.sub.5                                                                           3-CN                                                    H         C.sub.2 H.sub.5                                                                           4-CN                                                    H         C.sub.2 H.sub.5                                                                           2-CH.sub.3                                              H         C.sub.2 H.sub.5                                                                           3-CH.sub.3                                              H         C.sub.2 H.sub.5                                                                           4-CH.sub.3                                              H         C.sub.2 H.sub.5                                                                           2,3-(CH.sub.3).sub.2                                    H         C.sub.2 H.sub.5                                                                           2,4-(CH.sub.3).sub.2                                    H         C.sub.2 H.sub.5                                                                           2,5-(CH.sub.3).sub.2                                    H         C.sub.2 H.sub.5                                                                           2,6-(CH.sub.3).sub.2                                    H         C.sub.2 H.sub.5                                                                           3,4-(CH.sub.3).sub.2                                    H         C.sub.2 H.sub.5                                                                           3,5-(CH.sub.3).sub.2                                    H         C.sub.2 H.sub.5                                                                           2,4,5-(CH.sub.3).sub.3                                  H         C.sub.2 H.sub.5                                                                           2,4,6-(CH.sub.3).sub.3                                  H         C.sub.2 H.sub.5                                                                           3,4,5-(CH.sub.3).sub.3                                  H         C.sub.2 H.sub.5                                                                           2-C.sub.2 H.sub.5                                       H         C.sub.2 H.sub.5                                                                           3-C.sub.2 H.sub.5                                       H         C.sub.2 H.sub.5                                                                           4-C.sub.2 H.sub.5                                       H         C.sub.2 H.sub.5                                                                           3,4-(C.sub.2 H.sub.5).sub.2                             H         C.sub.2 H.sub.5                                                                           3,5-(C.sub.2 H.sub.5).sub.2                             H         C.sub.2 H.sub.5                                                                           3-n-C.sub.3 H.sub.7                                     H         C.sub.2 H.sub.5                                                                           4-n-C.sub.3 H.sub.7                                     H         C.sub.2 H.sub.5                                                                           3,4-(n-C.sub.3 H.sub.7).sub.2                           H         C.sub.2 H.sub.5                                                                           3,5-(n-C.sub.3 H.sub.7).sub.2                           H         C.sub.2 H.sub.5                                                                           3-i-C.sub.3 H.sub.7                                     H         C.sub.2 H.sub.5                                                                           4-i-C.sub.3 H.sub.7                                     H         C.sub.2 H.sub.5                                                                           3,4-(i-C.sub.3 H.sub.7).sub.2                           H         C.sub.2 H.sub.5                                                                           3,5-(i-C.sub.3 H.sub.7).sub.2                           H         C.sub.2 H.sub.5                                                                           3-Cyclopropyl                                           H         C.sub.2 H.sub.5                                                                           4-Cyclopropyl                                           H         C.sub.2 H.sub.5                                                                           3-n-C.sub.4 H.sub.9                                     H         C.sub.2 H.sub.5                                                                           4-n-C.sub.4 H.sub.9                                     H         C.sub.2 H.sub.5                                                                           3,4-(n-C.sub.4 H.sub.9).sub.2                           H         C.sub.2 H.sub.5                                                                           3,5-(n-C.sub.4 H.sub.9).sub.2                           H         C.sub.2 H.sub.5                                                                           3-s-C.sub.4 H.sub.9                                     H         C.sub.2 H.sub.5                                                                           4-s-C.sub.4 H.sub.9                                     H         C.sub.2 H.sub.5                                                                           3-i-C.sub.4 H.sub.9                                     H         C.sub.2 H.sub.5                                                                           4-i-C.sub.4 H.sub.9                                     H         C.sub.2 H.sub.5                                                                           3-t-C.sub.4 H.sub.9                                     H         C.sub.2 H.sub.5                                                                           4-t-C.sub.4 H.sub.9                                     H         C.sub.2 H.sub.5                                                                           3,4-(t-C.sub.4 H.sub.9).sub.2                           H         C.sub.2 H.sub.5                                                                           3,5-(t-C.sub.4 H.sub.9).sub.2                           H         C.sub.2 H.sub.5                                                                           3-n-C.sub.5 H.sub.11                                    H         C.sub.2 H.sub.5                                                                           4-n-C.sub.5 H.sub.11                                    H         C.sub.2 H.sub.5                                                                           3-n-C.sub.6 H.sub.13                                    H         C.sub.2 H.sub.5                                                                           4-n-C.sub.6 H.sub.13                                    H         C.sub.2 H.sub.5                                                                           3-Cyclohexyl                                            H         C.sub.2 H.sub.5                                                                           4-Cyclohexyl                                            H         C.sub.2 H.sub.5                                                                           3-Phenyl                                                H         C.sub.2 H.sub.5                                                                           4-Phenyl                                                H         C.sub.2 H.sub.5                                                                           3-Vinyl                                                 H         C.sub.2 H.sub.5                                                                           4-Vinyl                                                 H         C.sub.2 H.sub.5                                                                           3-Allyl                                                 H         C.sub.2 H.sub.5                                                                           4-Allyl                                                 H         C.sub.2 H.sub.5                                                                           3-Propargyl                                             H         C.sub.2 H.sub.5                                                                           4-Propargyl                                             H         C.sub.2 H.sub.5                                                                           3-(Propen-2-yl)                                         H         C.sub.2 H.sub.5                                                                           4-(Propen-2-yl)                                         H         C.sub.2 H.sub.5                                                                           2-CH.sub.3, 4-C.sub.2 H.sub.5                           H         C.sub.2 H.sub.5                                                                           2-CH.sub.3, 5-C.sub.2 H.sub.5                           H         C.sub.2 H.sub.5                                                                           2-CH.sub.3, 4-n-C.sub.3 H.sub.7                         H         C.sub.2 H.sub.5                                                                           2-CH.sub.3, 5-n-C.sub.3 H.sub.7                         H         C.sub.2 H.sub.5                                                                           2-CH.sub.3, 4-i-C.sub.3 H.sub.7                         H         C.sub.2 H.sub.5                                                                           2-CH.sub.3, 5-i-C.sub.3 H.sub.7                         H         C.sub.2 H.sub.5                                                                           2-CH.sub.3, 4-n-C.sub.4 H.sub.9                         H         C.sub.2 H.sub.5                                                                           2-CH.sub.3, 4-s-C.sub.4 H.sub.9                         H         C.sub.2 H.sub.5                                                                           2-CH.sub.3, 4-i-C.sub.4 H.sub.9                         H         C.sub.2 H.sub.5                                                                           2-CH.sub.3, 4-t-C.sub.4 H.sub.9                         H         C.sub.2 H.sub.5                                                                           2-CH.sub.3, 4-phenyl                                    H         C.sub.2 H.sub.5                                                                           2-CH.sub.3, 5-phenyl                                    H         C.sub.2 H.sub.5                                                                           2-CH.sub.3, 4-vinyl                                     H         C.sub.2 H.sub.5                                                                           2-CH.sub.3, 4-allyl                                     H         C.sub.2 H.sub.5                                                                           2-CH.sub.3, 4-propargyl                                 H         C.sub.2 H.sub.5                                                                           2-CH.sub.3, 4-(propen-2-yl)                             H         C.sub.2 H.sub.5                                                                           3-CH.sub.3, 4-C.sub.2 H.sub.5                           H         C.sub.2 H.sub.5                                                                           3-CH.sub.3, 5-C.sub.2 H.sub.5                           H         C.sub.2 H.sub.5                                                                           3-CH.sub.3, 4-n-C.sub.3 H.sub.7                         H         C.sub.2 H.sub.5                                                                           3-CH.sub.3, 5-n-C.sub.3 H.sub.7                         H         C.sub.2 H.sub.5                                                                           3-CH.sub.3, 4-i-C.sub.3 H.sub.7                         H         C.sub.2 H.sub.5                                                                           3-CH.sub.3, 5-i-C.sub.3 H.sub.7                         H         C.sub.2 H.sub.5                                                                           3-CH.sub.3, 4-cyclopropyl                               H         C.sub.2 H.sub.5                                                                           3-CH.sub.3, 4-t-C.sub.4 H.sub.9                         H         C.sub.2 H.sub.5                                                                           3-CH.sub.3, 5-t-C.sub.4 H.sub.9                         H         C.sub.2 H.sub.5                                                                           3-CH.sub.3, 4-phenyl                                    H         C.sub.2 H.sub.5                                                                           3-CH.sub.3, 5-phenyl                                    H         C.sub.2 H.sub.5                                                                           3-CH.sub.3, 4-vinyl                                     H         C.sub.2 H.sub.5                                                                           3-CH.sub.3, 4-allyl                                     H         C.sub.2 H.sub.5                                                                           3-CH.sub.3, 4-propargyl                                 H         C.sub.2 H.sub.5                                                                           3-CH.sub.3, 4-propen-2-yl                               H         C.sub.2 H.sub.5                                                                           3-C.sub.2 H.sub.5, 4-CH.sub.3                           H         C.sub.2 H.sub.5                                                                           3-i-C.sub.3 H.sub.7, 4-CH.sub.3                         H         C.sub.2 H.sub.5                                                                           3-t-C.sub.4 H.sub.9, 4-CH.sub.3                         H         C.sub.2 H.sub.5                                                                           3-Phenyl, 4-CH.sub.3                                    H         C.sub.2 H.sub.5                                                                           2-OH                                                    H         C.sub.2 H.sub.5                                                                           3-OH                                                    H         C.sub.2 H.sub.5                                                                           4-OH                                                    H         C.sub.2 H.sub.5                                                                           2-OCH.sub.3                                             H         C.sub.2 H.sub.5                                                                           3-OCH.sub.3                                             H         C.sub.2 H.sub.5                                                                           4-OCH.sub.3                                             H         C.sub.2 H.sub.5                                                                           2,3-(OCH.sub.3).sub.2                                   H         C.sub.2 H.sub.5                                                                           2,4-(OCH.sub.3).sub.2                                   H         C.sub.2 H.sub.5                                                                           2,5-(OCH.sub.3).sub.2                                   H         C.sub.2 H.sub.5                                                                           3,4-(OCH.sub.3).sub.2                                   H         C.sub.2 H.sub.5                                                                           3,5-(OCH.sub.3).sub.2                                   H         C.sub.2 H.sub.5                                                                           3,4,5-(OCH.sub.3).sub.3                                 H         C.sub.2 H.sub.5                                                                           3-OC.sub.2 H.sub.5                                      H         C.sub.2 H.sub.5                                                                           4-OC.sub.2 H.sub.5                                      H         C.sub.2 H.sub.5                                                                           3,4-(OC.sub.2 H.sub.5).sub.2                            H         C.sub.2 H.sub.5                                                                           3,5-(OC.sub.2 H.sub.5).sub.2                            H         C.sub.2 H.sub.5                                                                           3-O-n-C.sub.3 H.sub.7                                   H         C.sub.2 H.sub.5                                                                           4-O-n-C.sub.3 H.sub.7                                   H         C.sub.2 H.sub.5                                                                           3-O-i-C.sub.3 H.sub.7                                   H         C.sub.2 H.sub.5                                                                           4-O-i-C.sub.3 H.sub.7                                   H         C.sub.2 H.sub.5                                                                           3-O-Cyclopropyl                                         H         C.sub.2 H.sub.5                                                                           4-O-Cyclopropyl                                         H         C.sub.2 H.sub.5                                                                           3-O-n-C.sub.4 H.sub.9                                   H         C.sub.2 H.sub.5                                                                           4-O-n-C.sub.4 H.sub.9                                   H         C.sub.2 H.sub.5                                                                           3-O-s-C.sub.4 H.sub.9                                   H         C.sub.2 H.sub.5                                                                           4-O-s-C.sub.4 H.sub.9                                   H         C.sub.2 H.sub.5                                                                           3-O-i-C.sub.4 H.sub.9                                   H         C.sub.2 H.sub.5                                                                           4-O-i-C.sub.4 H.sub.9                                   H         C.sub.2 H.sub.5                                                                           3-O-t-C.sub.4 H.sub.9                                   H         C.sub.2 H.sub.5                                                                           4-O-t-C.sub.4 H.sub.9                                   H         C.sub.2 H.sub.5                                                                           3-O-n-C.sub.5 H.sub.11                                  H         C.sub.2 H.sub.5                                                                           4-O-n-C.sub.5 H.sub.11                                  H         C.sub.2 H.sub.5                                                                           3-O-n-C.sub.6 H.sub.13                                  H         C.sub.2 H.sub.5                                                                           4-O-n-C.sub.6 H.sub.13                                  H         C.sub.2 H.sub.5                                                                           3-O-Cyclohexyl                                          H         C.sub.2 H.sub.5                                                                           4-O-Cyclohexyl                                          H         C.sub.2 H.sub.5                                                                           3-O-Phenyl                                              H         C.sub.2 H.sub.5                                                                           4-O-Phenyl                                              H         C.sub.2 H.sub.5                                                                           3-O-Allyl                                               H         C.sub.2 H.sub.5                                                                           4-O-Allyl                                               H         C.sub.2 H.sub.5                                                                           2-CF.sub.3                                              H         C.sub.2 H.sub.5                                                                           3-CF.sub.3                                              H         C.sub.2 H.sub.5                                                                           4-CF.sub.3                                              H         C.sub.2 H.sub.5                                                                           2,4-(CF.sub.3).sub.2                                    H         C.sub.2 H.sub.5                                                                           3,5-(CF.sub.3).sub.2                                    H         C.sub.2 H.sub.5                                                                           3-CF.sub.2 Cl                                           H         C.sub.2 H.sub.5                                                                           4-CF.sub.2 Cl                                           H         C.sub.2 H.sub.5                                                                           3-CFCl.sub.2                                            H         C.sub.2 H.sub.5                                                                           4-CFCl.sub.2                                            H         C.sub.2 H.sub.5                                                                           3-CCl.sub.3                                             H         C.sub.2 H.sub.5                                                                           4-CCl.sub.3                                             H         C.sub.2 H.sub.5                                                                           3-CH.sub.2 CH.sub.2 F                                   H         C.sub.2 H.sub.5                                                                           4-CH.sub.2 CH.sub.2 F                                   H         C.sub.2 H.sub.5                                                                           3-CH.sub.2 CF.sub.3                                     H         C.sub.2 H.sub.5                                                                           4-CH.sub.2 CF.sub.3                                     H         C.sub.2 H.sub.5                                                                           3-C.sub.2 F.sub.5                                       H         C.sub.2 H.sub.5                                                                           4-C.sub.2 F.sub.5                                       H         C.sub.2 H.sub.5                                                                           3-CHCl.sub.2                                            H         C.sub.2 H.sub.5                                                                           4-CHCl.sub.2                                            H         C.sub.2 H.sub.5                                                                           3-CH.sub.2 Cl                                           H         C.sub.2 H.sub.5                                                                           4-CH.sub.2 Cl                                           H         C.sub.2 H.sub.5                                                                           3-CF.sub.2 CHF.sub.2                                    H         C.sub.2 H.sub.5                                                                           4-CF.sub.2 CHF.sub.2                                    H         C.sub.2 H.sub.5                                                                           3-CH.sub.2 CH.sub.2 Cl                                  H         C.sub.2 H.sub.5                                                                           4-CH.sub.2 CH.sub.2 Cl                                  H         C.sub.2 H.sub.5                                                                           2-OCF.sub.3                                             H         C.sub.2 H.sub.5                                                                           3-OCF.sub.3                                             H         C.sub.2 H.sub.5                                                                           4-OCF.sub.3                                             H         C.sub.2 H.sub.5                                                                           3-OCHF.sub.2                                            H         C.sub.2 H.sub.5                                                                           4-OCHF.sub.2                                            H         C.sub.2 H.sub.5                                                                           3-OC.sub.2 F.sub.5                                      H         C.sub.2 H.sub.5                                                                           4-OC.sub.2 F.sub.5                                      H         C.sub.2 H.sub.5                                                                           3-OCF.sub.2 CHF.sub.2                                   H         C.sub.2 H.sub.5                                                                           4-OCF.sub.2 CHF.sub.2                                   H         C.sub.2 H.sub.5                                                                           3-CH.sub.2 OCH.sub.3                                    H         C.sub.2 H.sub.5                                                                           4-CH.sub.2 OCH.sub.3                                    H         C.sub.2 H.sub.5                                                                           3-CH.sub.2 O-t-C.sub.4 H.sub.9                          H         C.sub.2 H.sub.5                                                                           4-CH.sub.2 O-t-C.sub.4 H.sub.9                          H         C.sub.2 H.sub.5                                                                           3-C(CH.sub.3)(OCH.sub.3).sub.2                          H         C.sub.2 H.sub.5                                                                           4-C(CH.sub.3)(OCH.sub.3).sub.2                          H         C.sub.2 H.sub.5                                                                           3-CH(OCH.sub.3).sub.2                                   H         C.sub.2 H.sub.5                                                                           4-CH(OCH.sub.3).sub.2                                   H         C.sub.2 H.sub.5                                                                           3-CH.sub.2 CN                                           H         C.sub.2 H.sub.5                                                                           4-CH.sub.2 CN                                           H         C.sub.2 H.sub.5                                                                           3-CHO                                                   H         C.sub.2 H.sub.5                                                                           4-CHO                                                   H         C.sub.2 H.sub.5                                                                           3-CO--CH.sub.3                                          H         C.sub.2 H.sub.5                                                                           4-CO--CH.sub.3                                          H         C.sub.2 H.sub.5                                                                           3-CO--C.sub.2 H.sub.5                                   H         C.sub.2 H.sub.5                                                                           4-CO--C.sub.2 H.sub.5                                   H         C.sub.2 H.sub.5                                                                           2-COOH                                                  H         C.sub.2 H.sub.5                                                                           3-COOH                                                  H         C.sub.2 H.sub.5                                                                           4-COOH                                                  H         C.sub.2 H.sub.5                                                                           3-COOCH.sub.3                                           H         C.sub.2 H.sub.5                                                                           4-COOCH.sub.3                                           H         C.sub.2 H.sub.5                                                                           3-COOC.sub.2 H.sub.5                                    H         C.sub.2 H.sub.5                                                                           4-COOC.sub.2 H.sub.5                                    H         C.sub.2 H.sub.5                                                                           3-COO-n-C.sub.3 H.sub.7                                 H         C.sub.2 H.sub.5                                                                           4-COO-n-C.sub.3 H.sub.7                                 H         C.sub.2 H.sub.5                                                                           3-COO-i-C.sub.3 H.sub.7                                 H         C.sub.2 H.sub.5                                                                           4-COO-i-C.sub.3 H.sub.7                                 H         C.sub.2 H.sub.5                                                                           3-COO-n-C.sub.4 H.sub.9                                 H         C.sub.2 H.sub.5                                                                           4-COO-n-C.sub.4 H.sub.9                                 H         C.sub.2 H.sub.5                                                                           3-COO-s-C.sub.4 H.sub.9                                 H         C.sub.2 H.sub.5                                                                           4-COO-s-C.sub.4 H.sub.9                                 H         C.sub.2 H.sub.5                                                                           3-COO-i-C.sub.4 H.sub.9                                 H         C.sub.2 H.sub.5                                                                           4-COO-i-C.sub.4 H.sub.9                                 H         C.sub.2 H.sub.5                                                                           3-COO-t-C.sub.4 H.sub.9                                 H         C.sub.2 H.sub.5                                                                           4-COO-t-C.sub.4 H.sub.9                                 H         C.sub.2 H.sub.5                                                                           3-COO-n-C.sub.5 H.sub.11                                H         C.sub.2 H.sub.5                                                                           4-COO-n-C.sub.5 H.sub.11                                H         C.sub.2 H.sub.5                                                                           3-COO-n-C.sub.6 H.sub.13                                H         C.sub.2 H.sub.5                                                                           4-COO-n-C.sub.6 H.sub.13                                H         C.sub.2 H.sub.5                                                                           2-CONH.sub.2                                            H         C.sub.2 H.sub.5                                                                           3-CONH.sub.2                                            H         C.sub.2 H.sub.5                                                                           4-CONH.sub.2                                            H         C.sub.2 H.sub.5                                                                           3-CONHCH.sub.3                                          H         C.sub.2 H.sub.5                                                                           4-CONHCH.sub.3                                          H         C.sub.2 H.sub.5                                                                           3-CON(CH.sub.3).sub.2                                   H         C.sub.2 H.sub.5                                                                           4-CON(CH.sub.3).sub.2                                   H         C.sub.2 H.sub.5                                                                           3-CON(C.sub.2 H.sub.5).sub.2                            H         C.sub.2 H.sub.5                                                                           4-CON(C.sub.2 H.sub.5).sub.2                            H         C.sub.2 H.sub.5                                                                           2-CSNH.sub.2                                            H         C.sub.2 H.sub.5                                                                           3-CSNH.sub.2                                            H         C.sub.2 H.sub.5                                                                           4-CSNH.sub.2                                            H         C.sub.2 H.sub.5                                                                           2-NH.sub.2                                              H         C.sub.2 H.sub.5                                                                           3-NH.sub.2                                              H         C.sub.2 H.sub.5                                                                           4-NH.sub.2                                              H         C.sub.2 H.sub.5                                                                           3-NHCH.sub.3                                            H         C.sub.2 H.sub.5                                                                           4-NHCH.sub.3                                            H         C.sub.2 H.sub.5                                                                           3-N(CH.sub.3).sub.2                                     H         C.sub.2 H.sub.5                                                                           4-N(CH.sub.3).sub.2                                     H         C.sub.2 H.sub.5                                                                           3-NHCO--CH.sub.3                                        H         C.sub.2 H.sub.5                                                                           4-NHCO--CH.sub.3                                        H         C.sub.2 H.sub.5                                                                           3-NCH.sub.3 --CO--CH.sub.3                              H         C.sub.2 H.sub.5                                                                           4-NCH.sub.3 --CO--CH.sub.3                              H         C.sub.2 H.sub.5                                                                           3-NHCOOCH.sub.3                                         H         C.sub.2 H.sub.5                                                                           4-NHCOOCH.sub.3                                         H         C.sub.2 H.sub.5                                                                           3-NCH.sub.3 --COOCH.sub.3                               H         C.sub.2 H.sub.5                                                                           4-NCH.sub.3 --COOCH.sub.3                               H         C.sub.2 H.sub.5                                                                           3-OCO--CH.sub.3                                         H         C.sub.2 H.sub.5                                                                           4-OCO--CH.sub.3                                         H         C.sub.2 H.sub.5                                                                           3-OCO-t-C.sub.4 H.sub.9                                 H         C.sub.2 H.sub.5                                                                           4-OCO-t-C.sub.4 H.sub.9                                 H         C.sub.2 H.sub.5                                                                           3-SH                                                    H         C.sub.2 H.sub.5                                                                           4-SH                                                    H         C.sub.2 H.sub.5                                                                           3-SCH.sub.3                                             H         C.sub.2 H.sub.5                                                                           4-SCH.sub.3                                             H         C.sub.2 H.sub.5                                                                           3-S-t-C.sub.4 H.sub.9                                   H         C.sub.2 H.sub.5                                                                           4-S-t-C.sub.4 H.sub.9                                   H         C.sub.2 H.sub.5                                                                           3-SO--CH.sub.3                                          H         C.sub.2 H.sub.5                                                                           4-SO--CH.sub.3                                          H         C.sub.2 H.sub.5                                                                           3-SO.sub.2 CH.sub.3                                     H         C.sub.2 H.sub.5                                                                           4-SO.sub.2 CH.sub.3                                     H         C.sub.2 H.sub.5                                                                           3-CH═NCH.sub.3                                      H         C.sub.2 H.sub.5                                                                           4-CH═NCH.sub.3                                      H         C.sub.2 H.sub.5                                                                           3-C(CH.sub.3)═NCH.sub.3                             H         C.sub.2 H.sub.5                                                                           4-C(CH.sub.3)═NCH.sub.3                             H         C.sub.2 H.sub.5                                                                           3-C(SCH.sub.3)═NOCH.sub.3                           H         C.sub.2 H.sub.5                                                                           4-C(SCH.sub.3)═NOCH.sub.3                           H         C.sub.2 H.sub.5                                                                           3-C(OCH.sub.3)═NOCH.sub.3                           H         C.sub.2 H.sub.5                                                                           4-C(OCH.sub.3)═NOCH.sub.3                           H         C.sub.2 H.sub.5                                                                           3-C(NH.sub.2)═NOCH.sub.3                            H         C.sub.2 H.sub.5                                                                           4-C(NH.sub.2)═NOCH.sub.3                            H         C.sub.2 H.sub.5                                                                           3-C(NHCH.sub.3)═NOCH.sub.3                          H         C.sub.2 H.sub.5                                                                           4-C(NHCH.sub.3)═NOCH.sub.3                          H         C.sub.2 H.sub.5                                                                           3-CH═NOCH.sub.3                                     H         C.sub.2 H.sub.5                                                                           4-CH═NOCH.sub.3                                     H         C.sub.2 H.sub.5                                                                           3-C(CH.sub.3)═NOCH.sub.3                            H         C.sub.2 H.sub.5                                                                           4-C(CH.sub.3)═NOCH.sub.3                            H         C.sub.2 H.sub.5                                                                           3-C(CH.sub.3)═NOC.sub.2 H.sub.5                     H         C.sub.2 H.sub.5                                                                           4-C(CH.sub.3)═NOC.sub.2 H.sub.5                     H         C.sub.2 H.sub.5                                                                           3-C(CH.sub.3)═NO-n-C.sub.3 H.sub.7                  H         C.sub.2 H.sub.5                                                                           4-C(CH.sub.3)═NO-n-C.sub.3 H.sub.7                  H         C.sub.2 H.sub.5                                                                           3-C(CH.sub.3)═NO-i-C.sub.3 H.sub.7                  H         C.sub.2 H.sub.5                                                                           4-C(CH.sub.3)═NO-i-C.sub.3 H.sub.7                  H         C.sub.2 H.sub.5                                                                           3-C(CH.sub.3)═NO-n-C.sub.4 H.sub.9                  H         C.sub.2 H.sub.5                                                                           4-C(CH.sub.3)═NO-n-C.sub.4 H.sub.9                  H         C.sub.2 H.sub.5                                                                           3-C(CH.sub.3)═NO-s-C.sub.4 H.sub.9                  H         C.sub.2 H.sub.5                                                                           4-C(CH.sub.3)═NO-s-C.sub.4 H.sub.9                  H         C.sub.2 H.sub.5                                                                           3-C(CH.sub.3)═NO-i-C.sub.4 H.sub.9                  H         C.sub.2 H.sub.5                                                                           4-C(CH.sub.3)═NO-i-C.sub.4 H.sub.9                  H         C.sub.2 H.sub.5                                                                           3-C(CH.sub.3)═NO-t-C.sub.4 H.sub.9                  H         C.sub.2 H.sub.5                                                                           4-C(CH.sub.3)═NO-t-C.sub.4 H.sub.9                  H         C.sub.2 H.sub.5                                                                           3-C(CH.sub.3)═NO-n-C.sub.5 H.sub.11                 H         C.sub.2 H.sub.5                                                                           4-C(CH.sub.3)═NO-n-C.sub.5 H.sub.11                 H         C.sub.2 H.sub.5                                                                           3-C(CH.sub.3)═NO-n-C.sub.6 H.sub.13                 H         C.sub.2 H.sub.5                                                                           4-C(CH.sub.3)═NO-n-C.sub.6 H.sub.13                 H         C.sub.2 H.sub.5                                                                           2-Cl, 4-CH.sub.3                                        H         C.sub.2 H.sub.5                                                                           2-Cl, 5-CH.sub.3                                        H         C.sub.2 H.sub.5                                                                           3-Cl, 4-CH.sub.3                                        H         C.sub.2 H.sub.5                                                                           3-Cl, 5-CH.sub.3                                        H         C.sub.2 H.sub.5                                                                           2-CH.sub.3, 4-Cl                                        H         C.sub.2 H.sub.5                                                                           2-CH.sub.3, 5-Cl                                        H         C.sub.2 H.sub.5                                                                           3-CH.sub.3, 4-Cl                                        H         C.sub.2 H.sub.5                                                                           3-Cl, 5-t-C.sub.4 H.sub.9                               H         C.sub.2 H.sub.5                                                                           2-Cl, 4-t-C.sub.4 H.sub.9                               H         C.sub.2 H.sub.5                                                                           2-F, 4-CH.sub.3                                         H         C.sub.2 H.sub.5                                                                           3-F, 4-CH.sub.3                                         H         C.sub.2 H.sub.5                                                                           3-F, 5-CH.sub.3                                         H         C.sub.2 H.sub.5                                                                           2-CH.sub.3, 4-F                                         H         C.sub.2 H.sub.5                                                                           3-CH.sub.3, 4-F                                         H         C.sub.2 H.sub.5                                                                           2-F, 4-t-C.sub.4 H.sub.9                                H         C.sub.2 H.sub.5                                                                           3-F, 4-t-C.sub.4 H.sub.9                                H         C.sub.2 H.sub.5                                                                           2-F, 4-OCH.sub.3                                        H         C.sub.2 H.sub.5                                                                           2-Br, 4-CH.sub.3                                        H         C.sub.2 H.sub.5                                                                           3-Br, 4-CH.sub.3                                        H         C.sub.2 H.sub.5                                                                           3-Br, 5-CH.sub.3                                        H         C.sub.2 H.sub.5                                                                           2-CH.sub.3, 4-Br                                        H         C.sub.2 H.sub.5                                                                           3-CH.sub.3, 4-Br                                        H         C.sub.2 H.sub.5                                                                           2-Br, 4-t-C.sub.4 H.sub.9                               H         C.sub.2 H.sub.5                                                                           2-Cl, 4-NO.sub.2                                        H         C.sub.2 H.sub.5                                                                           3-Cl, 4-NO.sub.2                                        H         C.sub.2 H.sub.5                                                                           3-Cl, 5-NO.sub.2                                        H         C.sub.2 H.sub.5                                                                           3-NO.sub.2, 4-Cl                                        H         C.sub.2 H.sub.5                                                                           3-Cl, 4-OCH                                             H         C.sub.2 H.sub.5                                                                           3-OCH.sub.3, 4-Cl                                       H         C.sub.2 H.sub.5                                                                           2-Cl, 5-CF.sub.3                                        H         C.sub.2 H.sub.5                                                                           3-Cl, 4-CF.sub.3                                        H         C.sub.2 H.sub.5                                                                           3-Cl, 5-CF.sub.3                                        H         C.sub.2 H.sub.5                                                                           3-CF.sub.3, 4-Cl                                        H         C.sub.2 H.sub.5                                                                           3-Cl, 5-OCF.sub.3                                       H         C.sub.2 H.sub.5                                                                           3-F, 5-CF.sub.3                                         H         C.sub.2 H.sub.5                                                                           2-CH.sub.3, 4-CN                                        H         C.sub.2 H.sub.5                                                                           3-NO.sub.2, 4-CH.sub.3                                  H         C.sub.2 H.sub.5                                                                           2-CH.sub.3, 4-OCH.sub.3                                 H         C.sub.2 H.sub.5                                                                           3-CH.sub.3, 4-OCH.sub.3                                 H         C.sub.2 H.sub.5                                                                           3-CH.sub.3, 5-OCH.sub.3                                 H         C.sub.2 H.sub.5                                                                           3-OCH.sub.3, 4-CH.sub.3                                 H         C.sub.2 H.sub.5                                                                           2-CH.sub.3, 4-O-i-C.sub.3 H.sub.7                       H         C.sub.2 H.sub.5                                                                           3-CH.sub.3, 4-O-i-C.sub.3 H.sub.7                       H         C.sub.2 H.sub.5                                                                           3-O-i-C.sub.3 H.sub.7, 4-CH.sub.3                       H         C.sub.2 H.sub.5                                                                           2-CH.sub.3, 4-CF.sub.3                                  H         C.sub.2 H.sub.5                                                                           2-CH.sub.3, 5-CF.sub.3                                  H         C.sub.2 H.sub.5                                                                           3-CH.sub.3, 4-CF.sub.3                                  H         C.sub.2 H.sub.5                                                                           3-CH.sub.3, 5-CF.sub.3                                  H         C.sub.2 H.sub.5                                                                           3-CF.sub.3, 4-CH.sub.3                                  H         C.sub.2 H.sub.5                                                                           3-CF.sub.3, 4-OCH.sub.3                                 H         C.sub.2 H.sub.5                                                                           3-OCH.sub.3, 4-CF.sub.3                                 H         C.sub.2 H.sub.5                                                                           2-CH.sub.3, 4-C(CH.sub.3)═NOCH.sub.3                H         C.sub.2 H.sub.5                                                                           3-CH.sub.3, 4-C(CH.sub.3)═NOCH.sub.3                H         C.sub.2 H.sub.5                                                                           2-OH, 5-CH.sub.3                                        H         C.sub.2 H.sub.5                                                                           3-CH.sub.3, 4-OC.sub.2 H.sub.5                          H         C.sub.2 H.sub.5                                                                           3-CH.sub.3, 4-O-t-C.sub.4 H.sub.9                       H         C.sub.2 H.sub.5                                                                           3-OC.sub.2 H.sub.5, 4-CH.sub.3                          H         C.sub.2 H.sub.5                                                                           3-O-t-C.sub.4 H.sub.9, 4-CH.sub.3                       H         C.sub.2 H.sub.5                                                                           2-C(COOCH.sub.3)═NOCH.sub.3                         H         C.sub.2 H.sub.5                                                     H         C.sub.2 H.sub.5                                                     CH.sub.3  C.sub.2 H.sub.5                                                                           H                                                       CH.sub.3  C.sub.2 H.sub.5                                                                           2-F                                                     CH.sub.3  C.sub.2 H.sub.5                                                                           3-F                                                     CH.sub.3  C.sub.2 H.sub.5                                                                           4-F                                                     CH.sub.3  C.sub.2 H.sub.5                                                                           2,4-F.sub.2                                             CH.sub.3  C.sub.2 H.sub.5                                                                           3,4-F.sub.2                                             CH.sub.3  C.sub.2 H.sub.5                                                                           3,5-F.sub.2                                             CH.sub.3  C.sub.2 H.sub.5                                                                           2-Cl                                                    CH.sub.3  C.sub.2 H.sub.5                                                                           3-Cl                                                    CH.sub.3  C.sub.2 H.sub.5                                                                           4-Cl                                                    CH.sub.3  C.sub.2 H.sub.5                                                                           2,4-Cl.sub.2                                            CH.sub.3  C.sub.2 H.sub.5                                                                           3,4-Cl.sub.2                                            CH.sub.3  C.sub.2 H.sub.5                                                                           3,5-Cl.sub.2                                            CH.sub.3  C.sub.2 H.sub.5                                                                           2-Br                                                    CH.sub.3  C.sub.2 H.sub.5                                                                           3-Br                                                    CH.sub.3  C.sub.2 H.sub.5                                                                           4-Br                                                    CH.sub.3  C.sub.2 H.sub.5                                                                           3,5-Br.sub.2                                            CH.sub.3  C.sub.2 H.sub.5                                                                           3-I                                                     CH.sub.3  C.sub.2 H.sub.5                                                                           4-I                                                     CH.sub.3  C.sub.2 H.sub.5                                                                           3-F, 5-Cl                                               CH.sub.3  C.sub.2 H.sub.5                                                                           3-F, 5-Br                                               CH.sub.3  C.sub.2 H.sub.5                                                                           3-Cl, 5-Br                                              CH.sub.3  C.sub.2 H.sub.5                                                                           3-Br, 4-F                                               CH.sub.3  C.sub.2 H.sub.5                                                                           2-NO.sub.2                                              CH.sub.3  C.sub.2 H.sub.5                                                                           3-NO.sub.2                                              CH.sub.3  C.sub.2 H.sub.5                                                                           4-NO.sub.2                                              CH.sub.3  C.sub.2 H.sub.5                                                                           2-CN                                                    CH.sub.3  C.sub.2 H.sub.5                                                                           3-CN                                                    CH.sub.3  C.sub.2 H.sub.5                                                                           4-CN                                                    CH.sub.3  C.sub.2 H.sub.5                                                                           2-CH.sub.3                                              CH.sub.3  C.sub.2 H.sub.5                                                                           3-CH.sub.3                                              CH.sub.3  C.sub.2 H.sub.5                                                                           4-CH.sub.3                                              CH.sub.3  C.sub.2 H.sub.5                                                                           2,4-(CH.sub.3).sub.2                                    CH.sub.3  C.sub.2 H.sub.5                                                                           2,5-(CH.sub.3).sub.2                                    CH.sub.3  C.sub.2 H.sub.5                                                                           3,4-(CH.sub.3).sub.2                                    CH.sub.3  C.sub.2 H.sub.5                                                                           3,5-(CH.sub.3).sub.2                                    CH.sub.3  C.sub.2 H.sub.5                                                                           2,4,5-(CH.sub.3).sub.3                                  CH.sub.3  C.sub.2 H.sub.5                                                                           2,4,6-(CH.sub.3).sub.3                                  CH.sub.3  C.sub.2 H.sub.5                                                                           3-C.sub.2 H.sub.5                                       CH.sub.3  C.sub.2 H.sub.5                                                                           4-C.sub.2 H.sub.5                                       CH.sub.3  C.sub.2 H.sub.5                                                                           3,4-(C.sub.2 H.sub.5).sub.2                             CH.sub.3  C.sub.2 H.sub.5                                                                           3,5-(C.sub.2 H.sub.5).sub.2                             CH.sub.3  C.sub.2 H.sub.5                                                                           3-n-C.sub.3 H.sub.7                                     CH.sub.3  C.sub.2 H.sub.5                                                                           4-n-C.sub.3 H.sub.7                                     CH.sub.3  C.sub.2 H.sub.5                                                                           3-i-C.sub.3 H.sub.7                                     CH.sub.3  C.sub.2 H.sub.5                                                                           4-i-C.sub.3 H.sub.7                                     CH.sub.3  C.sub.2 H.sub.5                                                                           3-Cyclopropyl                                           CH.sub.3  C.sub.2 H.sub.5                                                                           4-Cyclopropyl                                           CH.sub.3  C.sub.2 H.sub.5                                                                           3-n-C.sub.4 H.sub.9                                     CH.sub.3  C.sub.2 H.sub.5                                                                           4-n-C.sub.4 H.sub.9                                     CH.sub.3  C.sub.2 H.sub.5                                                                           3-t-C.sub.4 H.sub.9                                     CH.sub.3  C.sub.2 H.sub.5                                                                           4-t-C.sub.4 H.sub.9                                     CH.sub.3  C.sub.2 H.sub.5                                                                           3-n-C.sub.6 H.sub.13                                    CH.sub.3  C.sub.2 H.sub.5                                                                           4-n-C.sub.6 H.sub.13                                    CH.sub.3  C.sub.2 H.sub.5                                                                           3-Cyclohexyl                                            CH.sub.3  C.sub.2 H.sub.5                                                                           4-Cyclohexyl                                            CH.sub.3  C.sub.2 H.sub.5                                                                           3-Phenyl                                                CH.sub.3  C.sub.2 H.sub.5                                                                           4-Phenyl                                                CH.sub.3  C.sub.2 H.sub.5                                                                           4-Allyl                                                 CH.sub.3  C.sub.2 H.sub.5                                                                           4-Propargyl                                             CH.sub.3  C.sub.2 H.sub.5                                                                           2-CH.sub.3, 4-C.sub.2 H.sub.5                           CH.sub.3  C.sub.2 H.sub.5                                                                           2-CH.sub.3, 4-i-C.sub.3 H.sub.7                         CH.sub.3  C.sub.2 H.sub.5                                                                           2-CH.sub.3, 4-t-C.sub.4 H.sub.9                         CH.sub.3  C.sub.2 H.sub.5                                                                           2-CH.sub.3, 4-phenyl                                    CH.sub.3  C.sub.2 H.sub.5                                                                           3-CH.sub.3, 4-phenyl                                    CH.sub.3  C.sub.2 H.sub.5                                                                           3-OH                                                    CH.sub.3  C.sub.2 H.sub.5                                                                           4-OH                                                    CH.sub.3  C.sub.2 H.sub.5                                                                           3-OCH.sub.3                                             CH.sub.3  C.sub.2 H.sub.5                                                                           4-OCH.sub.3                                             CH.sub.3  C.sub.2 H.sub.5                                                                           3,4-(OCH.sub.3).sub.2                                   CH.sub.3  C.sub.2 H.sub.5                                                                           3,5-(OCH.sub.3).sub.2                                   CH.sub.3  C.sub.2 H.sub.5                                                                           3,4,5-(OCH.sub.3).sub.3                                 CH.sub.3  C.sub.2 H.sub.5                                                                           4-OC.sub.2 H.sub.5                                      CH.sub.3  C.sub.2 H.sub.5                                                                           4-O-i-C.sub.3 H.sub.7                                   CH.sub.3  C.sub.2 H.sub.5                                                                           3-O-t-C.sub.4 H.sub.9                                   CH.sub.3  C.sub.2 H.sub.5                                                                           4-O-t-C.sub.4 H.sub.9                                   CH.sub.3  C.sub.2 H.sub.5                                                                           4-O-n-C.sub.6 H.sub.13                                  CH.sub.3  C.sub.2 H.sub.5                                                                           3-O-Phenyl                                              CH.sub.3  C.sub.2 H.sub.5                                                                           4-O-Phenyl                                              CH.sub.3  C.sub.2 H.sub.5                                                                           4-O-Allyl                                               CH.sub.3  C.sub.2 H.sub.5                                                                           2-CF.sub.3                                              CH.sub.3  C.sub.2 H.sub.5                                                                           3-CF.sub.3                                              CH.sub.3  C.sub.2 H.sub.5                                                                           4-CF.sub.3                                              CH.sub.3  C.sub.2 H.sub.5                                                                           3,5-(CF.sub.3).sub.2                                    CH.sub.3  C.sub.2 H.sub.5                                                                           4-CH.sub.2 CF.sub.3                                     CH.sub.3  C.sub.2 H.sub.5                                                                           4-C.sub.2 F.sub.5                                       CH.sub.3  C.sub.2 H.sub.5                                                                           4-CF.sub.2 CHF.sub.2                                    CH.sub.3  C.sub.2 H.sub.5                                                                           3-OCF.sub.3                                             CH.sub.3  C.sub.2 H.sub.5                                                                           4-OCF.sub.3                                             CH.sub.3  C.sub.2 H.sub.5                                                                           4-OCH.sub.2 CF.sub.3                                    CH.sub.3  C.sub.2 H.sub.5                                                                           4-OC.sub.2 F.sub.5                                      CH.sub.3  C.sub.2 H.sub.5                                                                           4-OCF.sub.2 CHF.sub.2                                   CH.sub.3  C.sub.2 H.sub.5                                                                           3-CH.sub.2 OCH.sub.3                                    CH.sub.3  C.sub.2 H.sub.5                                                                           4-CH.sub.2 OCH.sub.3                                    CH.sub.3  C.sub.2 H.sub.5                                                                           4-CH.sub.2 --O-t-C.sub.4 H.sub.9                        CH.sub.3  C.sub.2 H.sub.5                                                                           4-CH(OCH.sub.3).sub.2                                   CH.sub.3  C.sub.2 H.sub.5                                                                           4-CH.sub.2 CN                                           CH.sub.3  C.sub.2 H.sub.5                                                                           3-CHO                                                   CH.sub.3  C.sub.2 H.sub.5                                                                           4-CHO                                                   CH.sub.3  C.sub.2 H.sub.5                                                                           3-CO--CH.sub.3                                          CH.sub.3  C.sub.2 H.sub.5                                                                           4-CO--CH.sub.3                                          CH.sub.3  C.sub.2 H.sub.5                                                                           3-COOH                                                  CH.sub.3  C.sub.2 H.sub.5                                                                           4-COOH                                                  CH.sub.3  C.sub.2 H.sub.5                                                                           3-COOCH.sub.3                                           CH.sub.3  C.sub.2 H.sub.5                                                                           4-COOCH.sub.3                                           CH.sub.3  C.sub.2 H.sub.5                                                                           3-COOC.sub.2 H.sub.5                                    CH.sub.3  C.sub.2 H.sub.5                                                                           4-COOC.sub.2 H.sub.5                                    CH.sub.3  C.sub.2 H.sub.5                                                                           3-COO-i-C.sub.3 H.sub.7                                 CH.sub.3  C.sub.2 H.sub.5                                                                           4-COO-i-C.sub.3 H.sub.7                                 CH.sub.3  C.sub.2 H.sub.5                                                                           3-COO-t-C.sub.4 H.sub.9                                 CH.sub.3  C.sub.2 H.sub.5                                                                           4-COO-t-C.sub.4 H.sub.9                                 CH.sub.3  C.sub.2 H.sub.5                                                                           3-COO-n-C.sub.6 H.sub.13                                CH.sub.3  C.sub.2 H.sub.5                                                                           4-COO-n-C.sub.6 H.sub.13                                CH.sub.3  C.sub.2 H.sub.5                                                                           3-CONH.sub.2                                            CH.sub.3  C.sub.2 H.sub.5                                                                           4-CONH.sub.2                                            CH.sub.3  C.sub.2 H.sub.5                                                                           3-CONHCH.sub.3                                          CH.sub.3  C.sub.2 H.sub.5                                                                           4-CONHCH.sub.3                                          CH.sub.3  C.sub.2 H.sub.5                                                                           3-CON(CH.sub.3).sub.2                                   CH.sub.3  C.sub.2 H.sub.5                                                                           4-CON(CH.sub.3).sub.2                                   CH.sub.3  C.sub.2 H.sub.5                                                                           3-CSNH.sub.2                                            CH.sub.3  C.sub.2 H.sub.5                                                                           4-CSNH.sub.2                                            CH.sub.3  C.sub.2 H.sub.5                                                                           3-NH.sub.2                                              CH.sub.3  C.sub.2 H.sub.5                                                                           4-NH.sub.2                                              CH.sub.3  C.sub.2 H.sub.5                                                                           4-NHCH.sub.3                                            CH.sub.3  C.sub.2 H.sub.5                                                                           4-N(CH.sub.3).sub.2                                     CH.sub.3  C.sub.2 H.sub.5                                                                           3-NHCO--CH.sub.3                                        CH.sub.3  C.sub.2 H.sub.5                                                                           4-NHCO--CH.sub.3                                        CH.sub.3  C.sub.2 H.sub.5                                                                           4-NCH.sub.3 --CO--CH.sub.3                              CH.sub.3  C.sub.2 H.sub.5                                                                           4-NHCOOCH.sub.3                                         CH.sub.3  C.sub.2 H.sub.5                                                                           4-NCH.sub.3 --COOCH.sub.3                               CH.sub.3  C.sub.2 H.sub.5                                                                           3-OCO--CH.sub.3                                         CH.sub.3  C.sub.2 H.sub.5                                                                           4-OCO--CH.sub.3                                         CH.sub.3  C.sub.2 H.sub.5                                                                           4-OCO-t-C.sub.4 H.sub.9                                 CH.sub.3  C.sub.2 H.sub.5                                                                           4-SH                                                    CH.sub.3  C.sub.2 H.sub.5                                                                           4-SCH.sub.3                                             CH.sub.3  C.sub.2 H.sub.5                                                                           4-S-t-C.sub.4 H.sub.9                                   CH.sub.3  C.sub.2 H.sub.5                                                                           4-SO--CH.sub.3                                          CH.sub.3  C.sub.2 H.sub.5                                                                           4-SO.sub.2 --CH.sub.3                                   CH.sub.3  C.sub.2 H.sub.5                                                                           4-C(CH.sub.3)═NCH.sub.3                             CH.sub.3  C.sub.2 H.sub.5                                                                           4-C(SCH.sub.3)═NOCH.sub.3                           CH.sub.3  C.sub.2 H.sub.5                                                                           4-C(OCH.sub.3)═NOCH.sub.3                           CH.sub.3  C.sub.2 H.sub.5                                                                           3-CH═NOCH.sub.3                                     CH.sub.3  C.sub.2 H.sub.5                                                                           4-CH═NOCH.sub.3                                     CH.sub.3  C.sub.2 H.sub.5                                                                           3-C(CH.sub.3)═NOCH.sub.3                            CH.sub.3  C.sub.2 H.sub.5                                                                           4-C(CH.sub.3)═NOCH.sub.3                            CH.sub.3  C.sub.2 H.sub.5                                                                           4-C(CH.sub.3)═NOC.sub.2 H.sub.5                     CH.sub.3  C.sub.2 H.sub.5                                                                           4-C(CH.sub.3)═NO-n-C.sub.3 H.sub.7                  CH.sub.3  C.sub.2 H.sub.5                                                                           4-C(CH.sub.3)═NO-i-C.sub.3 H.sub.7                  CH.sub.3  C.sub.2 H.sub.5                                                                           4-C(CH.sub.3)═NO-n-C.sub.4 H.sub.9                  CH.sub.3  C.sub.2 H.sub.5                                                                           4-C(CH.sub.3)═NO-t-C.sub.4 H.sub.9                  CH.sub.3  C.sub.2 H.sub.5                                                                           4-C(CH.sub.3)═NO-n-C.sub.5 H.sub.11                 CH.sub.3  C.sub.2 H.sub.5                                                                           4-C(CH.sub.3)═NO-n-C.sub.6 H.sub.13                 CH.sub.3  C.sub.2 H.sub.5                                                                           2-Cl, 4-CH.sub.3                                        CH.sub.3  C.sub.2 H.sub.5                                                                           3-Cl, 5-CH.sub.3                                        CH.sub.3  C.sub.2 H.sub.5                                                                           2-CH.sub.3, 4-Cl                                        CH.sub.3  C.sub.2 H.sub.5                                                                           3-CH.sub.3, 4-Cl                                        CH.sub.3  C.sub.2 H.sub.5                                                                           3-F, 5-CH.sub.3                                         CH.sub.3  C.sub.2 H.sub.5                                                                           3-Br, 5-CH.sub.3                                        CH.sub.3  C.sub.2 H.sub.5                                                                           3-Cl, 5-NO.sub.2                                        CH.sub.3  C.sub.2 H.sub.5                                                                           3-NO.sub.2, 4-Cl                                        CH.sub.3  C.sub.2 H.sub.5                                                                           3-Cl, 4-OCH.sub.3                                       CH.sub.3  C.sub.2 H.sub.5                                                                           3-OCH.sub.3, 4-Cl                                       CH.sub.3  C.sub.2 H.sub.5                                                                           3-Cl, 5-CF.sub.3                                        CH.sub.3  C.sub.2 H.sub.5                                                                           3-Cl, 5-OCF.sub.3                                       CH.sub.3  C.sub.2 H.sub.5                                                                           3-F, 5-CF.sub.3                                         CH.sub.3  C.sub.2 H.sub.5                                                                           2-CH.sub.3, 4-CN                                        CH.sub.3  C.sub.2 H.sub.5                                                                           2-CH.sub.3, 4-OCH.sub.3                                 CH.sub.3  C.sub.2 H.sub.5                                                                           2-CH.sub.3, 4-CF.sub.3                                  CH.sub.3  C.sub.2 H.sub.5                                                                           2-CH.sub.3, 4-C(CH.sub.3)═NOCH.sub.3                CH.sub.3  C.sub.2 H.sub.5                                                                           3-CH.sub.3, 4-C(CH.sub.3)═NOCH.sub.3                CH.sub.3  C.sub.2 H.sub.5                                                                           2-OH, 5-CH.sub.3                                        CH.sub.3  C.sub.2 H.sub.5                                                                           3-CH.sub.3, 4-O-t-C.sub.4 H.sub.9                       CH.sub.3  C.sub.2 H.sub.5                                                                           2-C(COOCH.sub.3)═NOCH.sub.3                         CH.sub.3  C.sub.2 H.sub.5                                                                           2,3-Butadienyl                                          CH.sub.3  C.sub.2 H.sub.5                                                                           3,4-Butadienyl                                          H         CH(CH.sub.3).sub.2                                                                        H                                                       H         CH(CH.sub.3).sub.2                                                                        2-F                                                     H         CH(CH.sub.3).sub.2                                                                        3-F                                                     H         CH(CH.sub.3).sub.2                                                                        4-F                                                     H         CH(CH.sub.3).sub.2                                                                        2,3-F.sub.2                                             H         CH(CH.sub.3).sub.2                                                                        2,4-F.sub.2                                             H         CH(CH.sub.3).sub.2                                                                        2,5-F.sub.2                                             H         CH(CH.sub.3).sub.2                                                                        2,6-F.sub.2                                             H         CH(CH.sub.3).sub.2                                                                        3,4-F.sub.2                                             H         CH(CH.sub.3).sub.2                                                                        3,5-F.sub.2                                             H         CH(CH.sub.3).sub.2                                                                        2-Cl                                                    H         CH(CH.sub.3).sub.2                                                                        3-Cl                                                    H         CH(CH.sub.3).sub.2                                                                        4-Cl                                                    H         CH(CH.sub.3).sub.2                                                                        2,4-Cl.sub.2                                            H         CH(CH.sub.3).sub.2                                                                        2,5-Cl.sub.2                                            H         CH(CH.sub.3).sub.2                                                                        3,4-Cl.sub.2                                            H         CH(CH.sub.3).sub.2                                                                        3,5-Cl.sub.2                                            H         CH(CH.sub.3).sub.2                                                                        2-Br                                                    H         CH(CH.sub.3).sub.2                                                                        3-Br                                                    H         CH(CH.sub.3).sub.2                                                                        4-Br                                                    H         CH(CH.sub.3).sub.2                                                                        2,4-Br.sub.2                                            H         CH(CH.sub.3).sub.2                                                                        3,4-Br.sub.2                                            H         CH(CH.sub.3).sub.2                                                                        3,5-Br.sub.2                                            H         CH(CH.sub.3).sub.2                                                                        2-I                                                     H         CH(CH.sub.3).sub.2                                                                        3-I                                                     H         CH(CH.sub.3).sub.2                                                                        4-I                                                     H         CH(CH.sub.3).sub.2                                                                        2-F, 4-Cl                                               H         CH(CH.sub.3).sub.2                                                                        2-F, 5-Cl                                               H         CH(CH.sub.3).sub.2                                                                        2-F, 4-Br                                               H         CH(CH.sub.3).sub.2                                                                        2-F, 5-Br                                               H         CH(CH.sub.3).sub.2                                                                        2-Cl, 4-Br                                              H         CH(CH.sub.3).sub.2                                                                        2-Cl, 5-Br                                              H         CH(CH.sub.3).sub.2                                                                        3-F, 4-Cl                                               H         CH(CH.sub.3).sub.2                                                                        3-F, 5-Cl                                               H         CH(CH.sub.3).sub.2                                                                        3-F, 4-Br                                               H         CH(CH.sub.3).sub.2                                                                        3-F, 5-Br                                               H         CH(CH.sub.3).sub.2                                                                        3-Cl, 4-Br                                              H         CH(CH.sub.3).sub.2                                                                        3-Cl, 5-Br                                              H         CH(CH.sub.3).sub.2                                                                        3-Cl, 4-F                                               H         CH(CH.sub.3).sub.2                                                                        3-Br, 4-F                                               H         CH(CH.sub.3).sub.2                                                                        3-Br, 4-Cl                                              H         CH(CH.sub.3).sub.2                                                                        2-NO.sub.2                                              H         CH(CH.sub.3).sub.2                                                                        3-NO.sub.2                                              H         CH(CH.sub.3).sub.2                                                                        4-NO.sub.2                                              H         CH(CH.sub.3).sub.2                                                                        2-CN                                                    H         CH(CH.sub.3).sub.2                                                                        3-CN                                                    H         CH(CH.sub.3).sub.2                                                                        4-CN                                                    H         CH(CH.sub.3).sub.2                                                                        2-CH.sub.3                                              H         CH(CH.sub.3).sub.2                                                                        3-CH.sub.3                                              H         CH(CH.sub.3).sub.2                                                                        4-CH.sub.3                                              H         CH(CH.sub.3).sub.2                                                                        2,3-(CH.sub.3).sub.2                                    H         CH(CH.sub.3).sub.2                                                                        2,4-(CH.sub.3).sub.2                                    H         CH(CH.sub.3).sub.2                                                                        2,5-(CH.sub.3).sub.2                                    H         CH(CH.sub.3).sub.2                                                                        2,6-(CH.sub.3).sub.2                                    H         CH(CH.sub.3).sub.2                                                                        3,4-(CH.sub.3).sub.2                                    H         CH(CH.sub.3).sub.2                                                                        3,5-(CH.sub.3).sub.2                                    H         CH(CH.sub.3).sub.2                                                                        2,4,5-(CH.sub.3).sub.3                                  H         CH(CH.sub.3).sub.2                                                                        2,4,6-(CH.sub.3).sub.3                                  H         CH(CH.sub.3).sub.2                                                                        3,4,5-(CH.sub.3).sub.3                                  H         CH(CH.sub.3).sub.2                                                                        2-C.sub.2 H.sub.5                                       H         CH(CH.sub.3).sub.2                                                                        3-C.sub.2 H.sub.5                                       H         CH(CH.sub.3).sub.2                                                                        4-C.sub.2 H.sub.5                                       H         CH(CH.sub.3).sub.2                                                                        3,4-(C.sub.2 H.sub.5).sub.2                             H         CH(CH.sub.3).sub.2                                                                        3,5-(C.sub.2 H.sub.5).sub.2                             H         CH(CH.sub.3).sub.2                                                                        3-n-C.sub.3 H.sub.7                                     H         CH(CH.sub.3).sub.2                                                                        4-n-C.sub.3 H.sub.7                                     H         CH(CH.sub.3).sub.2                                                                        3,4-(n-C.sub.3 H.sub.7).sub.2                           H         CH(CH.sub.3).sub.2                                                                        3,5-(n-C.sub.3 H.sub.7).sub.2                           H         CH(CH.sub.3).sub.2                                                                        3-i-C.sub.3 H.sub.7                                     H         CH(CH.sub.3).sub.2                                                                        4-i-C.sub.3 H.sub.7                                     H         CH(CH.sub.3).sub.2                                                                        3,4-(i-C.sub.3 H.sub.7).sub.2                           H         CH(CH.sub.3).sub.2                                                                        3,5-(i-C.sub.3 H.sub.7).sub.2                           H         CH(CH.sub.3).sub.2                                                                        3-Cyclopropyl                                           H         CH(CH.sub.3).sub.2                                                                        4-Cyclopropyl                                           H         CH(CH.sub.3).sub.2                                                                        3-n-C.sub.4 H.sub.9                                     H         CH(CH.sub.3).sub.2                                                                        4-n-C.sub.4 H.sub.9                                     H         CH(CH.sub.3).sub.2                                                                        3,4-(n-C.sub.4 H.sub.9).sub.2                           H         CH(CH.sub.3).sub.2                                                                        3,5-(n-C.sub.4 H.sub.9).sub.2                           H         CH(CH.sub.3).sub.2                                                                        3-s-C.sub.4 H.sub.9                                     H         CH(CH.sub.3).sub.2                                                                        4-s-C.sub.4 H.sub.9                                     H         CH(CH.sub.3).sub.2                                                                        3-i-C.sub.4 H.sub.9                                     H         CH(CH.sub.3).sub.2                                                                        4-i-C.sub.4 H.sub.9                                     H         CH(CH.sub.3).sub.2                                                                        3-t-C.sub.4 H.sub.9                                     H         CH(CH.sub.3).sub.2                                                                        4-t-C.sub.4 H.sub.9                                     H         CH(CH.sub.3).sub.2                                                                        3,4-(t-C.sub.4 H.sub.9).sub.2                           H         CH(CH.sub.3).sub.2                                                                        3,5-(t-C.sub.4 H.sub.9).sub.2                           H         CH(CH.sub.3).sub.2                                                                        3-n-C.sub.5 H.sub.11                                    H         CH(CH.sub.3).sub.2                                                                        4-n-C.sub.5 H.sub.11                                    H         CH(CH.sub.3).sub.2                                                                        3-n-C.sub.6 H.sub.13                                    H         CH(CH.sub.3).sub.2                                                                        4-n-C.sub.6 H.sub.13                                    H         CH(CH.sub.3).sub.2                                                                        3-Cyclohexyl                                            H         CH(CH.sub.3).sub.2                                                                        4-Cyclohexyl                                            H         CH(CH.sub.3).sub.2                                                                        3-Phenyl                                                H         CH(CH.sub.3).sub.2                                                                        4-Phenyl                                                H         CH(CH.sub.3).sub.2                                                                        3-Vinyl                                                 H         CH(CH.sub.3).sub.2                                                                        4-Vinyl                                                 H         CH(CH.sub.3).sub.2                                                                        3-Allyl                                                 H         CH(CH.sub.3).sub.2                                                                        4-Allyl                                                 H         CH(CH.sub.3).sub.2                                                                        3-Propargyl                                             H         CH(CH.sub.3).sub.2                                                                        4-Propargyl                                             H         CH(CH.sub.3).sub.2                                                                        3-(Propen-2-yl)                                         H         CH(CH.sub.3).sub.2                                                                        4-(Propen-2-yl)                                         H         CH(CH.sub.3).sub.2                                                                        2-CH.sub.3, 4-C.sub.2 H.sub.5                           H         CH(CH.sub.3).sub.2                                                                        2-CH.sub.3, 5-C.sub.2 H.sub.5                           H         CH(CH.sub.3).sub.2                                                                        2-CH.sub.3 --, 4-n-C.sub.3 H.sub.7                      H         CH(CH.sub.3).sub.2                                                                        2-CH.sub.3, 5-n-C.sub.3 H.sub.7                         H         CH(CH.sub.3).sub.2                                                                        2-CH.sub.3, 4-i-C.sub.3 H.sub.7                         H         CH(CH.sub.3).sub.2                                                                        2-CH.sub.3, 5-i-C.sub.3 H.sub.7                         H         CH(CH.sub.3).sub.2                                                                        2-CH.sub.3, 4-n-C.sub.4 H.sub.9                         H         CH(CH.sub.3).sub.2                                                                        2-CH.sub.3, 4-s-C.sub.4 H.sub.9                         H         CH(CH.sub.3).sub.2                                                                        2-CH.sub.3, 4-i-C.sub.4 H.sub.9                         H         CH(CH.sub.3).sub.2                                                                        2-CH.sub.3, 4-t-C.sub.4 H.sub.9                         H         CH(CH.sub.3).sub.2                                                                        2-CH.sub.3, 4-phenyl                                    H         CH(CH.sub.3).sub.2                                                                        2-CH.sub.3, 5-phenyl                                    H         CH(CH.sub.3).sub.2                                                                        2-CH.sub.3, 4-vinyl                                     H         CH(CH.sub.3).sub.2                                                                        2-CH.sub.3, 4-allyl                                     H         CH(CH.sub.3).sub.2                                                                        2-CH.sub.3, 4-propargyl                                 H         CH(CH.sub.3).sub.2                                                                        2-CH.sub.3, 4-(propen-2-yl)                             H         CH(CH.sub.3).sub.2                                                                        3-CH.sub.3, 4-C.sub.2 H.sub.5                           H         CH(CH.sub.3).sub.2                                                                        3-CH.sub.3, 5-C.sub.2 H.sub.5                           H         CH(CH.sub.3).sub.2                                                                        3-CH.sub.3, 4-n-C.sub.3 H.sub.7                         H         CH(CH.sub.3).sub.2                                                                        3-CH.sub.3, 5-n-C.sub.3 H.sub.7                         H         CH(CH.sub.3).sub.2                                                                        3-CH.sub.3, 4-i-C.sub.3 H.sub.7                         H         CH(CH.sub.3).sub.2                                                                        3-CH.sub.3, 5-i-C.sub.3 H.sub.7                         H         CH(CH.sub.3).sub.2                                                                        3-CH.sub.3, 4-cyclopropyl                               H         CH(CH.sub.3).sub.2                                                                        3-CH.sub.3, 4-t-C.sub.4 H.sub.9                         H         CH(CH.sub.3).sub.2                                                                        3-CH.sub.3, 5-t-C.sub.4 H.sub.9                         H         CH(CH.sub.3).sub.2                                                                        3-CH.sub.3, 4-phenyl                                    H         CH(CH.sub.3).sub.2                                                                        3-CH.sub.3, 5-phenyl                                    H         CH(CH.sub.3).sub.2                                                                        3-CH.sub.3, 4-vinyl                                     H         CH(CH.sub.3).sub.2                                                                        3-CH.sub.3, 4-allyl                                     H         CH(CH.sub.3).sub.2                                                                        3-CH.sub.3, 4-propargyl                                 H         CH(CH.sub.3).sub.2                                                                        3-CH.sub.3, 4-propen-2-yl                               H         CH(CH.sub.3).sub.2                                                                        3-C.sub.2 H.sub.5, 4-CH.sub.3                           H         CH(CH.sub.3).sub.2                                                                        3-i-C.sub.3 H.sub.7, 4-CH.sub.3                         H         CH(CH.sub.3).sub.2                                                                        3-t-C.sub.4 H.sub.9, 4-CH.sub.3                         H         CH(CH.sub.3).sub.2                                                                        3-Phenyl, 4-CH.sub.3                                    H         CH(CH.sub.3).sub.2                                                                        2-OH                                                    H         CH(CH.sub.3).sub.2                                                                        3-OH                                                    H         CH(CH.sub.3).sub.2                                                                        4-OH                                                    H         CH(CH.sub.3).sub.2                                                                        2-OCH.sub.3                                             H         CH(CH.sub.3).sub.2                                                                        3-OCH.sub.3                                             H         CH(CH.sub.3).sub.2                                                                        4-OCH.sub.3                                             H         CH(CH.sub.3).sub.2                                                                        2,3-(OCH.sub.3).sub.2                                   H         CH(CH.sub.3).sub.2                                                                        2,4-(OCH.sub.3).sub.2                                   H         CH(CH.sub.3).sub.2                                                                        2,5-(OCH.sub.3).sub.2                                   H         CH(CH.sub.3).sub.2                                                                        3,4-(OCH.sub.3).sub.2                                   H         CH(CH.sub.3).sub.2                                                                        3,5-(OCH.sub.3).sub.2                                   H         CH(CH.sub.3).sub.2                                                                        3,4,5-(OCH.sub.3).sub.3                                 H         CH(CH.sub.3).sub.2                                                                        3-OC.sub.2 H.sub.5                                      H         CH(CH.sub.3).sub.2                                                                        4-OC.sub.2 H.sub.5                                      H         CH(CH.sub.3).sub.2                                                                        3,4-(OC.sub.2 H.sub.5).sub.2                            H         CH(CH.sub.3).sub.2                                                                        3,5-(OC.sub.2 H.sub.5).sub.2                            H         CH(CH.sub.3).sub.2                                                                        3-O-n-C.sub.3 H.sub.7                                   H         CH(CH.sub.3).sub.2                                                                        4-O-n-C.sub.3 H.sub.7                                   H         CH(CH.sub.3).sub.2                                                                        3-O-i-C.sub.3 H.sub.7                                   H         CH(CH.sub.3).sub.2                                                                        4-O-i-C.sub.3 H.sub.7                                   H         CH(CH.sub.3).sub.2                                                                        3-O-Cyclopropyl                                         H         CH(CH.sub.3).sub.2                                                                        4-O-Cyclopropyl                                         H         CH(CH.sub.3).sub.2                                                                        3-O-n-C.sub.4 H.sub.9                                   H         CH(CH.sub.3).sub.2                                                                        4-O-n-C.sub.4 H.sub.9                                   H         CH(CH.sub.3).sub.2                                                                        3-O-s-C.sub.4 H.sub.9                                   H         CH(CH.sub.3).sub.2                                                                        4-O-s-C.sub.4 H.sub.9                                   H         CH(CH.sub.3).sub.2                                                                        3-O-i-C.sub.4 H.sub.9                                   H         CH(CH.sub.3).sub.2                                                                        4-O-i-C.sub.4 H.sub.9                                   H         CH(CH.sub.3).sub.2                                                                        3-O-t-C.sub.4 H.sub.9                                   H         CH(CH.sub.3).sub.2                                                                        4-O-t-C.sub.4 H.sub.9                                   H         CH(CH.sub.3).sub.2                                                                        3-O-n-C.sub.5 H.sub.11                                  H         CH(CH.sub.3).sub.2                                                                        4-O-n-C.sub.5 H.sub.11                                  H         CH(CH.sub.3).sub.2                                                                        3-O-n-C.sub.6 H.sub.13                                  H         CH(CH.sub.3).sub.2                                                                        4-O-n-C.sub.6 H.sub.13                                  H         CH(CH.sub.3).sub.2                                                                        3-O-Cyclohexyl                                          H         CH(CH.sub.3).sub.2                                                                        4-O-Cyclohexyl                                          H         CH(CH.sub.3).sub.2                                                                        3-O-Phenyl                                              H         CH(CH.sub.3).sub.2                                                                        4-O-Phenyl                                              H         CH(CH.sub.3).sub.2                                                                        3-O-Allyl                                               H         CH(CH.sub.3).sub.2                                                                        4-O-Allyl                                               H         CH(CH.sub.3).sub.2                                                                        2-CF.sub.3                                              H         CH(CH.sub.3).sub.2                                                                        3-CF.sub.3                                              H         CH(CH.sub.3).sub.2                                                                        4-CF.sub.3                                              H         CH(CH.sub.3).sub.2                                                                        2,4-(CF.sub.3).sub.2                                    H         CH(CH.sub.3).sub.2                                                                        3,5-(CF.sub.3).sub.2                                    H         CH(CH.sub.3).sub.2                                                                        3-CF.sub.2 Cl                                           H         CH(CH.sub.3).sub.2                                                                        4-CF.sub.2 Cl                                           H         CH(CH.sub.3).sub.2                                                                        3-CFCl.sub.2                                            H         CH(CH.sub.3).sub.2                                                                        4-CFCl.sub.2                                            H         CH(CH.sub.3).sub.2                                                                        3-CCl.sub.3                                             H         CH(CH.sub.3).sub.2                                                                        4-CCl.sub.3                                             H         CH(CH.sub.3).sub.2                                                                        3-CH.sub.2 CH.sub.2 F                                   H         CH(CH.sub.3).sub.2                                                                        4-CH.sub.2 CH.sub.2 F                                   H         CH(CH.sub.3).sub.2                                                                        3-CH.sub.2 CF.sub.3                                     H         CH(CH.sub.3).sub.2                                                                        4-CH.sub.2 CF.sub.3                                     H         CH(CH.sub.3).sub.2                                                                        3-C.sub.2 F.sub.5                                       H         CH(CH.sub.3).sub.2                                                                        4-C.sub.2 F.sub.5                                       H         CH(CH.sub.3).sub.2                                                                        3-CHCl.sub.2                                            H         CH(CH.sub.3).sub.2                                                                        4-CHCl.sub.2                                            H         CH(CH.sub.3).sub.2                                                                        3-CH.sub.2 Cl                                           H         CH(CH.sub.3).sub.2                                                                        4-CH.sub.2 Cl                                           H         CH(CH.sub.3).sub.2                                                                        3-CF.sub.2 CHF.sub.2                                    H         CH(CH.sub.3).sub.2                                                                        4-CF.sub.2 CHF.sub.2                                    H         CH(CH.sub.3).sub.2                                                                        3-CH.sub.2 CH.sub.2 Cl                                  H         CH(CH.sub.3).sub.2                                                                        4-CH.sub.2 CH.sub.2 Cl                                  H         CH(CH.sub.3).sub.2                                                                        2-OCF.sub.3                                             H         CH(CH.sub.3).sub.2                                                                        3-OCF.sub.3                                             H         CH(CH.sub.3).sub.2                                                                        4-OCF.sub.3                                             H         CH(CH.sub.3).sub.2                                                                        3-OCHF.sub.2                                            H         CH(CH.sub.3).sub.2                                                                        4-OCHF.sub.2                                            H         CH(CH.sub.3).sub.2                                                                        3-OC.sub.2 F.sub.5                                      H         CH(CH.sub.3).sub.2                                                                        4-OC.sub.2 F.sub.5                                      H         CH(CH.sub.3).sub.2                                                                        3-OCF.sub.2 CHF.sub.2                                   H         CH(CH.sub.3).sub.2                                                                        4-OCF.sub.2 CHF.sub.2                                   H         CH(CH.sub.3).sub.2                                                                        3-CH.sub.2 OCH.sub.3                                    H         CH(CH.sub.3).sub.2                                                                        4-CH.sub.2 OCH.sub.3                                    H         CH(CH.sub.3).sub.2                                                                        3-CH.sub.2 O-t-C.sub.4 H.sub.9                          H         CH(CH.sub.3).sub.2                                                                        4-CH.sub.2 O-t-C.sub.4 H.sub.9                          H         CH(CH.sub.3).sub.2                                                                        3-C(CH.sub.3)(OCH.sub.3).sub.2                          H         CH(CH.sub.3).sub.2                                                                        4-C(CH.sub.3)(OCH.sub.3).sub.2                          H         CH(CH.sub.3).sub.2                                                                        3-CH(OCH.sub.3).sub.2                                   H         CH(CH.sub.3).sub.2                                                                        4-CH(OCH.sub.3).sub.2                                   H         CH(CH.sub.3).sub.2                                                                        3-CH.sub.2 CN                                           H         CH(CH.sub.3).sub.2                                                                        4-CH.sub.2 CN                                           H         CH(CH.sub.3).sub.2                                                                        3-CHO                                                   H         CH(CH.sub.3).sub.2                                                                        4-CHO                                                   H         CH(CH.sub.3).sub.2                                                                        3-CO--CH.sub.3                                          H         CH(CH.sub.3).sub.2                                                                        4-CO--CH.sub.3                                          H         CH(CH.sub.3).sub.2                                                                        3-CO--C.sub.2 H.sub.5                                   H         CH(CH.sub.3).sub.2                                                                        4-CO--C.sub.2 H.sub.5                                   H         CH(CH.sub.3).sub.2                                                                        2-COOH                                                  H         CH(CH.sub.3).sub.2                                                                        3-COOH                                                  H         CH(CH.sub.3).sub.2                                                                        4-COOH                                                  H         CH(CH.sub.3).sub.2                                                                        3-COOCH.sub.3                                           H         CH(CH.sub.3).sub.2                                                                        4-COOCH.sub.3                                           H         CH(CH.sub.3).sub.2                                                                        3-COOC.sub.2 H.sub.5                                    H         CH(CH.sub.3).sub.2                                                                        4-COOC.sub.2 H.sub.5                                    H         CH(CH.sub.3).sub.2                                                                        3-COO-n-C.sub.3 H.sub.7                                 H         CH(CH.sub.3).sub.2                                                                        4-COO-n-C.sub.3 H.sub.7                                 H         CH(CH.sub.3).sub.2                                                                        3-COO-i-C.sub.3 H.sub.7                                 H         CH(CH.sub.3).sub.2                                                                        4-COO-i-C.sub.3 H.sub.7                                 H         CH(CH.sub.3).sub.2                                                                        3-COO-n-C.sub.4 H.sub.9                                 H         CH(CH.sub.3).sub.2                                                                        4-COO-n-C.sub.4 H.sub.9                                 H         CH(CH.sub.3).sub.2                                                                        3-COO-s-C.sub.4 H.sub.9                                 H         CH(CH.sub.3).sub.2                                                                        4-COO-s-C.sub.4 H.sub.9                                 H         CH(CH.sub.3).sub.2                                                                        3-COO-i-C.sub.4 H.sub.9                                 H         CH(CH.sub.3).sub.2                                                                        4-COO-i-C.sub.4 H.sub.9                                 H         CH(CH.sub.3).sub.2                                                                        3-COO-t-C.sub.4 H.sub.9                                 H         CH(CH.sub.3).sub.2                                                                        4-COO-t-C.sub.4 H.sub.9                                 H         CH(CH.sub.3).sub.2                                                                        3-COO-n-C.sub.5 H.sub.11                                H         CH(CH.sub.3).sub.2                                                                        4-COO-n-C.sub.5 H.sub.11                                H         CH(CH.sub.3).sub.2                                                                        3-COO-n-C.sub.6 H.sub.13                                H         CH(CH.sub.3).sub.2                                                                        4-COO-n-C.sub.6 H.sub.13                                H         CH(CH.sub.3).sub.2                                                                        2-CONH.sub.2                                            H         CH(CH.sub.3).sub.2                                                                        3-CONH.sub.2                                            H         CH(CH.sub.3).sub.2                                                                        4-CONH.sub.2                                            H         CH(CH.sub.3).sub.2                                                                        3-CONHCH.sub.3                                          H         CH(CH.sub.3).sub.2                                                                        4-CONHCH.sub.3                                          H         CH(CH.sub.3).sub.2                                                                        3-CON(CH.sub.3).sub.2                                   H         CH(CH.sub.3).sub.2                                                                        4-CON(CH.sub.3).sub.2                                   H         CH(CH.sub.3).sub.2                                                                        3-CON(C.sub.2 H.sub.5).sub.2                            H         CH(CH.sub.3).sub.2                                                                        4-CON(C.sub.2 H.sub.5).sub.2                            H         CH(CH.sub.3).sub.2                                                                        2-CSNH.sub.2                                            H         CH(CH.sub.3).sub.2                                                                        3-CSNH.sub.2                                            H         CH(CH.sub.3).sub.2                                                                        4-CSNH.sub.2                                            H         CH(CH.sub.3).sub.2                                                                        2-NH.sub.2                                              H         CH(CH.sub.3).sub.2                                                                        3-NH.sub.2                                              H         CH(CH.sub.3).sub.2                                                                        4-NH.sub.2                                              H         CH(CH.sub.3).sub.2                                                                        3-NHCH.sub.3                                            H         CH(CH.sub.3).sub.2                                                                        4-NHCH.sub.3                                            H         CH(CH.sub.3).sub.2                                                                        3-N(CH.sub.3).sub.2                                     H         CH(CH.sub.3).sub.2                                                                        4-N(CH.sub.3).sub.2                                     H         CH(CH.sub.3).sub.2                                                                        3-NHCO--CH.sub.3                                        H         CH(CH.sub.3).sub.2                                                                        4-NHCO--CH.sub.3                                        H         CH(CH.sub.3).sub.2                                                                        3-NCH.sub.3 --CO--CH.sub.3                              H         CH(CH.sub.3).sub.2                                                                        4-NCH.sub.3 --CO--CH.sub.3                              H         CH(CH.sub.3).sub.2                                                                        3-NHCOOCH.sub.3                                         H         CH(CH.sub.3).sub.2                                                                        4-NHCOOCH.sub.3                                         H         CH(CH.sub.3).sub.2                                                                        3-NCH.sub.3 --COOCH.sub.3                               H         CH(CH.sub.3).sub.2                                                                        4-NCH.sub.3 --COOCH.sub.3                               H         CH(CH.sub.3).sub.2                                                                        3-OCO--CH.sub.3                                         H         CH(CH.sub.3).sub.2                                                                        4-OCO--CH.sub.3                                         H         CH(CH.sub.3).sub.2                                                                        3-OCO-t-C.sub.4 H.sub.9                                 H         CH(CH.sub.3).sub.2                                                                        4-OCO-t-C.sub.4 H.sub.9                                 H         CH(CH.sub.3).sub.2                                                                        3-SH                                                    H         CH(CH.sub.3).sub.2                                                                        4-SH                                                    H         CH(CH.sub.3).sub.2                                                                        3-SCH.sub.3                                             H         CH(CH.sub.3).sub.2                                                                        4-SCH.sub.3                                             H         CH(CH.sub.3).sub.2                                                                        3-S-t-C.sub.4 H.sub.9                                   H         CH(CH.sub.3).sub.2                                                                        4-S-t-C.sub.4 H.sub.9                                   H         CH(CH.sub.3).sub.2                                                                        3-SO--CH.sub.3                                          H         CH(CH.sub.3).sub.2                                                                        4-SO--CH.sub.3                                          H         CH(CH.sub.3).sub.2                                                                        3-SO.sub.2 CH.sub.3                                     H         CH(CH.sub.3).sub.2                                                                        4-SO.sub.2 CH.sub.3                                     H         CH(CH.sub.3).sub.2                                                                        3-CH═NCH.sub.3                                      H         CH(CH.sub.3).sub.2                                                                        4-CH═NCH.sub.3                                      H         CH(CH.sub.3).sub.2                                                                        3-C(CH.sub.3)═NCH.sub.3                             H         CH(CH.sub.3).sub.2                                                                        4-C(CH.sub.3)═NCH.sub.3                             H         CH(CH.sub.3).sub.2                                                                        3-C(SCH.sub.3)═NOCH.sub.3                           H         CH(CH.sub.3).sub.2                                                                        4-C(SCH.sub.3)═NOCH.sub.3                           H         CH(CH.sub.3).sub.2                                                                        3-C(OCH.sub.3)═NOCH.sub.3                           H         CH(CH.sub.3).sub.2                                                                        4-C(OCH.sub.3)═NOCH.sub.3                           H         CH(CH.sub.3).sub.2                                                                        3-C(NH.sub.2)═NOCH.sub.3                            H         CH(CH.sub.3).sub.2                                                                        4-C(NH.sub.2)═NOCH.sub.3                            H         CH(CH.sub.3).sub.2                                                                        3-C(NHCH.sub.3)═NOCH.sub.3                          H         CH(CH.sub.3).sub.2                                                                        4-C(NHCH.sub.3)═NOCH.sub.3                          H         CH(CH.sub.3).sub.2                                                                        3-CH═NOCH.sub.3                                     H         CH(CH.sub.3).sub.2                                                                        4-CH═NOCH.sub.3                                     H         CH(CH.sub.3).sub.2                                                                        3-C(CH.sub.3)═NOCH.sub.3                            H         CH(CH.sub.3).sub.2                                                                        4-C(CH.sub.3)═NOCH.sub.3                            H         CH(CH.sub.3).sub.2                                                                        3-C(CH.sub.3)═NOC.sub.2 H.sub.5                     H         CH(CH.sub.3).sub.2                                                                        4-C(CH.sub.3)═NOC.sub.2 H.sub.5                     H         CH(CH.sub.3).sub.2                                                                        3-C(CH.sub.3)═NO-n-C.sub.3 H.sub.7                  H         CH(CH.sub.3).sub.2                                                                        4-C(CH.sub.3)═NO-n-C.sub.3 H.sub.7                  H         CH(CH.sub.3).sub.2                                                                        3-C(CH.sub.3)═NO-i-C.sub.3 H.sub.7                  H         CH(CH.sub.3).sub.2                                                                        4-C(CH.sub.3)═NO-i-C.sub.3 H.sub.7                  H         CH(CH.sub.3).sub.2                                                                        3-C(CH.sub.3)═NO-n-C.sub.4 H.sub.9                  H         CH(CH.sub.3).sub.2                                                                        4-C(CH.sub.3)═NO-n-C.sub.4 H.sub.9                  H         CH(CH.sub.3).sub.2                                                                        3-C(CH.sub.3)═NO-s-C.sub.4 H.sub.9                  H         CH(CH.sub.3).sub.2                                                                        4-C(CH.sub.3)═NO-s-C.sub.4 H.sub.9                  H         CH(CH.sub.3).sub.2                                                                        3-C(CH.sub.3)═NO-i-C.sub.4 H.sub.9                  H         CH(CH.sub.3).sub.2                                                                        4-C(CH.sub.3)═NO-i-C.sub.4 H.sub.9                  H         CH(CH.sub.3).sub.2                                                                        3-C(CH.sub.3)═NO-t-C.sub.4 H.sub.9                  H         CH(CH.sub.3).sub.2                                                                        4-C(CH.sub.3)═NO-t-C.sub.4 H.sub.9                  H         CH(CH.sub.3).sub.2                                                                        3-C(CH.sub.3)═NO-n-C.sub.5 H.sub.11                 H         CH(CH.sub.3).sub.2                                                                        4-C(CH.sub.3)═NO-n-C.sub.5 H.sub.11                 H         CH(CH.sub.3).sub.2                                                                        3-C(CH.sub.3)═NO-n-C.sub.6 H.sub.13                 H         CH(CH.sub.3).sub.2                                                                        4-C(CH.sub.3)═NO-n-C.sub.6 H.sub.13                 H         CH(CH.sub.3).sub.2                                                                        2-Cl, 4-CH.sub.3                                        H         CH(CH.sub.3).sub.2                                                                        2-Cl, 5-CH.sub.3                                        H         CH(CH.sub.3).sub.2                                                                        3-Cl, 4-CH.sub.3                                        H         CH(CH.sub.3).sub.2                                                                        3-Cl, 5-CH.sub.3                                        H         CH(CH.sub.3).sub.2                                                                        2-CH.sub.3, 4-Cl                                        H         CH(CH.sub.3).sub.2                                                                        2-CH.sub.3, 5-Cl                                        H         CH(CH.sub.3).sub.2                                                                        3-CH.sub.3, 4-Cl                                        H         CH(CH.sub.3).sub.2                                                                        3-Cl, 5-t-C.sub.4 H.sub.9                               H         CH(CH.sub.3).sub.2                                                                        2-Cl, 4-t-C.sub.4 H.sub.9                               H         CH(CH.sub.3).sub.2                                                                        2-F, 4-CH.sub.3                                         H         CH(CH.sub.3).sub.2                                                                        3-F, 4-CH.sub.3                                         H         CH(CH.sub.3).sub.2                                                                        3-F, 5-CH.sub.3                                         H         CH(CH.sub.3).sub.2                                                                        2-CH.sub.3, 4-F                                         H         CH(CH.sub.3).sub.2                                                                        3-CH.sub.3, 4-F                                         H         CH(CH.sub.3).sub.2                                                                        2-F, 4-t-C.sub.4 H.sub.9                                H         CH(CH.sub.3).sub.2                                                                        3-F, 4-t-C.sub.4 H.sub.9                                H         CH(CH.sub.3).sub.2                                                                        2-F, 4-OCH.sub.3                                        H         CH(CH.sub.3).sub.2                                                                        2-Br, 4-CH.sub.3                                        H         CH(CH.sub.3).sub.2                                                                        3-Br, 4-CH.sub.3                                        H         CH(CH.sub.3).sub.2                                                                        3-Br, 5-CH.sub.3                                        H         CH(CH.sub.3).sub.2                                                                        2-CH.sub.3, 4-Br                                        H         CH(CH.sub.3).sub.2                                                                        3-CH.sub.3, 4-Br                                        H         CH(CH.sub.3).sub.2                                                                        2-Br, 4-t-C.sub.4 H.sub.9                               H         CH(CH.sub.3).sub.2                                                                        2-Cl, 4-NO.sub.2                                        H         CH(CH.sub.3).sub.2                                                                        3-Cl, 4-NO.sub.2                                        H         CH(CH.sub.3).sub.2                                                                        3-Cl, 5-NO.sub.2                                        H         CH(CH.sub.3).sub.2                                                                        3-NO.sub.2, 4-Cl                                        H         CH(CH.sub.3).sub.2                                                                        3-Cl, 4-OCH                                             H         CH(CH.sub.3).sub.2                                                                        3-OCH.sub.3, 4-Cl                                       H         CH(CH.sub.3).sub.2                                                                        2-Cl, 5-CF.sub.3                                        H         CH(CH.sub.3).sub.2                                                                        3-Cl, 4-CF.sub.3                                        H         CH(CH.sub.3).sub.2                                                                        3-Cl, 5-CF.sub.3                                        H         CH(CH.sub.3).sub.2                                                                        3-CF.sub.3, 4-Cl                                        H         CH(CH.sub.3).sub.2                                                                        3-Cl, 5-OCF.sub.3                                       H         CH(CH.sub.3).sub.2                                                                        3-F, 5-CF.sub.3                                         H         CH(CH.sub.3).sub.2                                                                        2-CH.sub.3, 4-CN                                        H         CH(CH.sub.3).sub.2                                                                        3-NO.sub.2, 4-CH.sub.3                                  H         CH(CH.sub.3).sub.2                                                                        2-CH.sub.3, 4-OCH.sub.3                                 H         CH(CH.sub.3).sub.2                                                                        3-CH.sub.3, 4-OCH.sub.3                                 H         CH(CH.sub.3).sub.2                                                                        3-CH.sub.3, 5-OCH.sub.3                                 H         CH(CH.sub.3).sub.2                                                                        3-OCH.sub.3, 4-CH.sub.3                                 H         CH(CH.sub.3).sub.2                                                                        2-CH.sub.3, 4-O-i-C.sub.3 H.sub.7                       H         CH(CH.sub.3).sub.2                                                                        3-CH.sub.3, 4-O-i-C.sub.3 H.sub.7                       H         CH(CH.sub.3).sub.2                                                                        3-O-i-C.sub.3 H.sub.7, 4-CH.sub.3                       H         CH(CH.sub.3).sub.2                                                                        2-CH.sub.3, 4-CF.sub.3                                  H         CH(CH.sub.3).sub.2                                                                        2-CH.sub.3, 5-CF.sub.3                                  H         CH(CH.sub.3).sub.2                                                                        3-CH.sub.3, 4-CF.sub.3                                  H         CH(CH.sub.3).sub.2                                                                        3-CH.sub.3, 5-CF.sub.3                                  H         CH(CH.sub.3).sub.2                                                                        3-CF.sub.3, 4-CH.sub.3                                  H         CH(CH.sub.3).sub.2                                                                        3-CF.sub.3, 4-OCH.sub.3                                 H         CH(CH.sub.3).sub.2                                                                        3-OCH.sub.3, 4-CF.sub.3                                 H         CH(CH.sub.3).sub.2                                                                        2-CH.sub.3, 4-C(CH.sub.3)═NOCH.sub.3                H         CH(CH.sub.3).sub.2                                                                        3-CH.sub.3, 4-C(CH.sub.3)═NOCH.sub.3                H         CH(CH.sub.3).sub.2                                                                        2-OH, 5-CH.sub.3                                        H         CH(CH.sub.3).sub.2                                                                        3-CH.sub.3, 4-OC.sub.2 H.sub.5                          H         CH(CH.sub.3).sub.2                                                                        3-CH.sub.3, 4-O-t-C.sub.4 H.sub.9                       H         CH(CH.sub.3).sub.2                                                                        3-OC.sub.2 H.sub.5, 4-CH.sub.3                          H         CH(CH.sub.3).sub.2                                                                        3-O-t-C.sub.4 H.sub.9, 4-CH.sub.3                       H         CH(CH.sub.3).sub.2                                                                        2-C(COOCH.sub.3)═NOCH.sub.3                         H         CH(CH.sub.3).sub.2                                                                        2,3-Butadienyl                                          H         CH(CH.sub.3).sub.2                                                                        3,4-Butadienyl                                          CH.sub.3  CH(CH.sub.3).sub.2                                                                        H                                                       CH.sub.3  CH(CH.sub.3).sub.2                                                                        2-F                                                     CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-F                                                     CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-F                                                     CH.sub.3  CH(CH.sub.3).sub.2                                                                        2,4-F.sub.2                                             CH.sub.3  CH(CH.sub.3).sub.2                                                                        3,4-F.sub.2                                             CH.sub.3  CH(CH.sub.3).sub.2                                                                        3,5-F.sub.2                                             CH.sub.3  CH(CH.sub.3).sub.2                                                                        2-Cl                                                    CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-Cl                                                    CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-Cl                                                    CH.sub.3  CH(CH.sub.3).sub.2                                                                        2,4-Cl.sub.2                                            CH.sub.3  CH(CH.sub.3).sub.2                                                                        3,4-Cl.sub.2                                            CH.sub.3  CH(CH.sub.3).sub.2                                                                        3,5-Cl.sub.2                                            CH.sub.3  CH(CH.sub.3).sub.2                                                                        2-Br                                                    CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-Br                                                    CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-Br                                                    CH.sub.3  CH(CH.sub.3).sub.2                                                                        3,5-Br.sub.2                                            CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-I                                                     CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-I                                                     CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-F, 5-Cl                                               CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-F, 5-Br                                               CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-Cl, 5-Br                                              CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-Br, 4-F                                               CH.sub.3  CH(CH.sub.3).sub.2                                                                        2-NO.sub.2                                              CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-NO.sub.2                                              CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-NO.sub.2                                              CH.sub.3  CH(CH.sub.3).sub.2                                                                        2-CN                                                    CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-CN                                                    CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-CN                                                    CH.sub.3  CH(CH.sub.3).sub.2                                                                        2-CH.sub.3                                              CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-CH.sub.3                                              CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-CH.sub.3                                              CH.sub.3  CH(CH.sub.3).sub.2                                                                        2,4-(CH.sub.3).sub.2                                    CH.sub.3  CH(CH.sub.3).sub.2                                                                        2,5-(CH.sub.3).sub.2                                    CH.sub.3  CH(CH.sub.3).sub.2                                                                        3,4-(CH.sub.3).sub.2                                    CH.sub.3  CH(CH.sub.3).sub.2                                                                        3,5-(CH.sub.3).sub.2                                    CH.sub.3  CH(CH.sub.3).sub.2                                                                        2,4,5-(CH.sub.3).sub.3                                  CH.sub.3  CH(CH.sub.3).sub.2                                                                        2,4,6-(CH.sub.3).sub.3                                  CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-C.sub.2 H.sub.5                                       CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-C.sub.2 H.sub.5                                       CH.sub.3  CH(CH.sub.3).sub.2                                                                        3,4-(C.sub.2 H.sub.5).sub.2                             CH.sub.3  CH(CH.sub.3).sub.2                                                                        3,5-(C.sub.2 H.sub.5).sub.2                             CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-n-C.sub.3 H.sub.7                                     CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-n-C.sub.3 H.sub.7                                     CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-i-C.sub.3 H.sub.7                                     CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-i-C.sub.3 H.sub.7                                     CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-Cyclopropyl                                           CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-Cyclopropyl                                           CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-n-C.sub.4 H.sub.9                                     CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-n-C.sub.4 H.sub.9                                     CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-t-C.sub.4 H.sub.9                                     CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-t-C.sub.4 H.sub.9                                     CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-n-C.sub.6 H.sub.13                                    CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-n-C.sub.6 H.sub.13                                    CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-Cyclohexyl                                            CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-Cyclohexyl                                            CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-Phenyl                                                CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-Phenyl                                                CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-Allyl                                                 CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-Propargyl                                             CH.sub.3  CH(CH.sub.3).sub.2                                                                        2-CH.sub.3, 4-C.sub.2 H.sub.5                           CH.sub.3  CH(CH.sub.3).sub.2                                                                        2-CH.sub.3, 4-i-C.sub.3 H.sub.7                         CH.sub.3  CH(CH.sub.3).sub.2                                                                        2-CH.sub.3, 4-t-C.sub.4 H.sub.9                         CH.sub.3  CH(CH.sub.3).sub.2                                                                        2-CH.sub.3, 4-phenyl                                    CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-CH.sub.3, 4-phenyl                                    CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-OH                                                    CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-OH                                                    CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-OCH.sub.3                                             CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-OCH.sub.3                                             CH.sub.3  CH(CH.sub.3).sub.2                                                                        3,4-(OCH.sub.3).sub.2                                   CH.sub.3  CH(CH.sub.3).sub.2                                                                        3,5-(OCH.sub.3).sub.2                                   CH.sub.3  CH(CH.sub.3).sub.2                                                                        3,4,5-(OCH.sub.3).sub.3                                 CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-OC.sub.2 H.sub.5                                      CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-O-i-C.sub.3 H.sub.7                                   CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-O-t-C.sub.4 H.sub.9                                   CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-O-t-C.sub.4 H.sub.9                                   CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-O-n-C.sub.6 H.sub.13                                  CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-O-Phenyl                                              CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-O-Phenyl                                              CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-O-Allyl                                               CH.sub.3  CH(CH.sub.3).sub.2                                                                        2-CF.sub.3                                              CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-CF.sub.3                                              CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-CF.sub.3                                              CH.sub.3  CH(CH.sub.3).sub.2                                                                        3,5-(CF.sub.3).sub.2                                    CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-CH.sub.2 CF.sub.3                                     CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-C.sub.2 F.sub.5                                       CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-CF.sub.2 CHF.sub.2                                    CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-OCF.sub.3                                             CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-OCF.sub.3                                             CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-OCH.sub.2 CF.sub.3                                    CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-OC.sub.2 F.sub.5                                      CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-OCF.sub.2 CHF.sub.2                                   CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-CH.sub.2 OCH.sub.3                                    CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-CH.sub.2 OCH.sub.3                                    CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-CH.sub.2 --O-t-C.sub.4 H.sub.9                        CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-CH(OCH.sub.3).sub.2                                   CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-CH.sub.2 CN                                           CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-CHO                                                   CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-CHO                                                   CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-CO--CH.sub.3                                          CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-CO--CH.sub.3                                          CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-COOH                                                  CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-COOH                                                  CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-COOCH.sub.3                                           CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-COOCH.sub.3                                           CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-COOC.sub.2 H.sub.5                                    CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-COOC.sub.2 H.sub.5                                    CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-COO-i-C.sub.3 H.sub.7                                 CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-COO-i-C.sub.3 H.sub.7                                 CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-COO-t-C.sub.4 H.sub.9                                 CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-COO-t-C.sub.4 H.sub.9                                 CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-COO-n-C.sub.6 H.sub.13                                CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-COO-n-C.sub.6 H.sub.13                                CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-CONH.sub.2                                            CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-CONH.sub.2                                            CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-CONHCH.sub.3                                          CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-CONHCH.sub.3                                          CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-CON(CH.sub.3).sub.2                                   CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-CON(CH.sub.3).sub.2                                   CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-CSNH.sub.2                                            CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-CSNH.sub.2                                            CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-NH.sub.2                                              CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-NH.sub.2                                              CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-NHCH.sub.3                                            CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-N(CH.sub.3).sub.2                                     CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-NHCO--CH.sub.3                                        CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-NHCO--CH.sub.3                                        CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-NCH.sub.3 --CO--CH.sub.3                              CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-NHCOOCH.sub.3                                         CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-NCH.sub.3 --COOCH.sub.3                               CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-OCO--CH.sub.3                                         CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-OCO--CH.sub.3                                         CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-OCO-t-C.sub.4 H.sub.9                                 CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-SH                                                    CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-SCH.sub.3                                             CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-S-t-C.sub.4 H.sub.9                                   CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-SO--CH.sub.3                                          CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-SO.sub.2 --CH.sub.3                                   CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-C(CH.sub.3)═NCH.sub.3                             CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-C(SCH.sub.3)═NOCH.sub.3                           CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-C(OCH.sub.3)═NOCH.sub.3                           CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-CH═NOCH.sub.3                                     CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-CH═NOCH.sub.3                                     CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-C(CH.sub.3)═NOCH.sub.3                            CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-C(CH.sub.3)═NOCH.sub.3                            CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-C(CH.sub.3)═NOC.sub.2 H.sub.5                     CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-C(CH.sub.3)═NO-n-C.sub.3 H.sub.7                  CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-C(CH.sub.3)═NO-i-C.sub.3 H.sub.7                  CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-C(CH.sub.3)═NO-n-C.sub.4 H.sub.9                  CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-C(CH.sub.3)═NO-t-C.sub.4 H.sub.9                  CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-C(CH.sub.3)═NO-n-C.sub.5 H.sub.11                 CH.sub.3  CH(CH.sub.3).sub.2                                                                        4-C(CH.sub.3)═NO-n-C.sub.6 H.sub.13                 CH.sub.3  CH(CH.sub.3).sub.2                                                                        2-Cl, 4-CH.sub.3                                        CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-Cl, 5-CH.sub.3                                        CH.sub.3  CH(CH.sub.3).sub.2                                                                        2-CH.sub.3, 4-Cl                                        CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-CH.sub.3, 4-Cl                                        CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-F, 5-CH.sub.3                                         CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-Br, 5-CH.sub.3                                        CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-Cl, 5-NO.sub.2                                        CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-NO.sub.2, 4-Cl                                        CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-Cl, 4-OCH.sub.3                                       CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-OCH.sub.3, 4-Cl                                       CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-Cl, 5-CF.sub.3                                        CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-Cl, 5-OCF.sub.3                                       CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-F, 5-CF.sub.3                                         CH.sub.3  CH(CH.sub.3).sub.2                                                                        2-CH.sub.3, 4-CN                                        CH.sub.3  CH(CH.sub.3).sub.2                                                                        2-CH.sub.3, 4-OCH.sub.3                                 CH.sub.3  CH(CH.sub.3).sub.2                                                                        2-CH.sub.3, 4-CF.sub.3                                  CH.sub.3  CH(CH.sub.3).sub.2                                                                        2-CH.sub.3, 4-C(CH.sub.3)═NOCH.sub.3                CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-CH.sub.3, 4-C(CH.sub.3)═NOCH.sub.3                CH.sub.3  CH(CH.sub.3).sub.2                                                                        2-OH, 5-CH.sub.3                                        CH.sub.3  CH(CH.sub.3).sub.2                                                                        3-CH.sub.3, 4-O-t-C.sub.4 H.sub.9                       CH.sub.3  CH(CH.sub.3).sub.2                                                                        2-C(COOCH.sub.3)═NOCH.sub.3                         CH.sub.3  CH(CH.sub.3).sub.2                                                                        2,3-Butadienyl                                          CH.sub.3  CH(CH.sub.3).sub.2                                                                        3,4-Butadienyl                                          H         CF.sub.3    H                                                       H         CF.sub.3    2-F                                                     H         CF.sub.3    3-F                                                     H         CF.sub.3    4-F                                                     H         CF.sub.3    2,3-F.sub.2                                             H         CF.sub.3    2,4-F.sub.2                                             H         CF.sub.3    2,5-F.sub.2                                             H         CF.sub.3    2,6-F.sub.2                                             H         CF.sub.3    3,4-F.sub.2                                             H         CF.sub.3    3,5-F.sub.2                                             H         CF.sub.3    2-Cl                                                    H         CF.sub.3    3-Cl                                                    H         CF.sub.3    4-Cl                                                    H         CF.sub.3    2,4-Cl.sub.2                                            H         CF.sub.3    2,5-Cl.sub.2                                            H         CF.sub.3    3,4-Cl.sub.2                                            H         CF.sub.3    3,5-Cl.sub.2                                            H         CF.sub.3    2-Br                                                    H         CF.sub.3    3-Br                                                    H         CF.sub.3    4-Br                                                    H         CF.sub.3    2,4-Br.sub.2                                            H         CF.sub.3    3,4-Br.sub.2                                            H         CF.sub.3    3,5-Br.sub.2                                            H         CF.sub.3    2-I                                                     H         CF.sub.3    3-I                                                     H         CF.sub.3    4-I                                                     H         CF.sub.3    2-F, 4-Cl                                               H         CF.sub.3    2-F, 5-Cl                                               H         CF.sub.3    2-F, 4-Br                                               H         CF.sub.3    2-F, 5-Br                                               H         CF.sub.3    2-Cl, 4-Br                                              H         CF.sub.3    2-Cl, 5-Br                                              H         CF.sub.3    3-F, 4-Cl                                               H         CF.sub.3    3-F, 5-Cl                                               H         CF.sub.3    3-F, 4-Br                                               H         CF.sub.3    3-F, 5-Br                                               H         CF.sub.3    3-Cl, 4-Br                                              H         CF.sub.3    3-Cl, 5-Br                                              H         CF.sub.3    3-Cl, 4-F                                               H         CF.sub.3    3-Br, 4-F                                               H         CF.sub.3    3-Br, 4-Cl                                              H         CF.sub.3    2-NO.sub.2                                              H         CF.sub.3    3-NO.sub.2                                              H         CF.sub.3    4-NO.sub.2                                              H         CF.sub.3    2-CN                                                    H         CF.sub.3    3-CN                                                    H         CF.sub.3    4-CN                                                    H         CF.sub.3    2-CH.sub.3                                              H         CF.sub.3    3-CH.sub.3                                              H         CF.sub.3    4-CH.sub.3                                              H         CF.sub.3    2,3-(CH.sub.3).sub.2                                    H         CF.sub.3    2,4-(CH.sub.3).sub.2                                    H         CF.sub.3    2,5-(CH.sub.3).sub.2                                    H         CF.sub.3    2,6-(CH.sub.3).sub.2                                    H         CF.sub.3    3,4-(CH.sub.3).sub.2                                    H         CF.sub.3    3,5-(CH.sub.3).sub.2                                    H         CF.sub.3    2,4,5-(CH.sub.3).sub.3                                  H         CF.sub.3    2,4,6-(CH.sub.3).sub.3                                  H         CF.sub.3    3,4,5-(CH.sub.3).sub.3                                  H         CF.sub.3    2-C.sub.2 H.sub.5                                       H         CF.sub.3    3-C.sub.2 H.sub.5                                       H         CF.sub.3    4-C.sub.2 H.sub.5                                       H         CF.sub.3    3,4-(C.sub.2 H.sub.5).sub.2                             H         CF.sub.3    3,5-(C.sub.2 H.sub.5).sub.2                             H         CF.sub.3    3-n-C.sub.3 H.sub.7                                     H         CF.sub.3    4-n-C.sub.3 H.sub.7                                     H         CF.sub.3    3,4-(n-C.sub.3 H.sub.7).sub.2                           H         CF.sub.3    3,5-(n-C.sub.3 H.sub.7).sub.2                           H         CF.sub.3    3-i-C.sub.3 H.sub.7                                     H         CF.sub.3    4-i-C.sub.3 H.sub.7                                     H         CF.sub.3    3,4-(i-C.sub.3 H.sub.7).sub.2                           H         CF.sub.3    3,5-(i-C.sub.3 H.sub.7).sub.2                           H         CF.sub.3    3-Cyclopropyl                                           H         CF.sub.3    4-Cyclopropyl                                           H         CF.sub.3    3-n-C.sub.4 H.sub.9                                     H         CF.sub.3    4-n-C.sub.4 H.sub.9                                     H         CF.sub.3    3,4-(n-C.sub.4 H.sub.9).sub.2                           H         CF.sub.3    3,5-(n-C.sub.4 H.sub.9).sub.2                           H         CF.sub.3    3-s-C.sub.4 H.sub.9                                     H         CF.sub.3    4-s-C.sub.4 H.sub.9                                     H         CF.sub.3    3-i-C.sub.4 H.sub.9                                     H         CF.sub.3    4-i-C.sub.4 H.sub.9                                     H         CF.sub.3    3-t-C.sub.4 H.sub.9                                     H         CF.sub.3    4-t-C.sub.4 H.sub.9                                     H         CF.sub.3    3,4-(t-C.sub.4 H.sub.9).sub.2                           H         CF.sub.3    3,5-(t-C.sub.4 H.sub.9).sub.2                           H         CF.sub.3    3-n-C.sub.5 H.sub.11                                    H         CF.sub.3    4-n-C.sub.5 H.sub.11                                    H         CF.sub.3    3-n-C.sub.6 H.sub.13                                    H         CF.sub.3    4-n-C.sub.6 H.sub.13                                    H         CF.sub.3    3-Cyclohexyl                                            H         CF.sub.3    4-Cyclohexyl                                            H         CF.sub.3    3-Phenyl                                                H         CF.sub.3    4-Phenyl                                                H         CF.sub.3    3-Vinyl                                                 H         CF.sub.3    4-Vinyl                                                 H         CF.sub.3    3-Allyl                                                 H         CF.sub.3    4-Allyl                                                 H         CF.sub.3    3-Propargyl                                             H         CF.sub.3    4-Propargyl                                             H         CF.sub.3    3-(Propen-2-yl)                                         H         CF.sub.3    4-(Propen-2-yl)                                         H         CF.sub.3    2-CH.sub.3, 4-C.sub.2 H.sub.5                           H         CF.sub.3    2-CH.sub.3, 5-C.sub.2 H.sub.5                           H         CF.sub.3    2-CH.sub.3, 4-n-C.sub.3 H.sub.7                         H         CF.sub.3    2-CH.sub.3, 5-n-C.sub.3 H.sub.7                         H         CF.sub.3    2-CH.sub.3, 4-i-C.sub.3 H.sub.7                         H         CF.sub.3    2-CH.sub.3, 5-i-C.sub.3 H.sub.7                         H         CF.sub.3    2-CH.sub.3, 4-n-C.sub.4 H.sub.9                         H         CF.sub.3    2-CH.sub.3, 4-s-C.sub.4 H.sub.9                         H         CF.sub.3    2-CH.sub.3, 4-i-C.sub.4 H.sub.9                         H         CF.sub.3    2-CH.sub.3, 4-t-C.sub.4 H.sub.9                         H         CF.sub.3    2-CH.sub.3, 4-phenyl                                    H         CF.sub.3    2-CH.sub.3, 5-phenyl                                    H         CF.sub.3    2-CH.sub.3, 4-vinyl                                     H         CF.sub.3    2-CH.sub.3, 4-allyl                                     H         CF.sub.3    2-CH.sub.3, 4-propargyl                                 H         CF.sub.3    2-CH.sub.3, 4-(propen-2-yl)                             H         CF.sub.3    3-CH.sub.3, 4-C.sub.2 H.sub.5                           H         CF.sub.3    3-CH.sub.3, 5-C.sub.2 H.sub.5                           H         CF.sub.3    3-CH.sub.3, 4-n-C.sub.3 H.sub.7                         H         CF.sub.3    3-CH.sub.3, 5-n-C.sub.3 H.sub.7                         H         CF.sub.3    3-CH.sub.3, 4-i-C.sub.3 H.sub.7                         H         CF.sub.3    3-CH.sub.3, 5-i-C.sub.3 H.sub.7                         H         CF.sub.3    3-CH.sub.3, 4-cyclopropyl                               H         CF.sub.3    3-CH.sub.3, 4-t-C.sub.4 H.sub.9                         H         CF.sub.3    3-CH.sub.3, 5-t-C.sub.4 H.sub.9                         H         CF.sub.3    3-CH.sub.3, 4-phenyl                                    H         CF.sub.3    3-CH.sub.3, 5-phenyl                                    H         CF.sub.3    3-CH.sub.3, 4-vinyl                                     H         CF.sub.3    3-CH.sub.3, 4-allyl                                     H         CF.sub.3    3-CH.sub.3, 4-propargyl                                 H         CF.sub.3    3-CH.sub.3, 4-propen-2-yl                               H         CF.sub.3    3-C.sub.2 H.sub.5, 4-CH.sub.3                           H         CF.sub.3    3-i-C.sub.3 H.sub.7, 4-CH.sub.3                         H         CF.sub.3    3-t-C.sub.4 H.sub.9, 4-CH.sub.3                         H         CF.sub.3    3-Phenyl, 4-CH.sub.3                                    H         CF.sub.3    2-OH                                                    H         CF.sub.3    3-OH                                                    H         CF.sub.3    4-OH                                                    H         CF.sub.3    2-OCH.sub.3                                             H         CF.sub.3    3-OCH.sub.3                                             H         CF.sub.3    4-OCH.sub.3                                             H         CF.sub.3    2,3-(OCH.sub.3).sub.2                                   H         CF.sub.3    2,4-(OCH.sub.3).sub.2                                   H         CF.sub.3    2,5-(OCH.sub.3).sub.2                                   H         CF.sub.3    3,4-(OCH.sub.3).sub.2                                   H         CF.sub.3    3,5-(OCH.sub.3).sub.2                                   H         CF.sub.3    3,4,5-(OCH.sub.3).sub.3                                 H         CF.sub.3    3-OC.sub.2 H.sub.5                                      H         CF.sub.3    4-OC.sub.2 H.sub.5                                      H         CF.sub.3    3,4-(OC.sub.2 H.sub.5).sub.2                            H         CF.sub.3    3,5-(OC.sub.2 H.sub.5).sub.2                            H         CF.sub.3    3-O-n-C.sub.3 H.sub.7                                   H         CF.sub.3    4-O-n-C.sub.3 H.sub.7                                   H         CF.sub.3    3-O-i-C.sub.3 H.sub.7                                   H         CF.sub.3    4-O-i-C.sub.3 H.sub.7                                   H         CF.sub.3    3-O-Cyclopropyl                                         H         CF.sub.3    4-O-Cyclopropyl                                         H         CF.sub.3    3-O-n-C.sub.4 H.sub.9                                   H         CF.sub.3    4-O-n-C.sub.4 H.sub.9                                   H         CF.sub.3    3-O-s-C.sub.4 H.sub.9                                   H         CF.sub.3    4-O-s-C.sub.4 H.sub.9                                   H         CF.sub.3    3-O-i-C.sub.4 H.sub.9                                   H         CF.sub.3    4-O-i-C.sub.4 H.sub.9                                   H         CF.sub.3    3-O-t-C.sub.4 H.sub.9                                   H         CF.sub.3    4-O-t-C.sub.4 H.sub.9                                   H         CF.sub.3    3-O-n-C.sub.5 H.sub.11                                  H         CF.sub.3    4-O-n-C.sub.5 H.sub.11                                  H         CF.sub.3    3-O-n-C.sub.6 H.sub.13                                  H         CF.sub.3    4-O-n-C.sub.6 H.sub.13                                  H         CF.sub.3    3-O-Cyclohexyl                                          H         CF.sub.3    4-O-Cyclohexyl                                          H         CF.sub.3    3-O-Phenyl                                              H         CF.sub.3    4-O-Phenyl                                              H         CF.sub.3    3-O-Allyl                                               H         CF.sub.3    4-O-Allyl                                               H         CF.sub.3    2-CF.sub.3                                              H         CF.sub.3    3-CF.sub.3                                              H         CF.sub.3    4-CF.sub.3                                              H         CF.sub.3    2,4-(CF.sub.3).sub.2                                    H         CF.sub.3    3,5-(CF.sub.3).sub.2                                    H         CF.sub.3    3-CF.sub.2 Cl                                           H         CF.sub.3    4-CF.sub.2 Cl                                           H         CF.sub.3    3-CFCl.sub.2                                            H         CF.sub.3    4-CFCl.sub.2                                            H         CF.sub.3    3-CCl.sub.3                                             H         CF.sub.3    4-CCl.sub.3                                             H         CF.sub.3    3-CH.sub.2 CH.sub.2 F                                   H         CF.sub.3    4-CH.sub.2 CH.sub.2 F                                   H         CF.sub.3    3-CH.sub.2 CF.sub.3                                     H         CF.sub.3    4-CH.sub.2 CF.sub.3                                     H         CF.sub.3    3-C.sub.2 F.sub.5                                       H         CF.sub.3    5-C.sub.2 F.sub.5                                       H         CF.sub.3    3-CHCl.sub.2                                            H         CF.sub.3    4-CHCl.sub.2                                            H         CF.sub.3    3-CH.sub.2 Cl                                           H         CF.sub.3    4-CH.sub.2 Cl                                           H         CF.sub.3    3-CF.sub.2 CHF.sub.2                                    H         CF.sub.3    4-CF.sub.2 CHF.sub.2                                    H         CF.sub.3    3-CH.sub.2 CH.sub.2 Cl                                  H         CF.sub.3    4-CH.sub.2 CH.sub.2 Cl                                  H         CF.sub.3    2-OCF.sub.3                                             H         CF.sub.3    3-OCF.sub.3                                             H         CF.sub.3    4-OCF.sub.3                                             H         CF.sub.3    3-OCHF.sub.2                                            H         CF.sub.3    4-OCHF.sub.2                                            H         CF.sub.3    3-OC.sub.2 F.sub.5                                      H         CF.sub.3    4-OC.sub.2 F.sub.5                                      H         CF.sub.3    3-OCF.sub.2 CHF.sub.2                                   H         CF.sub.3    4-OCF.sub.2 CHF.sub.2                                   H         CF.sub.3    3-CH.sub.2 OCH.sub.3                                    H         CF.sub.3    4-CH.sub.2 OCH.sub.3                                    H         CF.sub.3    3-CH.sub.2 O-t-C.sub.4 H.sub.9                          H         CF.sub.3    4-CH.sub.2 O-t-C.sub.4 H.sub.9                          H         CF.sub.3    3-C(CH.sub.3)(OCH.sub.3).sub.2                          H         CF.sub.3    4-C(CH.sub.3)(OCH.sub.3).sub.2                          H         CF.sub.3    3-CH(OCH.sub.3).sub.2                                   H         CF.sub.3    4-CH(OCH.sub.3).sub.2                                   H         CF.sub.3    3-CH.sub.2 CN                                           H         CF.sub.3    4-CH.sub.2 CN                                           H         CF.sub.3    3-CHO                                                   H         CF.sub.3    4-CHO                                                   H         CF.sub.3    3-CO--CH.sub.3                                          H         CF.sub.3    4-CO--CH.sub.3                                          H         CF.sub.3    3-CO--C.sub.2 H.sub.5                                   H         CF.sub.3    4-CO--C.sub.2 H.sub.5                                   H         CF.sub.3    2-COOH                                                  H         CF.sub.3    3-COOH                                                  H         CF.sub.3    4-COOH                                                  H         CF.sub.3    3-COOCH.sub.3                                           H         CF.sub.3    4-COOCH.sub.3                                           H         CF.sub.3    3-COOC.sub.2 H.sub.5                                    H         CF.sub.3    4-COOC.sub.2 H.sub.5                                    H         CF.sub.3    3-COO-n-C.sub.3 H.sub.7                                 H         CF.sub.3    4-COO-n-C.sub.3 H.sub.7                                 H         CF.sub.3    3-COO-i-C.sub.3 H.sub.7                                 H         CF.sub.3    4-COO-i-C.sub.3 H.sub.7                                 H         CF.sub.3    3-COO-n-C.sub.4 H.sub.9                                 H         CF.sub.3    4-COO-n-C.sub.4 H.sub.9                                 H         CF.sub.3    3-COO-s-C.sub.4 H.sub.9                                 H         CF.sub.3    4-COO-s-C.sub.4 H.sub.9                                 H         CF.sub.3    3-COO-i-C.sub.4 H.sub.9                                 H         CF.sub.3    4-COO-i-C.sub.4 H.sub.9                                 H         CF.sub.3    3-COO-t-C.sub.4 H.sub.9                                 H         CF.sub.3    4-COO-t-C.sub.4 H.sub.9                                 H         CF.sub.3    3-COO-n-C.sub.5 H.sub.11                                H         CF.sub.3    4-COO-n-C.sub.5 H.sub.11                                H         CF.sub.3    3-COO-n-C.sub.6 H.sub.13                                H         CF.sub.3    4-COO-n-C.sub.6 H.sub.13                                H         CF.sub.3    2-CONH.sub.2                                            H         CF.sub.3    3-CONH.sub.2                                            H         CF.sub.3    4-CONH.sub.2                                            H         CF.sub.3    3-CONHCH.sub.3                                          H         CF.sub.3    4-CONHCH.sub.3                                          H         CF.sub.3    3-CON(CH.sub.3).sub.2                                   H         CF.sub.3    4-CON(CH.sub.3).sub.2                                   H         CF.sub.3    3-CON(C.sub.2 H.sub.5).sub.2                            H         CF.sub.3    4-CON(C.sub.2 H.sub.5).sub.2                            H         CF.sub.3    2-CSNH.sub.2                                            H         CF.sub.3    3-CSNH.sub.2                                            H         CF.sub.3    4-CSNH.sub.2                                            H         CF.sub.3    2-NH.sub.2                                              H         CF.sub.3    3-NH.sub.2                                              H         CF.sub.3    4-NH.sub.2                                              H         CF.sub.3    3-NHCH.sub.3                                            H         CF.sub.3    4-NHCH.sub.3                                            H         CF.sub.3    3-N(CH.sub.3).sub.2                                     H         CF.sub.3    4-N(CH.sub.3).sub.2                                     H         CF.sub.3    3-NHCO--CH.sub.3                                        H         CF.sub.3    4-NHCO--CH.sub.3                                        H         CF.sub.3    3-NCH.sub.3 --CO--CH.sub.3                              H         CF.sub.3    4-NCH.sub.3 --CO--CH.sub.3                              H         CF.sub.3    3-NHCOOCH.sub.3                                         H         CF.sub.3    4-NHCOOCH.sub.3                                         H         CF.sub.3    3-NCH.sub.3 --COOCH.sub.3                               H         CF.sub.3    4-NCH.sub.3 --COOCH.sub.3                               H         CF.sub.3    3-OCO--CH.sub.3                                         H         CF.sub.3    4-OCO--CH.sub.3                                         H         CF.sub.3    3-OCO-t-C.sub.4 H.sub.9                                 H         CF.sub.3    4-OCO-t-C.sub.4 H.sub.9                                 H         CF.sub.3    3-SH                                                    H         CF.sub.3    4-SH                                                    H         CF.sub.3    3-SCH.sub.3                                             H         CF.sub.3    4-SCH.sub.3                                             H         CF.sub.3    3-S-t-C.sub.4 H.sub.9                                   H         CF.sub.3    4-S-t-C.sub.4 H.sub.9                                   H         CF.sub.3    3-SO--CH.sub.3                                          H         CF.sub.3    4-SO--CH.sub.3                                          H         CF.sub.3    3-SO.sub.2 CH.sub.3                                     H         CF.sub.3    4-SO.sub.2 CH.sub.3                                     H         CF.sub.3    3-CH═NCH.sub.3                                      H         CF.sub.3    4-CH═NCH.sub.3                                      H         CF.sub.3    3-C(CH.sub.3)═NCH.sub.3                             H         CF.sub.3    4-C(CH.sub.3)═NCH.sub.3                             H         CF.sub.3    3-C(SCH.sub.3)═NOCH.sub.3                           H         CF.sub.3    4-C(SCH.sub.3)═NOCH.sub.3                           H         CF.sub.3    3-C(OCH.sub.3)═NOCH.sub.3                           H         CF.sub.3    4-C(OCH.sub.3)═NOCH.sub.3                           H         CF.sub.3    3-C(NH.sub.2)═NOCH.sub.3                            H         CF.sub.3    4-C(NH.sub.2)═NOCH.sub.3                            H         CF.sub.3    3-C(NHCH.sub.3)═NOCH.sub.3                          H         CF.sub.3    4-C(NHCH.sub.3)═NOCH.sub.3                          H         CF.sub.3    3-CH═NOCH.sub.3                                     H         CF.sub.3    4-CH═NOCH.sub.3                                     H         CF.sub.3    3-C(CH.sub.3)═NOCH.sub.3                            H         CF.sub.3    4-C(CH.sub.3)═NOCH.sub.3                            H         CF.sub.3    3-C(CH.sub.3)═NOC.sub.2 H.sub.5                     H         CF.sub.3    4-C(CH.sub.3)═NOC.sub.2 H.sub.5                     H         CF.sub.3    3-C(CH.sub.3)═NO-n-C.sub.3 H.sub.7                  H         CF.sub.3    4-C(CH.sub.3)═NO-n-C.sub.3 H.sub.7                  H         CF.sub.3    3-C(CH.sub.3)═NO-i-C.sub.3 H.sub.7                  H         CF.sub.3    4-C(CH.sub.3)═NO-i-C.sub.3 H.sub.7                  H         CF.sub.3    3-C(CH.sub.3)═NO-n-C.sub.4 H.sub.9                  H         CF.sub.3    4-C(CH.sub.3)═NO-n-C.sub.4 H.sub.9                  H         CF.sub.3    3-C(CH.sub.3)═NO-s-C.sub.4 H.sub.9                  H         CF.sub.3    4-C(CH.sub.3)═NO-s-C.sub.4 H.sub.9                  H         CF.sub.3    3-C(CH.sub.3)═NO-i-C.sub.4 H.sub.9                  H         CF.sub.3    4-C(CH.sub.3)═NO-i-C.sub.4 H.sub.9                  H         CF.sub.3    3-C(CH.sub.3)═NO-t-C.sub.4 H.sub.9                  H         CF.sub.3    4-C(CH.sub.3)═NO-t-C.sub.4 H.sub.9                  H         CF.sub.3    3-C(CH.sub.3)═NO-n-C.sub.5 H.sub.11                 H         CF.sub.3    4-C(CH.sub.3)═NO-n-C.sub.5 H.sub.11                 H         CF.sub.3    3-C(CH.sub.3)═NO-n-C.sub.6 H.sub.13                 H         CF.sub.3    4-C(CH.sub.3)═NO-n-C.sub.6 H.sub.13                 H         CF.sub.3    2-Cl, 4-CH.sub.3                                        H         CF.sub.3    2-Cl, 5-CH.sub.3                                        H         CF.sub.3    3-Cl, 4-CH.sub.3                                        H         CF.sub.3    3-Cl, 5-CH.sub.3                                        H         CF.sub.3    2-CH.sub.3, 4-Cl                                        H         CF.sub.3    2-CH.sub.3, 5-Cl                                        H         CF.sub.3    3-CH.sub.3, 4-Cl                                        H         CF.sub.3    3-Cl, 5-t-C.sub.4 H.sub.9                               H         CF.sub.3    2-Cl, 4-t-C.sub.4 H.sub.9                               H         CF.sub.3    2-F, 4-CH.sub.3                                         H         CF.sub.3    3-F, 4-CH.sub.3                                         H         CF.sub.3    3-F, 5-CH.sub.3                                         H         CF.sub.3    2-CH.sub.3, 4-F                                         H         CF.sub.3    3-CH.sub.3, 4-F                                         H         CF.sub.3    2-F, 4-t-C.sub.4 H.sub.9                                H         CF.sub.3    3-F, 4-t-C.sub.4 H.sub.9                                H         CF.sub.3    2-F, 4-OCH.sub.3                                        H         CF.sub.3    2-Br, 4-CH.sub.3                                        H         CF.sub.3    3-Br, 4-CH.sub.3                                        H         CF.sub.3    3-Br, 5-CH.sub.3                                        H         CF.sub.3    2-CH.sub.3, 4-Br                                        H         CF.sub.3    3-CH.sub.3, 4-Br                                        H         CF.sub.3    2-Br, 4-t-C.sub.4 H.sub.9                               H         CF.sub.3    2-Cl, 4-NO.sub.2                                        H         CF.sub.3    3-Cl, 4-NO.sub.2                                        H         CF.sub.3    3-Cl, 5-NO.sub.2                                        H         CF.sub.3    3-NO.sub.2, 4-Cl                                        H         CF.sub.3    3-Cl, 4-OCH                                             H         CF.sub.3    3-OCH.sub.3, 4-Cl                                       H         CF.sub.3    2-Cl, 5-CF.sub.3                                        H         CF.sub.3    3-Cl, 4-CF.sub.3                                        H         CF.sub.3    3-Cl, 5-CF.sub.3                                        H         CF.sub.3    3-CF.sub.3, 4-Cl                                        H         CF.sub.3    3-Cl, 5-OCF.sub.3                                       H         CF.sub.3    3-F, 5-CF.sub.3                                         H         CF.sub.3    2-CH.sub.3, 4-CN                                        H         CF.sub.3    3-NO.sub.2, 4-CH.sub.3                                  H         CF.sub.3    2-CH.sub.3, 4-OCH.sub.3                                 H         CF.sub.3    3-CH.sub.3, 4-OCH.sub.3                                 H         CF.sub.3    3-CH.sub.3, 5-OCH.sub.3                                 H         CF.sub.3    3-OCH.sub.3, 4-CH.sub.3                                 H         CF.sub.3    2-CH.sub.3, 4-O-i-C.sub.3 H.sub.7                       H         CF.sub.3    3-CH.sub.3, 4-O-i-C.sub.3 H.sub.7                       H         CF.sub.3    3-O-i-C.sub.3 H.sub.7, 4-CH.sub.3                       H         CF.sub.3    2-CH.sub.3, 4-CF.sub.3                                  H         CF.sub.3    2-CH.sub.3, 5-CF.sub.3                                  H         CF.sub.3    3-CH.sub.3, 4-CF.sub.3                                  H         CF.sub.3    3-CH.sub.3, 5-CF.sub.3                                  H         CF.sub.3    3-CF.sub.3, 4-CH.sub.3                                  H         CF.sub.3    3-CF.sub.3, 4-OCH.sub.3                                 H         CF.sub.3    3-OCH.sub.3, 4-CF.sub.3                                 H         CF.sub.3    2-CH.sub.3, 4-C(CH.sub.3)═NOCH.sub.3                H         CF.sub.3    3-CH.sub.3, 4-C(CH.sub.3)═NOCH.sub.3                H         CF.sub.3    2-OH, 5-CH.sub.3                                        H         CF.sub.3    3-CH.sub.3, 4-OC.sub.2 H.sub.5                          H         CF.sub.3    3-CH.sub.3, 4-O-t-C.sub.4 H.sub.9                       H         CF.sub.3    3-OC.sub.2 H.sub.5, 4-CH.sub.3                          H         CF.sub.3    3-O-t-C.sub.4 H.sub.9, 4-CH.sub.3                       H         CF.sub.3    2-C(COOCH.sub.3)═NOCH.sub.3                         H         CF.sub.3    2,3-Butadienyl                                          H         CF.sub.3    3,4-Butadienyl                                          CH.sub.3  CF.sub.3    H                                                       CH.sub.3  CF.sub.3    2-F                                                     CH.sub.3  CF.sub.3    3-F                                                     CH.sub.3  CF.sub.3    4-F                                                     CH.sub.3  CF.sub.3    2,4-F.sub.2                                             CH.sub.3  CF.sub.3    3,4-F.sub.2                                             CH.sub.3  CF.sub.3    3,5-F.sub.2                                             CH.sub.3  CF.sub.3    2-Cl                                                    CH.sub.3  CF.sub.3    3-Cl                                                    CH.sub.3  CF.sub.3    4-Cl                                                    CH.sub.3  CF.sub.3    2,4-Cl.sub.2                                            CH.sub.3  CF.sub.3    3,4-Cl.sub.2                                            CH.sub.3  CF.sub.3    3,5-Cl.sub.2                                            CH.sub.3  CF.sub.3    2-Br                                                    CH.sub.3  CF.sub.3    3-Br                                                    CH.sub.3  CF.sub.3    4-Br                                                    CH.sub.3  CF.sub.3    3,5-Br.sub.2                                            CH.sub.3  CF.sub.3    3-I                                                     CH.sub.3  CF.sub.3    4-I                                                     CH.sub.3  CF.sub.3    3-F, 5-Cl                                               CH.sub.3  CF.sub.3    3-F, 5-Br                                               CH.sub.3  CF.sub.3    3-Cl, 5-Br                                              CH.sub.3  CF.sub.3    3-Br, 4-F                                               CH.sub.3  CF.sub.3    2-NO.sub.2                                              CH.sub.3  CF.sub.3    3-NO.sub.2                                              CH.sub.3  CF.sub.3    4-NO.sub.2                                              CH.sub.3  CF.sub.3    2-CN                                                    CH.sub.3  CF.sub.3    3-CN                                                    CH.sub.3  CF.sub.3    4-CN                                                    CH.sub.3  CF.sub.3    2-CH.sub.3                                              CH.sub.3  CF.sub.3    3-CH.sub.3                                              CH.sub.3  CF.sub.3    4-CH.sub.3                                              CH.sub.3  CF.sub.3    2,4-(CH.sub.3).sub.2                                    CH.sub.3  CF.sub.3    2,5-(CH.sub.3).sub.2                                    CH.sub.3  CF.sub.3    3,4-(CH.sub.3).sub.2                                    CH.sub.3  CF.sub.3    3,5-(CH.sub.3).sub.2                                    CH.sub.3  CF.sub.3    2,4,5-(CH.sub.3).sub.3                                  CH.sub.3  CF.sub.3    2,4,6-(CH.sub.3).sub.3                                  CH.sub.3  CF.sub.3    3-C.sub.2 H.sub.5                                       CH.sub.3  CF.sub.3    4-C.sub.2 H.sub.5                                       CH.sub.3  CF.sub.3    3,4-(C.sub.2 H.sub.5).sub.2                             CH.sub.3  CF.sub.3    3,5-(C.sub.2 H.sub.5).sub.2                             CH.sub.3  CF.sub.3    3-n-C.sub.3 H.sub.7                                     CH.sub.3  CF.sub.3    4-n-C.sub.3 H.sub.7                                     CH.sub.3  CF.sub.3    3-i-C.sub.3 H.sub.7                                     CH.sub.3  CF.sub.3    4-i-C.sub.3 H.sub.7                                     CH.sub.3  CF.sub.3    3-Cyclopropyl                                           CH.sub.3  CF.sub.3    4-Cyclopropyl                                           CH.sub.3  CF.sub.3    3-n-C.sub.4 H.sub.9                                     CH.sub.3  CF.sub.3    4-n-C.sub.4 H.sub.9                                     CH.sub.3  CF.sub.3    3-t-C.sub.4 H.sub.9                                     CH.sub.3  CF.sub.3    4-t-C.sub.4 H.sub.9                                     CH.sub.3  CF.sub.3    3-n-C.sub.6 H.sub.13                                    CH.sub.3  CF.sub.3    4-n-C.sub.6 H.sub.13                                    CH.sub.3  CF.sub.3    3-Cyclohexyl                                            CH.sub.3  CF.sub.3    4-Cyclohexyl                                            CH.sub.3  CF.sub.3    3-Phenyl                                                CH.sub.3  CF.sub.3    4-Phenyl                                                CH.sub.3  CF.sub.3    4-Allyl                                                 CH.sub.3  CF.sub.3    4-Propargyl                                             CH.sub.3  CF.sub.3    2-CH.sub.3, 4-C.sub.2 H.sub.5                           CH.sub.3  CF.sub.3    2-CH.sub.3, 4-i-C.sub.3 H.sub.7                         CH.sub.3  CF.sub.3    2-CH.sub.3, 4-t-C.sub.4 H.sub.9                         CH.sub.3  CF.sub.3    2-CH.sub.3, 4-phenyl                                    CH.sub.3  CF.sub.3    3-CH.sub.3, 4-phenyl                                    CH.sub.3  CF.sub.3    3-OH                                                    CH.sub.3  CF.sub.3    4-OH                                                    CH.sub.3  CF.sub.3    3-OCH.sub.3                                             CH.sub.3  CF.sub.3    4-OCH.sub.3                                             CH.sub.3  CF.sub.3    3,4-(OCH.sub.3).sub.2                                   CH.sub.3  CF.sub.3    3,5-(OCH.sub.3).sub.2                                   CH.sub.3  CF.sub.3    3,4,5-(OCH.sub.3).sub.3                                 CH.sub.3  CF.sub.3    4-OC.sub.2 H.sub.5                                      CH.sub.3  CF.sub.3    4-O-i-C.sub.3 H.sub.7                                   CH.sub.3  CF.sub.3    3-O-t-C.sub.4 H.sub.9                                   CH.sub.3  CF.sub.3    4-O-t-C.sub.4 H.sub.9                                   CH.sub.3  CF.sub.3    4-O-n-C.sub.6 H.sub.13                                  CH.sub.3  CF.sub.3    3-O-Phenyl                                              CH.sub.3  CF.sub.3    4-O-Phenyl                                              CH.sub.3  CF.sub.3    4-O-Allyl                                               CH.sub.3  CF.sub.3    2-CF.sub.3                                              CH.sub.3  CF.sub.3    3-CF.sub.3                                              CH.sub.3  CF.sub.3    4-CF.sub.3                                              CH.sub.3  CF.sub.3    3,5-(CF.sub.3).sub.2                                    CH.sub.3  CF.sub.3    4-CH.sub.2 CF.sub.3                                     CH.sub.3  CF.sub.3    4-C.sub.2 F.sub.5                                       CH.sub.3  CF.sub.3    4-CF.sub.2 CHF.sub.2                                    CH.sub.3  CF.sub.3    3-OCF.sub.3                                             CH.sub.3  CF.sub.3    4-OCF.sub.3                                             CH.sub.3  CF.sub.3    4-OCH.sub.2 CF.sub.3                                    CH.sub.3  CF.sub.3    4-OC.sub.2 F.sub.5                                      CH.sub.3  CF.sub.3    4-OCF.sub.2 CHF.sub.2                                   CH.sub.3  CF.sub.3    3-CH.sub.2 OCH.sub.3                                    CH.sub.3  CF.sub.3    4-CH.sub.2 OCH.sub.3                                    CH.sub.3  CF.sub.3    4-CH.sub.2 --O-t-C.sub.4 H.sub.9                        CH.sub.3  CF.sub.3    4-CH(OCH.sub.3).sub.2                                   CH.sub.3  CF.sub.3    4-CH.sub.2 CN                                           CH.sub.3  CF.sub.3    3-CHO                                                   CH.sub.3  CF.sub.3    4-CHO                                                   CH.sub.3  CF.sub.3    3-CO--CH.sub.3                                          CH.sub.3  CF.sub.3    4-CO--CH.sub.3                                          CH.sub.3  CF.sub.3    3-COOH                                                  CH.sub.3  CF.sub.3    4-COOH                                                  CH.sub.3  CF.sub.3    3-COOCH.sub.3                                           CH.sub.3  CF.sub.3    4-COOCH.sub.3                                           CH.sub.3  CF.sub.3    3-COOC.sub.2 H.sub.5                                    CH.sub.3  CF.sub.3    4-COOC.sub.2 H.sub.5                                    CH.sub.3  CF.sub.3    3-COO-i-C.sub.3 H.sub.7                                 CH.sub.3  CF.sub.3    4-COO-i-C.sub.3 H.sub.7                                 CH.sub.3  CF.sub.3    3-COO-t-C.sub.4 H.sub.9                                 CH.sub.3  CF.sub.3    4-COO-t-C.sub.4 H.sub.9                                 CH.sub.3  CF.sub.3    3-COO-n-C.sub.6 H.sub.13                                CH.sub.3  CF.sub.3    4-COO-n-C.sub.6 H.sub.13                                CH.sub.3  CF.sub.3    3-CONH.sub.2                                            CH.sub.3  CF.sub.3    4-CONH.sub.2                                            CH.sub.3  CF.sub.3    3-CONHCH.sub.3                                          CH.sub.3  CF.sub.3    4-CONHCH.sub.3                                          CH.sub.3  CF.sub.3    3-CON(CH.sub.3).sub.2                                   CH.sub.3  CF.sub.3    4-CON(CH.sub.3).sub.2                                   CH.sub.3  CF.sub.3    3-CSNH.sub.2                                            CH.sub.3  CF.sub.3    4-CSNH.sub.2                                            CH.sub.3  CF.sub.3    3-NH.sub.2                                              CH.sub.3  CF.sub.3    4-NH.sub.2                                              CH.sub.3  CF.sub.3    4-NHCH.sub.3                                            CH.sub.3  CF.sub.3    4-N(CH.sub.3).sub.2                                     CH.sub.3  CF.sub.3    3-NHCO--CH.sub.3                                        CH.sub.3  CF.sub.3    4-NHCO--CH.sub.3                                        CH.sub.3  CF.sub.3    4-NCH.sub.3 --CO--CH.sub.3                              CH.sub.3  CF.sub.3    4-NHCOOCH.sub.3                                         CH.sub.3  CF.sub.3    4-NCH.sub.3 --COOCH.sub.3                               CH.sub.3  CF.sub.3    3-OCO--CH.sub.3                                         CH.sub.3  CF.sub.3    4-OCO--CH.sub.3                                         CH.sub.3  CF.sub.3    4-OCO-t-C.sub.4 H.sub.9                                 CH.sub.3  CF.sub.3    4-SH                                                    CH.sub.3  CF.sub.3    4-SCH.sub.3                                             CH.sub.3  CF.sub.3    4-S-t-C.sub.4 H.sub.9                                   CH.sub.3  CF.sub.3    4-SO--CH.sub.3                                          CH.sub.3  CF.sub.3    4-SO.sub.2 --CH.sub.3                                   CH.sub.3  CF.sub.3    4-C(CH.sub.3)═NCH.sub.3                             CH.sub.3  CF.sub.3    4-C(SCH.sub.3)═NOCH.sub.3                           CH.sub.3  CF.sub.3    4-C(OCH.sub.3)═NOCH.sub.3                           CH.sub.3  CF.sub.3    3-CH═NOCH.sub.3                                     CH.sub.3  CF.sub.3    4-CH═NOCH.sub.3                                     CH.sub.3  CF.sub.3    3-C(CH.sub.3)═NOCH.sub.3                            CH.sub.3  CF.sub.3    4-C(CH.sub.3)═NOCH.sub.3                            CH.sub.3  CF.sub.3    4-C(CH.sub.3)═NOC.sub.2 H.sub.5                     CH.sub.3  CF.sub.3    4-C(CH.sub.3)═NO-n-C.sub.3 H.sub.7                  CH.sub.3  CF.sub.3    4-C(CH.sub.3)═NO-i-C.sub.3 H.sub.7                  CH.sub.3  CF.sub.3    4-C(CH.sub.3)═NO-n-C.sub.4 H.sub.9                  CH.sub.3  CF.sub.3    4-C(CH.sub.3)═NO-t-C.sub.4 H.sub.9                  CH.sub.3  CF.sub.3    4-C(CH.sub.3)═NO-n-C.sub.5 H.sub.11                 CH.sub.3  CF.sub.3    4-C(CH.sub.3)═NO-n-C.sub.6 H.sub.13                 CH.sub.3  CF.sub.3    2-Cl, 4-CH.sub.3                                        CH.sub.3  CF.sub.3    3-Cl, 5-CH.sub.3                                        CH.sub.3  CF.sub.3    2-CH.sub.3, 4-Cl                                        CH.sub.3  CF.sub.3    3-CH.sub.3, 4-Cl                                        CH.sub.3  CF.sub.3    3-F, 5-CH.sub.3                                         CH.sub.3  CF.sub.3    3-Br, 5-CH.sub.3                                        CH.sub.3  CF.sub.3    3-Cl, 5-NO.sub.2                                        CH.sub.3  CF.sub.3    3-NO.sub.2, 4-Cl                                        CH.sub.3  CF.sub.3    3-Cl, 4-OCH.sub.3                                       CH.sub.3  CF.sub.3    3-OCH.sub.3, 4-Cl                                       CH.sub.3  CF.sub.3    3-Cl, 5-CF.sub.3                                        CH.sub.3  CF.sub.3    3-Cl, 5-OCF.sub.3                                       CH.sub.3  CF.sub.3    3-F, 5-CF.sub.3                                         CH.sub.3  CF.sub.3    2-CH.sub.3, 4-CN                                        CH.sub.3  CF.sub.3    2-CH.sub.3, 4-OCH.sub.3                                 CH.sub.3  CF.sub.3    2-CH.sub.3, 4-CF.sub.3                                  CH.sub.3  CF.sub.3    2-CH.sub.3, 4-C(CH.sub.3)═NOCH.sub.3                CH.sub.3  CF.sub.3    3-CH.sub.3, 4-C(CH.sub.3)═NOCH.sub.3                CH.sub.3  CF.sub.3    2-OH, 5-CH.sub.3                                        CH.sub.3  CF.sub.3    3-CH.sub.3, 4-O-t-C.sub.4 H.sub.9                       CH.sub.3  CF.sub.3    2-C(COOCH.sub.3)═NOCH.sub.3                         CH.sub.3  CF.sub.3    2,3-Butadienyl                                          CH.sub.3  CF.sub.3    3,4-Butadienyl                                          ______________________________________                                    

                  TABLE B                                                         ______________________________________                                        A         R       B                                                           ______________________________________                                        CH.sub.3  H       2-Pyridyl                                                   CH.sub.3  H       4-Cl-2-Pyridyl                                              CH.sub.3  H       4-CH.sub.3 -2-Pyridyl                                       CH.sub.3  H       4-CF.sub.3 -2-Pyridyl                                       CH.sub.3  H       4-OCH.sub.3 -2-Pyridyl                                      CH.sub.3  H       5-Cl-2-Pyridyl                                              CH.sub.3  H       5-CH.sub.3 -2-Pyridyl                                       CH.sub.3  H       5-CF.sub.3 -2-Pyridyl                                       CH.sub.3  H       5-OCH.sub.3 -2-Pyridyl                                      CH.sub.3  H       6-Cl-2-Pyridyl                                              CH.sub.3  H       6-CH.sub.3 -2-Pyridyl                                       CH.sub.3  H       6-CF.sub.3 -2-Pyridyl                                       CH.sub.3  H       6-OCH.sub.3 -2-Pyridyl                                      CH.sub.3  H       4,6-Cl.sub.2 -2-Pyridyl                                     CH.sub.3  H       4-CH.sub.3, 6-Cl-2-Pyridyl                                  CH.sub.3  H       4-Cl, 6-CH.sub.3 -2-Pyridyl                                 CH.sub.3  H       5,6-Cl.sub.2 -2-Pyridyl                                     CH.sub.3  H       5,6-(CH.sub.3).sub.2 -2-Pyridyl                             CH.sub.3  H       3-Pyridyl                                                   CH.sub.3  H       2-Cl-3-Pyridyl                                              CH.sub.3  H       4-CH.sub.3 -3-Pyridyl                                       CH.sub.3  H       5-Cl-3-Pyridyl                                              CH.sub.3  H       5-Br-3-Pyridyl                                              CH.sub.3  H       5-CH.sub.3 -3-Pyridyl                                       CH.sub.3  H       5-CF.sub.3 -3-Pyridyl                                       CH.sub.3  H       5-OCH.sub.3 -3-Pyridyl                                      CH.sub.3  H       6-F-3-Pyridyl                                               CH.sub.3  H       6-Cl-3-Pyridyl                                              CH.sub.3  H       6-Br-3-Pyridyl                                              CH.sub.3  H       6-CH.sub.3 -3-Pyridyl                                       CH.sub.3  H       6-t-C.sub.4 H.sub.9 -3-Pyridyl                              CH.sub.3  H       6-CF.sub.3 -3-Pyridyl                                       CH.sub.3  H       6-OCH.sub.3 -3-Pyridyl                                      CH.sub.3  H       4,6-(CH.sub.3).sub.2 -3-Pyridyl                             CH.sub.3  H       5,6-Cl.sub.2 -3-Pyridyl                                     CH.sub.3  H       5-Cl, 6-CH.sub.3 -3-Pyridyl                                 CH.sub.3  H       4-Pyridyl                                                   CH.sub.3  H       2-Cl-4-Pyridyl                                              CH.sub.3  H       2-CH.sub.3 -4-Pyridyl                                       CH.sub.3  H       2-CF.sub.3 -4-Pyridyl                                       CH.sub.3  H       2-OCH.sub.3 -4-Pyridyl                                      CH.sub.3  H       2,6-Cl.sub.2 -4-Pyridyl                                     CH.sub.3  H       2,6-(CH.sub.3).sub.2 -4-Pyridyl                             CH.sub.3  H       2,6-(t-C.sub.4 H.sub.9).sub.2 -4-Pyridyl                    CH.sub.3  H       2-Cl, 6-CH.sub.3 -4-Pyridyl                                 CH.sub.3  H       3-Pyridazinyl                                               CH.sub.3  H       5-CH.sub.3 -3-Pyridazinyl                                   CH.sub.3  H       6-Cl-3-Pyridazinyl                                          CH.sub.3  H       4-Pyridazinyl                                               CH.sub.3  H       6-CF.sub.3 -4-Pyridazinyl                                   CH.sub.3  H       2-Pyrimidinyl                                               CH.sub.3  H       4-Cl-2-Pyrimidinyl                                          CH.sub.3  H       4-CH.sub.3 -2-Pyrimidinyl                                   CH.sub.3  H       4-CF.sub.3 -2-Pyrimidinyl                                   CH.sub.3  H       4-OCH.sub.3 -2-Pyrimidinyl                                  CH.sub.3  H       4,6-(CH.sub.3).sub.2 -2-Pyrimidinyl                         CH.sub.3  H       4-CF.sub.3, 6-OCH.sub.3 -2-Pyrimidinyl                      CH.sub.3  H       5-Cl-2-Pyrimidinyl                                          CH.sub.3  H       5-CH.sub.3 -2-Pyrimidinyl                                   CH.sub.3  H       4-CH.sub.3, 5-Cl-2-Pyrimidinyl                              CH.sub.3  H       4-Pyrimidinyl                                               CH.sub.3  H       2-CH.sub.3 -4-Pyrimidinyl                                   CH.sub.3  H       2-OCH.sub.3 -4-Pyrimidinyl                                  CH.sub.3  H       6-Cl-4-Pyrimidinyl                                          CH.sub.3  H       6-CH.sub.3 -4-Pyrimidinyl                                   CH.sub.3  H       6-CF.sub.3 -4-Pyrimidinyl                                   CH.sub.3  H       6-OCH.sub.3 -4-Pyrimidinyl                                  CH.sub.3  H       2-CH.sub.3, 6-CF.sub.3 -4-Pyrimidinyl                       CH.sub.3  H       2-n-C.sub.3 H.sub.7, 6-CF.sub.3 -4-Pyrimidinyl              CH.sub.3  H       2-OCH.sub.3, 6-CH.sub.3 -4-Pyrimidinyl                      CH.sub.3  H       5-Pyrimidinyl                                               CH.sub.3  H       4-CH.sub.3 -5-Pyrimidinyl                                   CH.sub.3  H       2-CH.sub.3 -5-Pyrimidinyl                                   CH.sub.3  H       2-OCH.sub.3 -5-Pyrimidinyl                                  CH.sub.3  H       2-CH.sub.3, 4-CF.sub.3 -5-Pyrimidinyl                       CH.sub.3  H       2-Pyrazinyl                                                 CH.sub.3  H       5-Cl-2-Pyrazinyl                                            CH.sub.3  H       5-CH.sub.3 -2-Pyrazinyl                                     CH.sub.3  H       6-CF.sub.3 -2-Pyrazinyl                                     CH.sub.3  H       6-OCH.sub.3 -2-Pyrazinyl                                    CH.sub.3  H       5,6-(CH.sub.3).sub.2 -2-Pyrazinyl                           CH.sub.3  H       2-Quinolinyl                                                CH.sub.3  H       5-CH.sub.3 -2-Quinolinyl                                    CH.sub.3  H       6-Cl-2-Quinolinyl                                           CH.sub.3  H       6-CH.sub.3 -2-Quinolinyl                                    CH.sub.3  H       7-CH.sub.3 -2-Quinolinyl                                    CH.sub.3  H       5,7-Cl.sub.2 -2-Quinolinyl                                  CH.sub.3  H       3-Quinolinyl                                                CH.sub.3  H       6-CH.sub.3 -3-Quinolinyl                                    CH.sub.3  H       7-Cl-3-Quinolinyl                                           CH.sub.3  H       8-Cl-3-Quinolinyl                                           CH.sub.3  H       8-OCH.sub.3 -Quinolinyl                                     CH.sub.3  H       4-Quinolinyl                                                CH.sub.3  H       3-Isoquinolinyl                                             CH.sub.3  H       6-CH.sub.3 -3-Isoquinolinyl                                 CH.sub.3  H       7-Cl-3-Isoquinolinyl                                        CH.sub.3  H       8-OCH.sub.3 -3-Isoquinolinyl                                CH.sub.3  H       3-Cinnolinyl                                                CH.sub.3  H       8-CH.sub.3 -3-Cinnolinyl                                    CH.sub.3  H       2-Quinazolinyl                                              CH.sub.3  H       6-CH.sub.3 -2-Quinazolinyl                                  CH.sub.3  H       2-Quinazolinyl                                              CH.sub.3  H       7-Cl-2-Quinoxalinyl                                         CH.sub.3  H       6,8-(CH.sub.3).sub.2 -2-Quinoxalinyl                        CH.sub.3  H       1,5-Naphthyridin-2-yl                                       CH.sub.3  H       2-Pivaloylamino-4-hydroxypteridin-                                            6-yl                                                        CH.sub.3  H       2-Furyl                                                     CH.sub.3  H       4-Cl-2-Furyl                                                CH.sub.3  H       4-CH.sub.3 -2-Furyl                                         CH.sub.3  H       5-Cl-2-Furyl                                                CH.sub.3  H       5-CH.sub.3 -2-Furyl                                         CH.sub.3  H       4,5-Cl.sub.2 -2-Furyl                                       CH.sub.3  H       3-Furyl                                                     CH.sub.3  H       4-CH.sub.3 -3-Furyl                                         CH.sub.3  H       5-Cl-3-Furyl                                                CH.sub.3  H       5-CH.sub.3 -3-Furyl                                         CH.sub.3  H       2-Thienyl                                                   CH.sub.3  H       4-Cl-2-Thienyl                                              CH.sub.3  H       4-CH.sub.3 -2-Thienyl                                       CH.sub.3  H       5-Cl-2-Thienyl                                              CH.sub.3  H       5-Br-2-Thienyl                                              CH.sub.3  H       5-CH.sub.3 -2-Thienyl                                       CH.sub.3  H       5-CF.sub.3 -2-Thienyl                                       CH.sub.3  H       5-OCH.sub.3 -2-Thienyl                                      CH.sub.3  H       5-NO.sub.2 -2-Thienyl                                       CH.sub.3  H       4,5(CH.sub.3).sub.2 -2-Thienyl                              CH.sub.3  H       3-Thienyl                                                   CH.sub.3  H       5-Cl-3-Thienyl                                              CH.sub.3  H       5-CH.sub.3 -3-Thienyl                                       CH.sub.3  H       5-CF.sub.3 -3-Thienyl                                       CH.sub.3  H       1-CH.sub.3 -2-Pyrryl                                        CH.sub.3  H       1-CH.sub.3 -4-OCH.sub.3 -2-Pyrryl                           CH.sub.3  H       1,5-(CH.sub.3).sub.2 -2-Pyrryl                              CH.sub.3  H       1-CH.sub.3 -3-Pyrryl                                        CH.sub.3  H       1-CH.sub.3 -5-Cl-3-Pyrryl                                   CH.sub.3  H       1-C.sub.6 H.sub.5 -3-Pyrryl                                 CH.sub.3  H       1-(4-Cl-C.sub.6 H.sub.4)-3-Pyrryl                           CH.sub.3  H       2-Oxazolyl                                                  CH.sub.3  H       4-CF.sub.3 -2-Oxazolyl                                      CH.sub.3  H       5-Cl-2-Oxazolyl                                             CH.sub.3  H       5-CH.sub.3 -2-oxazolyl                                      CH.sub.3  H       4-Oxazolyl                                                  CH.sub.3  H       2-Cl-4-Oxazolyl                                             CH.sub.3  H       2-CH.sub.3 -4-Oxazolyl                                      CH.sub.3  H       5-Oxazolyl                                                  CH.sub.3  H       2-Cl-5-Oxazolyl                                             CH.sub.3  H       2-CH.sub.3 -5-Oxazolyl                                      CH.sub.3  H       2-Thiazolyl                                                 CH.sub.3  H       4-CH.sub.3 -2-Thiazolyl                                     CH.sub.3  H       5-Cl-2-Thiazolyl                                            CH.sub.3  H       5-OCH.sub.3 -2-Thiazolyl                                    CH.sub.3  H       4-Thiazolyl                                                 CH.sub.3  H       2-CH.sub.3 -4-Thiazolyl                                     CH.sub.3  H       2-Cl-4-Thiazolyl                                            CH.sub.3  H       5-Thiazolyl                                                 CH.sub.3  H       2-Cl-5-Thiazolyl                                            CH.sub.3  H       2-CH.sub.2 -5-Thiazolyl                                     CH.sub.3  H       2,4-(CH.sub.3).sub.2 -5-Thiazolyl                           CH.sub.3  H       1-CH.sub.3 -2-Imidazolyl                                    CH.sub.3  H       1,4-(CH.sub.3).sub.2 -2-Imidazolyl                          CH.sub.3  H       1-CH.sub.3 -4-Imidazolyl                                    CH.sub.3  H       1,2-(CH.sub.3).sub.2 -4-Imidazolyl                          CH.sub.3  H       1-CH.sub.3, 2-OCH.sub.3 -4-Imidazolyl                       CH.sub.3  H       1-CH.sub.3 -5-Imidazolyl                                    CH.sub.3  H       1-CH.sub.3, 2-Cl-5-Imidazolyl                               CH.sub.3  H       1-C.sub.6 H.sub.5 -4-Imidazolyl                             CH.sub.3  H       1-(4-F-C.sub.6 H.sub.4)-4-Imidazolyl                        CH.sub.3  H       3-Isoxazolyl                                                CH.sub.3  H       5-Cl-3-Isoxazolyl                                           CH.sub.3  H       5-CH.sub.3 -3-Isoxazolyl                                    CH.sub.3  H       5-Isoxazolyl                                                CH.sub.3  H       3-CH.sub.3 -5-Isoxazolyl                                    CH.sub.3  H       3-CF.sub.3 -5-Isoxazolyl                                    CH.sub.3  H       3-Isothiazolyl                                              CH.sub.3  H       5-CH.sub.3 -3-Isothiazolyl                                  CH.sub.3  H       5-Isothiazolyl                                              CH.sub.3  H       3-Cl-5-Isothiazolyl                                         CH.sub.3  H       1-CH.sub.3 -3-Pyrazolyl                                     CH.sub.3  H       1-CH.sub.3, 5-Cl-Pyrazolyl                                  CH.sub.3  H       1-CH.sub.3 -4-Pyrazolyl                                     CH.sub.3  H       1-CH.sub.3 -5-Pyrazolyl                                     CH.sub.3  H       1,3-(CH.sub.3).sub.2 -5-Pyrazolyl                           CH.sub.3  H       1-C.sub.6 H.sub.5 -3-Pyrazolyl                              CH.sub.3  H       1-(4-CH.sub.3 C.sub.6 H.sub.4)-3-pyrazolyl                  CH.sub.3  H       1-C.sub.6 H.sub.5 -4-Pyrazolyl                              CH.sub.3  H       1-(4-ClC.sub.6 H.sub.4)-4-Pyrazolyl                         CH.sub.3  H       1,2,4-oxadiazol-3-yl                                        CH.sub.3  H       5-CH.sub.3 -1,2,4-Oxadiazol-3-yl                            CH.sub.3  H       1,2,4-Oxadiazol-5-yl                                        CH.sub.3  H       3-CH.sub.3 -1,2,4-Oxadiazol-5-yl-                           CH.sub.3  H       1,3,4-Oxadiazolyl                                           CH.sub.3  H       5-CH.sub.3 -1,3,4-Oxadiazol-2-yl                            CH.sub.3  H       1,2,4-Thiadiazol-3-yl                                       CH.sub.3  H       1,2,4-Thiadiazol-5-yl                                       CH.sub.3  H       1,3,4-Thiadiazolyl                                          CH.sub.3  H       5-i-C.sub.3 H.sub.7 -1,3,4-Thiadiazol-2-yl                  CH.sub.3  H       1-CH.sub.3 -1,2,4-Triazol-3-yl                              CH.sub.3  H       1-CH.sub.3 -5-CF.sub.3 -1,2,4-Triazol-3-yl                  CH.sub.3  H       1-CH.sub.3 -1,2,4-Triazol-5-yl                              CH.sub.3  H       1-C.sub.6 H.sub.5 -1,2,4-Triazol-3-yl                       CH.sub.3  H       1-CH.sub.3 -Tetrazol-5-yl                                   CH.sub.3  H       1-C.sub.6 H.sub.5 -Tetrazol-5-yl                            CH.sub.3  H       1,2,4-Triazin-3-yl                                          CH.sub.3  H       1,3,5-Triazin-2-yl                                          CH.sub.3  H       4,6-(CH.sub.3).sub.2 -1,3,5-Triazin-2-yl                    CH.sub.3  H       4,6-(CF.sub.3).sub.2 -1,3,5-Triazin-2-yl                    CH.sub.3  H       4,6-(OCH.sub.3).sub.2 -1,3,5-Triazin-2-yl                   CH.sub.3  H       1,2,4,5-Tetrazin-3-yl                                       CH.sub.3  H       6-CH.sub.3 -1,2,4,5-Tetrazin-3-yl                           CH.sub.3  H       2-Benzofuryl                                                CH.sub.3  H       6-Cl-2-Benzofuryl                                           CH.sub.3  H       6-CH.sub.3 -2-Benzofuryl                                    CH.sub.3  H       7-CH.sub.3 -2-Benzyofuryl                                   CH.sub.3  H       2-Thionaphthenyl                                            CH.sub.3  H       6-Cl-2-Thionaphthenyl                                       CH.sub.3  H       6-CH.sub.3 -2-Thionaphthenyl                                CH.sub.3  H       7-Br-2-Thionaphthenyl                                       CH.sub.3  H       1-CH.sub.3 -2-Indolyl                                       CH.sub.3  H       1,7-(CH.sub.3).sub.2 -2-Indolyl                             CH.sub.3  H       1-CH.sub.3 -3-Indolyl                                       CH.sub.3  H       2-Benzoxazolyl                                              CH.sub.3  H       6-CH.sub.3 -2-Benzoxazolyl                                  CH.sub.3  H       6-Br-2-Benzoxazolyl                                         CH.sub.3  H       7-Cl-2-Benzoxazolyl                                         CH.sub.3  H       2-Benzothiazolyl                                            CH.sub.3  H       6-CF.sub.3 -2-Benzothiazolyl                                CH.sub.3  H       6-CH.sub.3 -2-Benzothiazolyl                                CH.sub.3  H       7-Br-2-Benzothiazolyl                                       CH.sub.3  H       1-CH.sub.3 -2-Benzimidazolyl                                CH.sub.3  H       1-CH.sub.3 -6-Cl-2-Benzimidazolyl                           CH.sub.3  H       1-CH.sub.3 -7-CH.sub.3 -2-Benzimidazolyl                    CH.sub.3  H       3-[1,2]-Benzisoxazolyl                                      CH.sub.3  H       3-[1,2]-Benzisothiazolyl                                    CH.sub.3  H       1-CH.sub.3 -3-Benzpyrazolyl                                 CH.sub.3  H       2-Purinyl                                                   CH.sub.3  H       6-CH.sub.3 -2-Purinyl                                       CH.sub.3  H       6-Purinyl                                                   CH.sub.3  H       2-CH.sub.3 -6-Purinyl                                       CH.sub.3  H       2,4-(CH.sub.3).sub.2 -6-Purinyl                             CH.sub.3  CH.sub.3                                                                              2-Pyridyl                                                   CH.sub.3  CH.sub.3                                                                              4-CH.sub.3 -2-Pyridyl                                       CH.sub.3  CH.sub.3                                                                              5-CF.sub.3 -2-Pyridyl                                       CH.sub.3  CH.sub.3                                                                              6-Cl-2-Pyridyl                                              CH.sub.3  CH.sub.3                                                                              6-OCH.sub.3 -2-Pyridyl                                      CH.sub.3  CH.sub.3                                                                              5,6-Cl-2-Pyridyl                                            CH.sub.3  CH.sub.3                                                                              3-Pyridyl                                                   CH.sub.3  CH.sub.3                                                                              5-Br-3-Pyridyl                                              CH.sub.3  CH.sub.3                                                                              6-F-3-Pyridyl                                               CH.sub.3  CH.sub.3                                                                              6-t-C.sub.4 H.sub.9 -3-Pyridyl                              CH.sub.3  CH.sub.3                                                                              6-OCH.sub.3 -3-Pyridyl                                      CH.sub.3  CH.sub.3                                                                              6-CF.sub.3 -3-Pyridyl                                       CH.sub.3  CH.sub.3                                                                              4-Pyridyl                                                   CH.sub.3  CH.sub.3                                                                              2-CH.sub.3 -4-Pyridyl                                       CH.sub.3  CH.sub.3                                                                              2-Cl, 6-CH.sub.3 -4-Pyridyl                                 CH.sub.3  CH.sub.3                                                                              3-Pyridazinyl                                               CH.sub.3  CH.sub.3                                                                              6-Cl-3-Pyridazinyl                                          CH.sub.3  CH.sub.3                                                                              4-Pyridazinyl                                               CH.sub.3  CH.sub.3                                                                              2-Pyrimidinyl                                               CH.sub.3  CH.sub.3                                                                              4-CH.sub.3 -2-Pyrimidinyl                                   CH.sub.3  CH.sub.3                                                                              4-CF.sub.3, 6-OCH.sub.3 -2-Pyrimidinyl                      CH.sub.3  CH.sub.3                                                                              5-Cl-2-Pyrimidinyl                                          CH.sub.3  CH.sub.3                                                                              4-Pyrimidinyl                                               CH.sub.3  CH.sub.3                                                                              2-OCH.sub.3 -4-Pyrimidinyl                                  CH.sub.3  CH.sub.3                                                                              6-Cl-4-Pyrimidinyl                                          CH.sub.3  CH.sub.3                                                                              2-n-C.sub.3 H.sub.7 -6-CF.sub.3 -4-Pyrimidinyl              CH.sub.3  CH.sub.3                                                                              5-Pyrimidinyl                                               CH.sub.3  CH.sub.3                                                                              2-CH.sub.3 -5-Pyrimidinyl                                   CH.sub.3  CH.sub.3                                                                              2-Pyrazinyl                                                 CH.sub.3  CH.sub.3                                                                              5-CH.sub.3 -2-Pyrazinyl                                     CH.sub.3  CH.sub.3                                                                              6-OCH.sub.3 -2-Pyrazinyl                                    CH.sub.3  CH.sub.3                                                                              2-Quinolinyl                                                CH.sub.3  CH.sub.3                                                                              6-CH.sub.3 -2-Quinolinyl                                    CH.sub.3  CH.sub.3                                                                              5,7-Cl.sub.2 -2-Quinolinyl                                  CH.sub.3  CH.sub.3                                                                              3-Quinolinyl                                                CH.sub.3  CH.sub.3                                                                              8-OCH.sub.3 -3-Quinolinyl                                   CH.sub.3  CH.sub.3                                                                              4-Quinolinyl                                                CH.sub.3  CH.sub.3                                                                              3-Isoquinolinyl                                             CH.sub.3  CH.sub.3                                                                              7-Cl-3-Isoquinolinyl                                        CH.sub.3  CH.sub.3                                                                              3-Cinnolinyl                                                CH.sub.3  CH.sub.3                                                                              8-CH.sub.3 -3-Cinnolinyl                                    CH.sub.3  CH.sub.3                                                                              2-Quinazolinyl                                              CH.sub.3  CH.sub.3                                                                              2-Quinoxalinyl                                              CH.sub.3  CH.sub.3                                                                              1,5-Napthyridin-2-yl                                        CH.sub.3  CH.sub.3                                                                              2-Furyl                                                     CH.sub.3  CH.sub.3                                                                              4-CH.sub.3 -3-Furyl                                         CH.sub.3  CH.sub.3                                                                              5-Cl-2-Furyl                                                CH.sub.3  CH.sub.3                                                                              3-Furyl                                                     CH.sub.3  CH.sub.3                                                                              5-CH.sub.3 -3-Furyl                                         CH.sub.3  CH.sub.3                                                                              2-Thienyl                                                   CH.sub.3  CH.sub.3                                                                              4-CH.sub.3 -2-Thienyl                                       CH.sub.3  CH.sub.3                                                                              5-Br-2-Thienyl                                              CH.sub.3  CH.sub.3                                                                              5-CF.sub.3 -2-Thienyl                                       CH.sub.3  CH.sub.3                                                                              5-NO.sub.2 -2-Thienyl                                       CH.sub.3  CH.sub.3                                                                              4,5-(CH.sub.3).sub.2 -2-Thienyl                             CH.sub.3  CH.sub.3                                                                              3-Thienyl                                                   CH.sub.3  CH.sub.3                                                                              5-CH.sub.3 -3-Thienyl                                       CH.sub.3  CH.sub.3                                                                              1-CH.sub.3 -2-Pyrryl                                        CH.sub.3  CH.sub.3                                                                              1-CH.sub.3 -3-Pyrryl                                        CH.sub.3  CH.sub.3                                                                              1-(4-Cl-C.sub.6 H.sub.4)-3-Pyrryl                           CH.sub.3  CH.sub.3                                                                              2-Oxazolyl                                                  CH.sub.3  CH.sub.3                                                                              5-CH.sub.3 -2-oxazolyl                                      CH.sub.3  CH.sub.3                                                                              4-Oxazolyl                                                  CH.sub.3  CH.sub.3                                                                              2-Cl-4-Oxazolyl                                             CH.sub.3  CH.sub.3                                                                              5-Oxazolyl                                                  CH.sub.3  CH.sub.3                                                                              2-CH.sub.3 -5-Oxazolyl                                      CH.sub.3  CH.sub.3                                                                              2-Thiazolyl                                                 CH.sub.3  CH.sub.3                                                                              4-CH.sub.3 -2-Thiazolyl                                     CH.sub.3  CH.sub.3                                                                              5-OCH.sub.3 -2-Thiazolyl                                    CH.sub.3  CH.sub.3                                                                              4-Thiazolyl                                                 CH.sub.3  CH.sub.3                                                                              2-Cl-4-Thiazolyl                                            CH.sub.3  CH.sub.3                                                                              5-Thiazolyl                                                 CH.sub.3  CH.sub.3                                                                              2,4-(CH.sub.3).sub.2 -5-Thiazolyl                           CH.sub.3  CH.sub.3                                                                              1-CH.sub.3 -2-Imidazolyl                                    CH.sub.3  CH.sub.3                                                                              1-CH.sub.3 -4-Imidazolyl                                    CH.sub.3  CH.sub.3                                                                              1-CH.sub.3 -5-Imidazolyl                                    CH.sub.3  CH.sub.3                                                                              1-C.sub.6 H.sub.5 -5-Imidazolyl                             CH.sub.3  CH.sub.3                                                                              3-Isoxazolyl                                                CH.sub.3  CH.sub.3                                                                              5-CH.sub.3 -3-Isoxazolyl                                    CH.sub.3  CH.sub.3                                                                              5-Isoxazolyl                                                CH.sub.3  CH.sub.3                                                                              3-Isothiazolyl                                              CH.sub.3  CH.sub.3                                                                              5-Isothiazolyl                                              CH.sub.3  CH.sub.3                                                                              1-CH.sub.3 -3-Pyrazolyl                                     CH.sub.3  CH.sub.3                                                                              1-CH.sub.3 -4-Pyrazolyl                                     CH.sub.3  CH.sub.3                                                                              1-CH.sub.3 -5-Pyrazolyl                                     CH.sub.3  CH.sub.3                                                                              1,3-(CH.sub.3).sub.2 -5-Pyrazolyl                           CH.sub.3  CH.sub.3                                                                              1-(4-CH.sub.3 -C.sub.6 H.sub.4)-4-Pyrazolyl                 CH.sub.3  CH.sub.3                                                                              1,2,4-Oxadiazol-3-yl                                        CH.sub.3  CH.sub.3                                                                              1,2,4-Oxadiazol-5-yl                                        CH.sub.3  CH.sub.3                                                                              1,3,4-Oxadiazolyl                                           CH.sub.3  CH.sub.3                                                                              5-CH.sub.3 -1,3,4-Oxadiazol-2-yl                            CH.sub.3  CH.sub.3                                                                              1,2,4-Thiadiazol-3-yl                                       CH.sub.3  CH.sub.3                                                                              1,2,4-Thiadiazol-5-yl                                       CH.sub.3  CH.sub.3                                                                              1,3,4-Thiadiazolyl                                          CH.sub.3  CH.sub.3                                                                              5-OC.sub.3 H.sub.7 -1,3,4-Thiadiazolyl                      CH.sub.3  CH.sub.3                                                                              1-CH.sub.3 -1,2,4-Triazol-3-yl                              CH.sub.3  CH.sub.3                                                                              1-CH.sub.3 -5-CF.sub.3 -1,2,4-Triazol-3-yl                  CH.sub.3  CH.sub.3                                                                              l-C.sub.6 H.sub.5 -1,2,4-Triazol-S-yl                       CH.sub.3  CH.sub.3                                                                              I-CH.sub.3 -Tetrazol-5-yl                                   CH.sub.3  CH.sub.3                                                                              1,2,4-Triazin-3-yl                                          CH.sub.3  CH.sub.3                                                                              1,3,5-Triazin-2-yl                                          CH.sub.3  CH.sub.3                                                                              4,6-(OCH.sub.3)-1,3,5-Triazin-2-yl                          CH.sub.3  CH.sub.3                                                                              1,2,4,5-Tetrazin-3-yl                                       CH.sub.3  CH.sub.3                                                                              2-Benzofuryl                                                CH.sub.3  CH.sub.3                                                                              6-CH.sub.3 -2-Benzofuryl                                    CH.sub.3  CH.sub.3                                                                              2-Thionaphthenyl                                            CH.sub.3  CH.sub.3                                                                              7-Br-2-Thionaphthenyl                                       CH.sub.3  CH.sub.3                                                                              1-CH.sub.3 -2-Indolyl                                       CH.sub.3  CH.sub.3                                                                              2-Benzoxazolyl                                              CH.sub.3  CH.sub.3                                                                              6-Br-2-Benzoxazolyl                                         CH.sub.3  CH.sub.3                                                                              2-Benzothiazolyl                                            CH.sub.3  CH.sub.3                                                                              6-CF.sub.3 -2-Benzothiazolyl                                CH.sub.3  CH.sub.3                                                                              1-CH.sub.3 -2-Benzimidazolyl                                CH.sub.3  CH.sub.3                                                                              3-[1,2]-Benzisoxazolyl                                      CH.sub.3  CH.sub.3                                                                              2-Purinyl                                                   CH.sub.3  CH.sub.3                                                                              6-Purinyl                                                   H         H       2-Pyridyl                                                   H         H       5-CF.sub.3 -2-Pyridyl                                       H         H       3-Pyridyl                                                   H         H       6-t-C.sub.4 H.sub.9 -3-Pyridyl                              H         H       4-Pyridyl                                                   H         H       2-CH.sub.3 -4-Pyridyl                                       H         H       3-Pyridazinyl                                               H         H       2-Pyrimidinyl                                               H         H       4-CF.sub.3, 6-OCH.sub.3 -2-Pyrimidinyl                      H         H       4-Pyrimidinyl                                               H         H       6-Cl-4-Pyrimidinyl                                          H         H       2-n-C.sub.3 H.sub.7 -6-CF.sub.3 -4-Primidinyl               H         H       5-Pyrimidinyl                                               H         H       2-Pyrazinyl                                                 H         H       2-Quinolinyl                                                H         H       3-Quinolinyl                                                H         H       3-Isoquinolinyl                                             H         H       2-Quinoxalinyl                                              H         H       2-Furyl                                                     H         H       5-Cl-2-Furyl                                                H         H       3-Furyl                                                     H         H       2-Thienyl                                                   H         H       5-NO.sub.2 -2-Thienyl                                       H         H       3-Thienyl                                                   H         H       1-(4-ClC.sub.6 H.sub.4)-3-Pyrryl                            H         H       2-Oxazolyl                                                  H         H       4-Oxazolyl                                                  H         H       5-Oxazolyl                                                  H         H       2-Thiazolyl                                                 H         H       4-Thiazolyl                                                 H         H       5-Thiazolyl                                                 H         H       2,4-(CH.sub.3).sub.2 -5-Thiazolyl                           H         H       1-CH.sub.3 -4-Imidazolyl                                    H         H       3-Isoxazolyl                                                H         H       5-CH.sub.3 -3-Isoxazolyl                                    H         H       5-Isoxazolyl                                                H         H       3-Isothiazolyl                                              H         H       1-CH.sub.3 -3-pyrazolyl                                     H         H       1-(4-CH.sub.3C.sub.6 H.sub.4)-4-Pyrazolyl                   H         H       1,2,4-oxadiazol-3-yl                                        H         H       1,3,4-Thiadiazolyl                                          H         H       1-C.sub.6 H.sub.5 -1,2,4-Triazol-5-yl                       H         H       1,3,5-Triazin-2-yl                                          H         H       4,6-(OCH.sub.3).sub.2 -1,3,5-Triazin-2-yl                   H         H       2-Benzofuryl                                                H         H       2-Thionaphthenyl                                            H         H       7-Br-2-Thionaphthenyl                                       H         H       1-CH.sub.3 -2-Indolyl                                       H         H       2-Benzoxazolyl                                              H         H       6-Br-2-Benzoxazolyl                                         H         H       2-Benzothiazolyl                                            H         H       6-CF.sub.3 -2-Benzothiazolyl                                H         H       1-CH.sub.3 -2-Benzimidazolyl                                H         H       6-Purinyl                                                   H         CH.sub.3                                                                              2-Pyridyl                                                   H         CH.sub.3                                                                              5-CF.sub.3 -2-Pyridyl                                       H         CH.sub.3                                                                              3-Pyridyl                                                   H         CH.sub.3                                                                              6-t-C.sub.4 H.sub.9 -3-Pyridyl                              H         CH.sub.3                                                                              4-Pyridyl                                                   H         CH.sub.3                                                                              2-CH.sub.3 -4-Pyridyl                                       H         CH.sub.3                                                                              3-Pyridazinyl                                               H         CH.sub.3                                                                              2-Pyrimidinyl                                               H         CH.sub.3                                                                              4-CF.sub.3, 6-OCH.sub.3 -2-Pyrimidinyl                      H         CH.sub.3                                                                              4-Pyrimidinyl                                               H         CH.sub.3                                                                              6-Cl-4-Pyrimidinyl                                          H         CH.sub.3                                                                              2-n-C.sub.3 H.sub.7 -6-CF.sub.3 -4-Pyrimidinyl              H         CH.sub.3                                                                              5-Pyrimidinyl                                               H         CH.sub.3                                                                              2-Pyrazinyl                                                 H         CH.sub.3                                                                              2-Quinolinyl                                                H         CH.sub.3                                                                              3-Quinolinyl                                                H         CH.sub.3                                                                              3-Isoquinolinyl                                             H         CH.sub.3                                                                              2-Quinoxalinyl                                              H         CH.sub.3                                                                              2-Furyl                                                     H         CH.sub.3                                                                              5-Cl-2-Furyl                                                H         CH.sub.3                                                                              3-Puryl                                                     H         CH.sub.3                                                                              2-Thienyl                                                   H         CH.sub.3                                                                              5-NO.sub.2 -2-Thienyl                                       H         CH.sub.3                                                                              3-Thienyl                                                   H         CH.sub.3                                                                              1-(4-ClC.sub.6 H.sub.4)-3-Pyrryl                            H         CH.sub.3                                                                              2-Oxazolyl                                                  H         CH.sub.3                                                                              4-Oxagolyl                                                  H         CH.sub.3                                                                              5-Oxazolyl                                                  H         CH.sub.3                                                                              2-Thiazolyl                                                 H         CH.sub.3                                                                              4-Thiazolyl                                                 H         CH.sub.3                                                                              5-Thiazolyl                                                 H         CH.sub.3                                                                              2,4-(CH.sub.3).sub.2 -5-Thiazolyl                           H         CH.sub.3                                                                              1-CH.sub.3 -4-Imidazolyl                                    H         CH.sub.3                                                                              3-Isoxazolyl                                                H         CH.sub.3                                                                              5-CH.sub.3 -3-Isoxazolyl                                    H         CH.sub.3                                                                              5-Isoxazolyl                                                H         CH.sub.3                                                                              3-Isothiazolyl                                              H         CH.sub.3                                                                              1-CH.sub.3 -3-Pyrazolyl                                     H         CH.sub.3                                                                              1-(4-CH.sub.3C.sub.6 H.sub.4)-4-Pyrazolyl                   H         CH.sub.3                                                                              1,2,4-oxadiazol-3-yl                                        H         CH.sub.3                                                                              1,3,4-Thiadiazolyl                                          H         CH.sub.3                                                                              1-C.sub.6 H.sub.5 -1,2,4-Triazol-5-yl                       H         CH.sub.3                                                                              1,3,5-Triazin-2-yl                                          H         CH.sub.3                                                                              4,6-(OCH.sub.3).sub.2 -1,3,5-Triazin-2-yl                   H         CH.sub.3                                                                              2-Benzofuryl                                                H         CH.sub.3                                                                              2-Thionaphthenyl                                            H         CH.sub.3                                                                              7-Br-2-Thionaphthenyl                                       H         CH.sub.3                                                                              1-CH.sub.3 -2-Indolyl                                       H         CH.sub.3                                                                              2-Benzoxazolyl                                              H         CH.sub.3                                                                              6-Br-2-Benzoxazolyl                                         H         CH.sub.3                                                                              2-Benzothiazolyl                                            H         CH.sub.3                                                                              6-CF.sub.3 -2-Benzothiazolyl                                H         CH.sub.3                                                                              1-CH.sub.3 -2-Benzimidazolyl                                H         CH.sub.3                                                                              6-Purinyl                                                   Cyclopropyl                                                                             H       2-Pyridyl                                                   Cyclopropyl                                                                             H       5-CF.sub.3 -2-Pyridyl                                       Cyclopropyl                                                                             H       3-Pyridyl                                                   Cyclopropyl                                                                             H       6-t-C.sub.4 H.sub.9 -3-Pyridyl                              Cyclopropyl                                                                             H       4-Pyridyl                                                   Cyclopropyl                                                                             H       2-CH.sub.3 -4-Pyridyl                                       Cyclopropyl                                                                             H       3-pyridazinyl                                               Cyclopropyl                                                                             H       2-Pyrimidinyl                                               Cyclopropyl                                                                             H       4-CF.sub.3, 6-OCH.sub.3 -2-Pyrimidinyl                      Cyclopropyl                                                                             H       4-Pyrimidinyl                                               Cyclopropyl                                                                             H       6-Cl-4-Pyrimidinyl                                          Cyclopropyl                                                                             H       2-n-C.sub.3 H.sub.7 -6-CF.sub.3 -4-Pyrimidinyl              Cyclopropyl                                                                             H       5-Pyrimidinyl                                               Cyclopropyl                                                                             H       2-Pyrazinyl                                                 Cyclopropyl                                                                             H       2-Quinolinyl                                                Cyclopropyl                                                                             H       3-Quinolinyl                                                Cyclopropyl                                                                             H       3-Isoquinolinyl                                             Cyclopropyl                                                                             H       2-Quinoxalinyl                                              Cyclopropyl                                                                             H       2-Furyl                                                     Cyclopropyl                                                                             H       5-Cl-2-Furyl                                                Cyclopropyl                                                                             H       3-Furyl                                                     Cyclopropyl                                                                             H       2-Thienyl                                                   Cyclopropyl                                                                             H       5-NO.sub.2 -2-Thienyl                                       Cyclopropyl                                                                             H       3-Thienyl                                                   Cyclopropyl                                                                             H       1-(4-ClC.sub.6 H.sub.4)-3-Pyrryl                            Cyclopropyl                                                                             H       2-Oxazolyl                                                  Cyclopropyl                                                                             H       4-Oxazolyl                                                  Cyclopropyl                                                                             H       5-Oxazolyl                                                  Cyclopropyl                                                                             H       2-Thiazolyl                                                 cyclopropyl                                                                             H       4-Thiazolyl                                                 Cyclopropyl                                                                             H       5-Thiazolyl                                                 Cyclopropyl                                                                             H       2,4-(CH.sub.3).sub.2 -5-Thiazolyl                           Cyclopropyl                                                                             H       1-CH.sub.3 -4-Imidazolyl                                    Cyclopropyl                                                                             H       3-Isoxazolyl                                                Cyclopropyl                                                                             H       5-CH.sub.3 -3-Isoxazolyl                                    Cyclopropyl                                                                             H       5-Isoxazolyl                                                Cyclopropyl                                                                             H       3-Isothiazolyl                                              Cyclopropyl                                                                             H       1-CH.sub.3 -3-pyrazolyl                                     Cyclopropyl                                                                             H       1-(4-CH.sub.3C.sub.6 H.sub.4)-4-Pyrazolyl                   Cyclopropyl                                                                             H       1,2,4-Oxadiazol-3-yl                                        Cyclopropyl                                                                             H       1,3,4-Thiadiazolyl                                          Cyclopropyl                                                                             H       1-C.sub.6 H.sub.5 -1,2,4-Triazol-5-yl                       Cyclopropyl                                                                             H       1,3,5-Triazin-2-yl                                          Cyclopropyl                                                                             H       4,6-(OCH.sub.3).sub.2 -1,3,5-Triazin-2-yl                   Cyclopropyl                                                                             H       2-Benzofuryl                                                Cyclopropyl                                                                             H       2-Thionaphthenyl                                            Cyclopropyl                                                                             H       7-Br-2-Thionaphthenyl                                       Cyclopropyl                                                                             H       1-CH.sub.3 -2-Indolyl                                       Cyclopropyl                                                                             H       2-Benzoxazolyl                                              Cyclopropyl                                                                             H       6-Br-2-Benzoxazolyl                                         Cyclopropyl                                                                             H       2-Benzothiazolyl                                            Cyclopropyl                                                                             H       6-CF.sub.3 -2-Benzothiazolyl                                Cyclopropyl                                                                             H       1-CH.sub.3 -2-Benzimidazolyl                                Cyclopropyl                                                                             H       6-Purinyl                                                   Cyclopropyl                                                                             CH.sub.3                                                                              2-Pyridyl                                                   Cyclopropyl                                                                             CH.sub.3                                                                              5-CF.sub.3 -2-Pyridyl                                       Cyclopropyl                                                                             CH.sub.3                                                                              3-Pyridyl                                                   Cyclopropyl                                                                             CH.sub.3                                                                              6-t-C.sub.4 H.sub.9 -3-Pyridyl                              Cyclopropyl                                                                             CH.sub.3                                                                              4-Pyridyl                                                   Cyclopropyl                                                                             CH.sub.3                                                                              2-CH.sub.3 -4-Pyridyl                                       Cyclopropyl                                                                             CH.sub.3                                                                              3-Pyridazinyl                                               Cyclopropyl                                                                             CH.sub.3                                                                              2-Pyrimidinyl                                               Cyclopropyl                                                                             CH.sub.3                                                                              4-CF.sub.3, 6-OCH.sub.3 -2-Pyrimidinyl                      Cyclopropyl                                                                             CH.sub.3                                                                              4-Pyrimidinyl                                               Cyclopropyl                                                                             CH.sub.3                                                                              6-Cl-4-Pyrimidinyl                                          Cyclopropyl                                                                             CH.sub.3                                                                              2-n-C.sub.3 H.sub.7 -6-CF.sub.3 -4-Pyrimidinyl              Cyclopropyl                                                                             CH.sub.3                                                                              5-Pyrimidinyl                                               Cyclopropyl                                                                             CH.sub.3                                                                              2-Pyrazinyl                                                 Cyclopropyl                                                                             CH.sub.3                                                                              2-Quinolinyl                                                Cyclopropyl                                                                             CH.sub.3                                                                              3-Quinolinyl                                                Cyclopropyl                                                                             CH.sub.3                                                                              3-Isoquinolinyl                                             Cyclopropyl                                                                             CH.sub.3                                                                              2-Quinoxalinyl                                              Cyclopropyl                                                                             CH.sub.3                                                                              2-Furyl                                                     Cyclopropyl                                                                             CH.sub.3                                                                              5-Cl-2-Furyl                                                Cyclopropyl                                                                             CH.sub.3                                                                              3-Furyl                                                     Cyclopropyl                                                                             CH.sub.3                                                                              2-Thienyl                                                   Cyclopropyl                                                                             CH.sub.3                                                                              5-NO.sub.2 -2-Thienyl                                       Cyclopropyl                                                                             CH.sub.3                                                                              3-Thienyl                                                   Cyclopropyl                                                                             CH.sub.3                                                                              1-(4-ClC.sub.6 H.sub.4)-3-Pyrryl                            Cyclopropyl                                                                             CH.sub.3                                                                              2-oxazolyl                                                  Cyclopropyl                                                                             CH.sub.3                                                                              4-Oxazolyl                                                  Cyclopropyl                                                                             CH.sub.3                                                                              5-Oxazolyl                                                  Cyclopropyl                                                                             CH.sub.3                                                                              2-Thiazolyl                                                 Cyclopropyl                                                                             CH.sub.3                                                                              4-Thiazolyl                                                 Cyclopropyl                                                                             CH.sub.3                                                                              5-Thiazolyl                                                 Cyclopropyl                                                                             CH.sub.3                                                                              2,4-(CH.sub.3).sub.2 -5-Thiazolyl                           Cyclopropyl                                                                             CH.sub.3                                                                              1-CH.sub.3 -4-Imidazolyl                                    Cyclopropyl                                                                             CH.sub.3                                                                              3-Isoxazolyl                                                Cyclopropyl                                                                             CH.sub.3                                                                              5-CH.sub.3 -3-Isoxazolyl                                    Cyclopropyl                                                                             CH.sub.3                                                                              5-Isoxazolyl                                                Cyclopropyl                                                                             CH.sub.3                                                                              3-Isothiazolyl                                              Cyclopropyl                                                                             CH.sub.3                                                                              1-CH.sub.3 -3-Pyrazolyl                                     Cyclopropyl                                                                             CH.sub.3                                                                              1-(4-CH.sub.3C.sub.6 H.sub.4)-4-Pyrazolyl                   Cyclopropyl                                                                             CH.sub.3                                                                              1,2,4-Oxadiazol-3-yl                                        Cyclopropyl                                                                             CH.sub.3                                                                              1,3,4-Thiadiazolyl                                          Cyclopropyl                                                                             CH.sub.3                                                                              1-C.sub.6 H.sub.5 -1,2,4-Triazol-5-yl                       Cyclopropyl                                                                             CH.sub.3                                                                              1,3,5-Triazin-2-yl                                          Cyclopropyl                                                                             CH.sub.3                                                                              4,6-(OCH.sub.3).sub.2 -1,3,5-Triazin-2-yl                   Cyclopropyl                                                                             CH.sub.3                                                                              2-Benzofuryl                                                Cyclopropyl                                                                             CH.sub.3                                                                              2-Thionaphthenyl                                            Cyclopropyl                                                                             CH.sub.3                                                                              7-Br-2-Thionaphthenyl                                       Cyclopropyl                                                                             CH.sub.3                                                                              1-CH.sub.3 -2-Indolyl                                       Cyclopropyl                                                                             CH.sub.3                                                                              2-Benzoxazolyl                                              Cyclopropyl                                                                             CH.sub.3                                                                              6-Br-2-Benzoxazolyl                                         Cyclopropyl                                                                             CH.sub.3                                                                              2-Benzothiazolyl                                            Cyclopropyl                                                                             CH.sub.3                                                                              6-CF.sub.3 -2-Benzothiazolyl                                Cyclopropyl                                                                             CH.sub.3                                                                              1-CH.sub.3 -2-Benzothiadazolyl                              Cyclopropyl                                                                             CH.sub.3                                                                              6-Purinyl                                                   ______________________________________                                        A            B                R                                               ______________________________________                                        CH.sub.3     CH.sub.3         H                                               CH.sub.3     C.sub.2 H.sub.5  H                                               CH.sub.3     n-C.sub.3 H.sub.7                                                                              H                                               CH.sub.3     i-C.sub.3 H.sub.7                                                                              H                                               CH.sub.3     s-C.sub.4 H.sub.9                                                                              H                                               CH.sub.3     t-C.sub.4 H.sub.9                                                                              H                                               CH.sub.3     n-C.sub.5 H.sub.11                                                                             H                                               CH.sub.3     n-C.sub.6 H.sub.13                                                                             H                                               CH.sub.3     n-C.sub.12 H.sub.25                                                                            H                                               CH.sub.3     Cyclopropyl      H                                               CH.sub.3     Cyclobutyl       H                                               CH.sub.3     Cyclopentyl      H                                               CH.sub.3     Cyclohexyl       H                                               CH.sub.3     Cycloheptyl      H                                               CH.sub.3     CHO              H                                               CH.sub.3     COCH.sub.3       H                                               CH.sub.3     CO-i-C.sub.3 H.sub.7                                                                           H                                               CH.sub.3     CO-t-C.sub.4 H.sub.9                                                                           H                                               CH.sub.3     COC.sub.6 H.sub.5                                                                              H                                               CH.sub.3     CO-3-Pyridyl     H                                               CH.sub.3     CO-2-Furyl       H                                               CH.sub.3     CO-4-Thiazolyl   H                                               CH.sub.3     CO-2-Quinolyl    H                                               CH.sub.3     COOCH.sub.3      H                                               CH.sub.3     COOC.sub.2 H.sub.5                                                                             H                                               CH.sub.3     COO-n-C.sub.3 H.sub.7                                                                          H                                               CH.sub.3     COO-i-C.sub.3 H.sub.7                                                                          H                                               CH.sub.3     COO-n-C.sub.4 H.sub.9                                                                          H                                               CH.sub.3     COO-t-C.sub.4 H.sub.9                                                                          H                                               CH.sub.3     COOCH.sub.2 C.sub.6 H.sub.5                                                                    H                                               CH.sub.3     CH.sub.3         CH.sub.3                                        CH.sub.3     C.sub.2 H.sub.5  CH.sub.3                                        CH.sub.3     n-C.sub.3 H.sub.7                                                                              CH.sub.3                                        CH.sub.3     i-C.sub.3 H.sub.7                                                                              CH.sub.3                                        CH.sub.3     s-C.sub.4 H.sub.9                                                                              CH.sub.3                                        CH.sub.3     t-C.sub.4 H.sub.9                                                                              CH.sub.3                                        CH.sub.3     n-C.sub.5 H.sub.11                                                                             CH.sub.3                                        CH.sub.3     n-C.sub.6 H.sub.13                                                                             CH.sub.3                                        CH.sub.3     n-C.sub.12 H.sub.25                                                                            CH.sub.3                                        CH.sub.3     Cyclopropyl      CH.sub.3                                        CH.sub.3     Cyclobutyl       CH.sub.3                                        CH.sub.3     Cyclopentyl      CH.sub.3                                        CH.sub.3     Cyclohexyl       CH.sub.3                                        CH.sub.3     Cyclopentyl      CH.sub.3                                        CH.sub.3     CHO              CH.sub.3                                        CH.sub.3     COCH.sub.3       CH.sub.3                                        CH.sub.3     CO-i-C.sub.3 H.sub.7                                                                           CH.sub.3                                        CH.sub.3     CO-t-C.sub.4 H.sub.9                                                                           CH.sub.3                                        CH.sub.3     COC.sub.6 H.sub.5                                                                              CH.sub.3                                        CH.sub.3     CO-3-Pyridyl     CH.sub.3                                        CH.sub.3     CO-2-Furyl       CH.sub.3                                        CH.sub.3     CO-4-Thiazolyl   CH.sub.3                                        CH.sub.3     CO-2-Quinolyl    CH.sub.3                                        CH.sub.3     COOCH.sub.3      CH.sub.3                                        CH.sub.3     COOC.sub.2 H.sub.5                                                                             CH.sub.3                                        CH.sub.3     COO-n-C.sub.3 H.sub.7                                                                          CH.sub.3                                        CH.sub.3     COO-i-C.sub.3 H.sub.7                                                                          CH.sub.3                                        CH.sub.3     COO-n-C.sub.4 H.sub.9                                                                          CH.sub.3                                        CH.sub.3     COO-t-C.sub.4 H.sub.9                                                                          CH.sub.3                                        CH.sub.3     COOCH.sub.2 C.sub.6 H.sub.5                                                                    CH.sub.3                                        H            CH.sub.3         H                                               H            i-C.sub.3 H.sub.7                                                                              H                                               H            t-C.sub.4 H.sub.9                                                                              H                                               H            n-C.sub.6 H.sub.13                                                                             H                                               H            Cyclopropyl      H                                               H            cyclohexyl       H                                               H            COCH.sub.3       H                                               H            CO-t-C.sub.4 H.sub.9                                                                           H                                               H            COC.sub.6 H.sub.5                                                                              H                                               H            CO-3-Pyridyl     H                                               H            CO-2-Furyl       H                                               H            COOCH.sub.3      H                                               H            COOi-C.sub.3 H.sub.7                                                                           H                                               H            COOt-C.sub.4 H.sub.9                                                                           H                                               H            COOCH.sub.2 C.sub.6 H.sub.5                                                                    H                                               H            CH.sub.3         CH.sub.3                                        H            i-C.sub.3 H.sub.7                                                                              CH.sub.3                                        H            t-C.sub.4 H.sub.9                                                                              CH.sub.3                                        H            n-C.sub.6 H.sub.13                                                                             CH.sub.3                                        H            Cyclopropyl      CH.sub.3                                        H            Cyclohexyl       CH.sub.3                                        H            COCH.sub.3       CH.sub.3                                        H            O-t-C.sub.4 H.sub.9                                                                            CH.sub.3                                        H            COC.sub.6 H.sub.5                                                                              CH.sub.3                                        H            CO-3-Pyridyl     CH.sub.3                                        H            CO-2-Furyl       CH.sub.3                                        H            COOCH.sub.3      CH.sub.3                                        H            COOi-C.sub.3 H.sub.7                                                                           CH.sub.3                                        H            COOt-C.sub.4 H.sub.9                                                                           CH.sub.3                                        H            COOCH.sub.2 C.sub.6 H.sub.5                                                                    CH.sub.3                                        ______________________________________                                         ##STR10##                                                                     ##STR11##                H                                                    ##STR12##                H                                                    ##STR13##                H                                                    ##STR14##                H                                                    ##STR15##                H                                                    ##STR16##                CH.sub.3                                             ##STR17##                CH.sub.3                                             ##STR18##                CH.sub.3                                             ##STR19##                CH.sub.3                                             ##STR20##                CH.sub.3                                            ______________________________________                                    

The compounds I are suitable as fungicides.

The compounds I are distinguished by an outstanding activity against abroad spectrum of phytopathogenic fungi, in particular from the class ofAscomycetes and Basidiomycetes. They are systemically active in somecases and can be employed as foliar and soil fungicides.

They are of particular importance for the control of a multiplicity offungi on various crop plants such as wheat, rye, barley, oats, rice,corn, grass, cotton, soybean, coffee, sugar cane, grapes, fruit anddecorative plants and vegetable plants such as cucumbers, beans andCucurbitaceae, and on the seeds of these plants.

They are specifically suitable for the control of the following plantdiseases: Erysiphe graminis (powdery mildew) in cereals, Erysiphecichoracearum and Sphaerotheca fuliginea on Cucurbitaceae, Podosphaeraleucotricha on apples, Uncinula necator on vines, Puccinia species oncereals., Rhizoctonia species on cotton and lawns, Ustilago species oncereals and sugar cane, Venturia inaequalis (scab) on apples,Helminthosporium species on cereals, Septoria nodorum on wheat, Botrytiscinerea (gray mold) on strawberries, vines, Cercospora arachidicola ongroundnuts, Pseudocercosporella herpotrichoides on wheat, barley,Pyricularia oryzae on rice, Phytophthora infestans on potatoes andtomatoes, Fusarium and Verticillium species on various plants,Plasmopara viticola on vines, Alternaria species on vegetables andfruit.

The compounds I are applied by treating the fungi or the plants, seeds,materials or the soil to be protected from fungal attack with afungicidally effective amount of the active compounds. They are appliedbefore or after the infection of the materials, plants or seeds by thefungi.

They can be converted into the customary formulations, such assolutions, emulsions, suspensions, dusts, powders, pastes and granules.The application form depends on the particular intended use; they shouldin any case guarantee a fine and uniform dispersion of theortho-substituted benzyl ester of a cyclopropanecarboxylic acid. Theformulations are prepared in a known manner, eg. by extending the activecompound with solvents and/or carriers, if desired using emulsifiers anddispersants, it also being possible to use other organic solvents asauxiliary solvents when water is used as a diluent. Suitable auxiliarysubstances for this purpose are essentially: solvents such as aromatics(eg. xylene), chlorinated aromatics (eg. chlorobenzenes), paraffins (eg.mineral oil fractions), alcohols (eg. methanol, butanol), ketones (eg.cyclohexanone), amines (eg. ethanolamine, dimethylformamide) and water;carriers such as ground natural minerals (eg. kaolins, clays, talc,chalk) and ground synthetic minerals (eg. highly disperse silicic acid,silicates); emulsifiers such as nonionic and anionic emulsifiers (eg.polyoxyethylene fatty alcohol ethers, alkylsulfonates andarylsulfonates) and dispersants such as lignin-sulfite waste liquors andmethylcellulose.

The fungicidal compositions in general contain from 0.1 to 95,preferably from 0.5 to 90%, by weight of active compound.

Depending on the type of effect desired, the application rates are from0.01 to 2.0 kg of active compound per ha.

In seed treatment, active compound amounts of from 0.001 to 0.1 g,preferably 0.01 to 0.05 g, per kilogram of seed are in general needed.

The compositions according to the invention can also be present asfungicides together with other active compounds in the application form,eg. with herbicides, insecticides, growth regulators, fungicides oralternatively with fertilizers.

On mixing with fungicides, in many cases an increase in the fungicidalspectrum of action is obtained here.

The following list of fungicides with which the compounds according tothe invention can be applied together should illustrate the combinationpossibilities, but not restrict them:

sulfur, dithiocarbamates and their derivatives, such as ferricdimethyldithiocarbamate, zinc dimethyldithiocarbamate, zincethylenebisdithiocarbamate, manganese ethylenebisdithiocarbamate,manganese zinc ethylenediamine bisdithiocarbamate, tetramethylthiuramdisulfide, ammonia complex of zinc (N,N-ethylenebisdithiocarbamate),ammonia complex of zinc (N,N'-propylenebisdithiocarbamate), zinc(N,N'-propylenebisdithiocarbamate), N,N'-polypropylenebis(thiocarbamoyl)disulfide;

nitro derivatives, such as dinitro(-1-methylheptyl)phenyl crotonate,2-sec-butyl-4,6-dinitrophenyl 3,3-dimethylacrylate,2-sec-butyl-4,6-dinitrophenyl isopropylcarbonate, diisopropyl5-nitroisophthalate;

heterocyclic substances, such as 2-heptadecyl-2-imidazoline acetate,2,4-dichloro-6-(o-chloroanilino)-s-triazine, O,O-diethylphthalimidophosphonothioate, 5-amino-1-[bis(dimethylamino)phosphinyl]-3-phenyl-1,2,4-triazole,2,3-dicyano-1,4-dithioanthraquinone,2-thio-1,3-dithiolo[4,5-b]quinoxaline, methyl-1-(butylcarbamoyl)-2-benzimidazole carbamate,2-methoxycarbonylaminobenzimidazole, 2-(fur-2-yl)benzimidazole,2-(thiazol-4-yl)benzimidazole,N-(1,1,2,2-tetrachloroethylthio)tetrahydrophthalimide,N-trichloromethylthiotetrahydrophthalimide,N-trichloromethylthiophthalimide;

N-dichlorofluoromethylthio-N',N'-dimethyl-N-phenylsulfadiamide,5-ethoxy-3-trichloromethyl-1,2,3-thiadiazole,2-thiocyanatomethylthiobenzothiazole, 1,4-dichloro-2,5-dimethoxybenzene,4-(2-chlorophenylhydrazono)-3-methyl-5-isoxazolone,2-thiopyridine-1-oxide, 8-hydroxyquinoline or its copper salt,2,3-dihydro-5-carboxanilido-6-methyl-1,4-oxathiin,2,3-dihydro-5-carboxanilido-6-methyl-1,4-oxathiin-4,4-dioxide,2-methyl-5,6-dihydro-4H-pyran-3-carboxanilide,2-methylfuran-3-carboxanilide, 2,5-dimethylfuran-3-carboxanilide,2,4,5-trimethylfuran-3-carboxanilide,N-cyclohexyl-2,5-dimethylfuran-3-carboxamide,N-cyclohexyl-N-methoxy-2,5-dimethylfuran-3-carboxamide,2-methylbenzanilide, 2-iodobenzanilide,N-formyl-N-morpholine-2,2,2-trichloroethyl acetal,piperazine-1,4-diylbis(1-(2,2,2-trichloroethyl))formamide,1-(3,4-dichloroanilino)-1-formylamino-2,2,2-trichloroethane,2,6-dimethyl-N-tridecylmorpholine or its salts,2,6-dimethyl-N-cyclododecylmorpholine or its salts,N-[3-(p-tert-butylphenyl)-2-methylpropyl]-cis-2,6-dimethylmorpholine,N-[3-(p-tert-butylphenyl)-2-methylpropyl]piperidine,-1-[2-(2,4-dichlorophenyl)-4-ethyl-1,3-dioxolan-2-ylethyl]-1H-1,2,4-triazole,1-[2-(2,4-dichlorophenyl)-4-n-propyl-1,3-dioxolan-2-ylethyl]-1H-1,2,4-triazole,N-(n-propyl)-N-(2,4,6-trichlorophenoxyethyl)-N'-imidazolylurea,1-(4-chlorophenoxy)-3,3-dimethyl-1-(1H-1,2,4-triazol-1-yl)-2-butanone,1-(4-chlorophenoxy)-3,3-dimethyl-1-(1H-1,2,4-triazol -1-yl)-2-butanol,α-(2-chlorophenyl)-α-(4-chlorophenyl)-5-pyrimidinemethanol,5-butyl-2-dimethylamino-4-hydroxy-6-methylpyrimidine,bis(p-chlorophenyl)-3-pyridinemethanol,1,2-bis(3-ethoxycarbonyl-2-thioureido)benzene,1,2-bis(3-methoxycarbonyl-2-thioureido)benzene,

and also various fungicides, such as dodecylguanidine acetate,3-[3-(3,5-dimethyl-2-oxycyclohexyl)-2-hydroxyethyl]glutarimide,hexachlorobenzene, DL-methyl-N-(2,6-dimethylphenyl)-N-2-furoylalaninate, DL-N-(2,6-dimethylphenyl)-N-(2'- methoxyacetyl)alanine methylester, N-(2,6-dimethylphenyl)-N-chloroacetyl-D,L-2-aminobutyrolactone,DL-N-(2,6-dimethylphenyl)-N-(phenylacetyl)alanine methyl ester,5-methyl-5-vinyl-3-(3,5-dichlorophenyl)-2,4-dioxo-1,3-oxazolidine,3-[3,5-dichlorophenyl-(5-methyl-5-methoxymethyl]-1,3-oxazolidine-2,4-dione,3-(3,5-dichlorophenyl)-1-isopropylcarbamoylhydantoin,N-(3,5-dichlorophenyl)-1,2-dimethylcyclopropane-1,2-dicarboximide,2-cyano-[N-ethylaminocarbonyl-2-methoximino]acetamide,1-[2-(2,4-dichlorophenyl)pentyl]-1H-1,2,4-triazole,2,4-difluoro-α-(1H-1,2,4-triazolyl-1-methyl)benzhydryl alcohol,N-(3-chloro-2,6-dinitro-4-trifluoromethylphenyl)-5-trifluoromethyl-3-chloro-2-aminopyridine,1-((bis(4-fluorophenyl)methylsilyl)methyl)-1H-1,2,4-triazole.

The compounds of the formula I are additionally suitable to controlpests from the class of insects, arachnida and nematodes effectively.They can be employed as pesticides in plant protection and in thehygiene, stored products protection and veterinary sector.

The harmful insects include from the order of the butterflies(Lepidoptera), for example, Agrotis ypsilon, Agrotis segetum, Alabamaargillacea, Anticarsia gemmatalis, Argyresthia conjugella, Autographagamma, Bupalus piniarius, Cacoecia murinana, Capua reticulana,Cheimatobia brumata, Choristoneura fumiferana, Choristoneuraoccidentalis, Cirphis unipuncta, Cydia pomonella, Dendrolimus pini,Diaphania nitidalis, Diatraea grandiosella, Earias insulana,Elasmopalpus lignosellus, Eupoecilia ambiguella, Evetria bouliana,Feltia subterranea, Galleria mellonella, Grapholita funebrana,Grapholita molesta, Heliothis armigera, Heliothis virescens, Heliothiszea, Hellula undalis, Hibernia defoliaria, Hyphantria cunea, Hyponomeutamalinellus, Keiferia lycopersicella, Lambdina fiscellaria, Laphygmaexigua, Leucoptera coffeella, Leucoptera scitella, Lithocolletisblancardella, Lobesia botrana, Loxostege sticticalis, Lymantria dispar,Lymantria monacha, Lyonetia clerkella, Malacosoma neustria, Mamestrabrassicae, Orgyia pseudotsugata, Ostrinia nubilalis, Panolis flammea,Pectinophora gossypiella, Peridroma saucia, Phalera bucephala,Phthorimaea operculella, Phyllocnistis citrella, Pieris brassicae,Plathypena scabra, Plutella xylostella, Pseudoplusia includens,Rhyacionia frustrana, Scrobipalpula absoluta, Sitotroga cerealella,Sparganothis pilleriana, Spodoptera frugiperda, Spodoptera littoralis,Spodoptera litura, Thaumatopoea pityocampa, Tortrix viridana,Trichoplusia ni, Zeiraphera canadensis.

From the order of the beetles (Coleoptera), for example, Agrilussinuatus, Agriotes lineatus, Agriotes obscurus, Amphimallussolstitialis, Anisandrus dispar, Anthonomus grandis, Anthonomus pomorum,Atomaria linearis, Blastophagus piniperda, Blitophaga undata, Bruchusrufimanus, Bruchus pisorum, Bruchus lentis, Byctiscus betulae, Cassidanebulosa, Cerotoma trifurcata, Ceuthorrhynchus assimilis, Ceuthorrynchusnapi, Chaetocnema tibialis, Conoderus vespertinus, Crioceris asparagi,Diabrotica longicornis, Diabrotica 12-punctata, Diabrotica virgifera,Epilachna varivestis, Epitrix hirtipennis, Eutinobothrus brasiliensis,Hylobius abietis, Hypera brunneipennis, Hypera postica, Ips typographus,Lema bilineata, Lema melanopus, Leptinotarsa decemlineata, Limoniuscalifornicus, Lissorhoptrus oryzophilus, Melanotus communis, Meligethesaeneus, Melolontha hippocastani, Melolontha melolontha, Onlema oryzae,Ortiorrhynchus sulcatus, Otiorrhynchus ovatus, Phaedon cochleariae,Phyllotetra chrysocephala, Phyllophaga sp., Phyllopertha horticola,Phyllotetra nemorum, Phyllotetra striolata, Popillia japonica, Sitonalineatus, Sitophilus granaria.

From the order of the dipterous insects (Diptera), for example, Aedesaegypti, Aedes vexans, Anastrepha ludens, Anopheles maculipennis,Ceratitis capitata, Chrysomya bezziana, Chrysomya hominivorax, Chrysomyamacellaria, Contarinia sorghicola, Cordylobia anthropophaga, Culexpipiens, Dacus cucurbitae, Dacus oleae, Dasineura brassicae, Fanniacanicularis, Gasterophilus intestinalis, Glossina morsitans, Haematobiairritans, Haplodiplosis equestris, Hylemyia platura, Hypoderma lineata,Liriomyza sativae, Liriomyza trifolii, Lucilia caprina, Lucilia cuprina,Lucilia sericata, Lycoria pectoralis, Mayetiola destructor, Muscadomestica, Muscina stabulans, Oestrus ovis, Oscinella frit, Pegomyahysocyami, Phorbia antiqua, Phorbia brassicae, Phorbia coarctata,Rhagoletis cerasi, Rhagoletis pomonella, Tabanus bovinus, Tipulaoleracea, Tipula paludosa.

From the order of the thrips (Thysanoptera), for example, Frankliniellafusca, Frankliniella occidentalis, Frankliniella tritici, Scirtothripscitri, Thrips oryzae, Thrips palmi, Thrips tabaci.

From the order of the hymenopterous insects (Hymenoptera), for example,Athalia rosae, Atta cephalotes, Atta sexdens, Atta texana, Hoplocampaminuta, Hoplocampa testudinea, Monomorium pharaonis, Solenopsisgeminata, Solenopsis invicta.

From the order of the bed bugs (Heteroptera), for example, Acrosternumhilare, Blissus leucopterus, Cyrtopeltis notatus, Dysdercus cingulatus,Dysdercus intermedius, Eurygaster integriceps, Euschistusimpictiventris, Leptoglossus phyllopus, Lygus lineolaris, Lyguspratensis, Nezara viridula, Piesma quadrata, Solubea insularis, Thyantaperditor.

From the order of the plant-sucking insects (Homoptera), for example,Acyrthosiphon onobrychis, Adelges laricis, Aphidula nasturtii, Aphisfabae, Aphis pomi, Aphis sambuci, Brachycaudus cardui, Brevicorynebrassicae, Cerosipha gossypii, Dreyfusia nordmannianae, Dreyfusiapiceae, Dyasphis radicola, Dysaulacorthum pseudosolani, Empoasca fabae,Macrosiphum avenae, Macrosiphum euphorbiae, Macrosiphon rosae, Megouraviciae, Metopolophium dirhodum, Myzodes persicae, Myzus cerasi,Nilaparvata lugens, Pemphigus bursarius, Perkinsiella saccharicida,Phorodon humuli, Psylla mali, Psylla piri, Rhopalomyzus ascalonicus,Rhopalosiphum maidis, Sappaphis mala, Sappaphis mali, Schizaphisgraminum, Schizoneura lanuginosa, Trialeurodes vaporariorum, Viteusvitifolii.

From the order of the termites (Isoptera), for example, Calotermesflavicollis, Leucotermes flavipes, Reticulitermes lucifugus, Termesnatalensis.

From the order of the orthopterous insects (Orthoptera), for example,Acheta domestica, Blatta orientalis, Blattella germanica, Forficulaauricularia, Gryllotalpa gryllotalpa, Locusta migratoria, Melanoplusbivittatus, Melanoplus femurrubrum, Melanoplus mexicanus, Melanoplussanguinipes, Melanoplus spretus, Nomadacris septemfasciata, Periplanetaamericana, Schistocerca americana, Schistocerca peregrina, Stauronotusmaroccanus, Tachycines asynamorus.

From the class of the Arachnoidea, for example spiders (Acarina) such asAmblyomma americanum, Amblyomma variegatum, Argas persicus, Boophilusannulatus, Boophilus decoloratus, Boophilus microplus, Brevipalpusphoenicis, Bryobia praetiosa, Dermacentor silvarum, Eotetranychuscarpini, Eriophyes sheldoni, Hyalomma truncatum, Ixodes ricinus, Ixodesrubicundus, Ornithodorus moubata, Otobius megnini, Paratetranychuspilosus, Dermanyssus gallinae, Phyllocoptruta oleivora,Polyphagotarsonemus latus, Psoroptes ovis, Rhipicephalus appendiculatus,Rhipicephalus evertsi, Sarcoptes scabiei, Tetranychus cinnabarinus,Tetranychus kanzawai, Tetranychus pacificus, Tetranychus telarius,Tetranychus urticae.

From the class of the nematodes, for example, root gall nematodes, eg.Meloidogyne hapla, Meloidogyne incognita, Meloidogyne javanica,cyst-forming nematodes, eg. Globodera rostochiensis, Heterodera avenae,Heterodera glycines, Heterodera schachtii, Heterodera trifolii, stem andleaf eelworms, eg. Belonolaimus longicaudatus, Ditylenchus destructor,Ditylenchus dipsaci, Heliocotylenchus multicinctus, Longidoruselongatus, Radopholus similis, Rotylenchus robustus, Trichodorusprimitivus, Tylenchorhynchus claytoni, Tylenchorhynchus dubius,Pratylenchus neglectus, Pratylenchus penetrans, Pratylenchus curvitatus,Pratylenchus goodeyi.

The active compounds can be applied as such or in the form of theirformulations or the application forms prepared therefrom, eg. in theform of directly sprayable solutions, powders, suspensions ordispersions, emulsions, oil dispersions, pastes, dusts, scatteringcompositions or granules by spraying, atomizing, dusting, scattering orpouring. The application forms depend entirely on the purposes of use;they should in any case as far as possible guarantee the finestdispersion of the active compounds according to the invention.

The active compound concentrations in the ready-for-applicationpreparations can be varied within substantial ranges.

In general, they are from 0.0001 to 10%, preferably from 0.01 to 1%.

The active compounds can also be used with success in ultra-low volumeprocesses (ULV), where it is possible to apply formulations containingmore than 95% by weight of active compound or even the active compoundwithout additives.

The application rate of active compound for controlling pests underoutdoor conditions is from 0.1 to 2.0, preferably from 0.2 to 1.0 kg/ha.

For the preparation of directly sprayable solutions, emulsions, pastesor oil dispersions, mineral oil fractions of medium to high boilingpoint, such as kerosene or diesel oil, and also coal tar oils and oilsof vegetable or animal origin, aliphatic, cyclic and aromatichydrocarbons, eg. benzene, toluene, xylene, paraffin,tetrahydronaphthalene, alkylated naphthalenes or their derivatives,methanol, ethanol, propanol, butanol, chloroform, carbon tetrachloride,cyclohexanol, cyclohexanone, chlorobenzene, isophorone, strongly polarsolvents, eg. dimethylformamide, dimethyl sulfoxide, N-methylpyrrolidoneand water are suitable.

Aqueous application forms can be prepared from emulsion concentrates,pastes or wettable powders (oil dispersions) by addition of water. Forthe preparation of emulsions, pastes or oil dispersions, the substancescan be homogenized in water as such or dissolved in an oil or solvent,by means of wetting agents, tackifiers, dispersants or emulsifiers.However, the concentrates consisting of active substance, wetting agent,tackifier, dispersant or emulsifier and possibly solvent or oil can alsobe prepared, which are suitable for dilution with water.

Suitable surface-active substances are alkali metal, alkaline earthmetal and ammonium salts of lignosulfonic acid, naphthalenesulfonicacid, phenolsulfonic acid, dibutylnaphthalenesulfonic acid,alkylarylsulfonates, alkylsulfates, alkylsulfonates, fatty alcoholsulfates and fatty acids and their alkali metal and alkaline earth metalsalts, salts of sulfated fatty alcohol glycol ethers, condensationproducts of sulfonated naphthalene and naphthalene derivatives withformaldehyde, condensation products of naphthalene or ofnaphthalenesulfonic acid with phenol and formaldehyde, polyoxyethyleneoctylphenyl ether, ethoxylated isooctylphenol, octylphenol, nonylphenol,alkylphenyl polyglycol ether, tributylphenyl polyglycol ether, alkylarylpolyether alcohols, isotridecyl alcohol, fatty alcohol ethylene oxidecondensates, ethoxylated castor oil, polyoxyethylene alkyl ethers,ethoxylated polyoxypropylene, lauryl alcohol polyglycol ether acetal,sorbitol esters, lignin-sulfite waste liquors and methylcellulose.

Powders, scattering compositions and dusts can be prepared by mixing orjoint grinding of the active substances with a solid carrier.

The formulations in general contain from 0.01 to 95% by weight,preferably from 0.1 to 90% by weight, of the active compound. The activecompounds are employed here in a purity of from 90% to 100%, preferably95% to 100% (according to NMR spectrum).

Examples of formulations are:

I. 5 parts by weight of an active compound are intimately mixed with 95parts by weight of finely divided kaolin. A dust which contains 5% byweight of the active compound is obtained in this way.

II. 30 parts by weight of an active compound are intimately mixed with amixture of 92 parts by weight of powdered silica gel and 8 parts byweight of paraffin oil which has been sprayed on the surface of thissilica gel. A preparation of the active compound having good adhesion isobtained in this way (active compound content 23% by weight).

III. 10 parts by weight of an active compound are dissolved in a mixturewhich consists of 90 parts by weight of xylene, 6 parts by weight of theaddition product of 8 to 10 mol of ethylene oxide to 1 mol of oleic acidN-monoethanolamide, 2 parts by weight of calcium salt ofdodecylbenzenesulfonic acid and 2 parts by weight of the additionproduct of 40 mol of ethylene oxide to 1 mol of castor oil (activecompound content 9% by weight).

IV. 20 parts by weight of an active compound are dissolved in a mixturewhich consists of 60 parts by weight of cyclohexanone, 30 parts byweight of isobutanol, 5 parts by weight of the addition product of 7 molof ethylene oxide to 1 mol of isooctylphenol and 5 parts by weight ofthe 15 addition product of 40 mol of ethylene oxide to 1 mol of castoroil (active compound content 16% by weight).

V. 80 parts by weight of an active compound are well mixed with 3 partsby weight of the sodium salt of diisobutyl-naphthalene-alpha-sulfonicacid, 10 parts by weight of the sodium salt of a lignosulfonic acid froma sulfite waste liquor and 7 parts by weight of powdered silica gel andthe mixture is ground in a hammer mill (active compound content 80% byweight).

VI. 90 parts by weight of an active compound are mixed with parts byweight of N-methyl-α-pyrrolidone and a solution is obtained which issuitable for application in the form of very small drops (activecompound content 90% by weight).

VII. 20 parts by weight of an active compound are dissolved in a mixturewhich consists of 40 parts by weight of cyclohexanone, 30 parts byweight of isobutanol, 20 parts by weight of the addition product of 7mol of ethylene oxide to 1 mol of isooctylphenol and 10 parts by weightof the addition product of 40 mol of ethylene oxide to 1 mol of castoroil. By pouring the solution into and finely dispersing it in 100,000parts by weight of water, an aqueous dispersion is obtained whichcontains 0.02% by weight of the active compound.

VIII. 20 parts by weight of an active compound are well mixed with 3parts by weight of the sodium salt of diisobutyl-naphthalene-α-sulfonicacid, 17 parts by weight of the sodium salt of a lignosulfonic acid froma sulfite waste liquor and 60 parts by weight of powdered silica gel andthe mixture is ground in a hammer mill. By finely dispersing the mixturein 20,000 parts by weight of water, a spray liquor is obtained whichcontains 0.1% by weight of the active compound.

Granules, eg. coated, impregnated and homogeneous granules, can beproduced by binding the active compounds to solid carriers. Solidcarriers are eg. mineral earths, such as silica gel, silicic acids,silicates, talc, kaolin, attapulgite, limestone, lime, chalk, bole,loess, clay, dolomite, diatomaceous earth, calcium sulfate and magnesiumsulfate, magnesium oxide, ground synthetic materials, fertilizers, suchas eg. ammonium sulfate, ammonium phosphate, ammonium nitrate, ureas andvegetable products, such as grain meal, tree bark, wood and nut shellmeal, cellulose powder and other solid carriers.

Oils of various types, herbicides, fungicides, other pesticides andbactericides can be added to the active compounds, if appropriate alsojust immediately before application (tank mix). These agents can beadmixed to the compositions according to the invention in the weightratio 1:10-10:1.

SYNTHESIS EXAMPLES

The procedures presented in the synthesis examples below are utilizedwith appropriate modification of the starting compounds to obtainfurther compounds I. The compounds thus obtained are shown in thefollowing table C with physical data.

The following examples are intended to illustrate the preparation of thenovel active compounds.

EXAMPLE 1

Preparation of [2-(α-Methoxyimino)Methoxycarbonylmethyl]Benzaldazine(No. I.11)

2.2 g (10 mmol) of methyl α-methoxyimino-(2-formylphenyl)acetate aredissolved in 50 ml of glacial acetic acid and 0.25 g (5 mmol) ofhydrazine hydrate is added at room temperature (RT). The color of thereaction mixture becomes lighter, and after stirring for 5 min alight-yellow precipitate is formed. The mixture is stirred for a further25 min at RT, and the precipitate is filtered off with suction andwashed with pentane. The title compound is obtained as a light-yellowpowder of m.p. 207°-209° C.; yield 1.6 g (73% of theory).

¹ H NMR (CDCl₃, δ scale): 3.86 (s, 3 H, COOCH₃); 4.04 (s, 3 H, NOCH₃);7.29 (mc, 1 H), 7.52 (mc, 2 H) and 7.91 (mc, 1 H; aromatic protons );8.47 (s, 1 H, CH═N )

EXAMPLE 2

Preparation of-1-Methyl-1-(4'-Methylphenyl)-4-[2'-(α-Methoxyimino)Methoxycarbonylmethylene]Phenyl-2,3-Diazabutadiene(No. 1.04)

The two-phase mixture of 10.1 g (200 mmol) of 100% strength hydrazinehydrate, 2.5 ml of water and 13.4 g (100 mmol) of 4-methylacetophenoneis heated to 60° C. for 10 h. It is allowed to cool, treated with waterand extracted 3× with ether, and the organic phases are dried oversodium sulfate and concentrated in vacuo. 12.5 g (85% of theory) of4-methylacetophenone hydrazone are obtained as an almost colorless oil.

1.6 g of the 4-methylacetophenone hydrazone prepared as described aboveare dissolved in 100 ml of tetrahydrofuran and added dropwise at RT to asolution of 2.2 g (10 mmol) of methyl α-methoxy-imino(2-formylphenyl)acetate in 30 ml of glacial acetic acid. The mixture is stirred for 30min, neutralized with saturated sodium carbonate solution with slightice-cooling and extracted with diethyl ether, and the extract is driedover sodium sulfate to which a spatula tipful of sodium hydrogencarbonate has been added and is concentrated in vacuo. After separationof the symmetrical azines obtained as by-products (cf. scheme 1) bycolumn chromatography (ethyl acetate/cyclohexane 96:4 to 80:20, silicagel 60), the title compound is obtained as yellow crystals, m.p.127°-129° C., in 1.7 g (48% of theory) yield.

¹ H NMR (CDCl₃, δ scale): 2.41 and 2.46 (2 s, 3 H each, Ar--CH₃ andN═C--CH₃); 3.82 (s, 3 H, COOCH₃); 4.04 (s, 3 H, NOCH₃); 7.1-7.3 (m, 3H); 7.48 (mc, 2 H), 7.78 (d, 2 H) and 7.85 (mc, 1 H; aromatic protons);8.38 (s, 1 H, CH═N).

EXAMPLE 3

Preparation of-1-Methyl-1-(4'-Methylphenyl)-4-[2'-(α-Methoxyimino)Methylaminocarbonylmethylene]Phenyl-2,3-Diazabutadiene(No. I.09)

1.0 g (2.9 mmol) of1-methyl-1-(4'-methylphenyl)-4-[2'-(α-methoxy-imino)methoxycarbonylmethylene]phenyl-2,3-diazabutadiene(product from Example 2) is dissolved in 20 ml of tetrahydrofuran (THF),1.3 ml of 40% strength aqueous methylamine solution (14.5 mmol) areadded and the reaction mixture is stirred overnight at RT; a smallamount of a finely divided solid precipitates. This preci-pitate isfiltered off with suction and washed with pentane, the title compoundprecipitating in the filtrate. Precipitation is completed by addition offurther pentane. The precipitate is filtered off with suction, washedwith pentane and dried by allowing to stand in air. Pale yellowcrystals, m.p. 182°-185° C., yield 0.8 g (80% of theory).

¹ H NMR (CDCl₃, δ scale): 2.42 and 2.47 (2 s, 3 H each, Ar--CH₃ andN═C--CH₃); 2.93 (d, 3 H, CONHCH₃); 3.96 (s, 3 H, NOCH₃); 6.87 (br, H,CONH); 7.24 (mc, 3 H), 7.50 (mc, 2 H), 7.80 (d, 2 H) and 8.03 (mc, 1 H;aromatic protons); 8.27 (s, 1 H, CH═N).

                                      TABLE C                                     __________________________________________________________________________     ##STR21##                          I                                                                          melting                                                                       point                                        No.                                                                              R  A  B            Y    Z     [°C.]                                 __________________________________________________________________________    I.01                                                                             H  CH.sub.3                                                                         C.sub.6 H.sub.5                                                                            OCH.sub.3                                                                          NOCH.sub.3                                                                          125-126                                      I.02                                                                             H  CH.sub.3                                                                         4-ClC.sub.6 H.sub.4                                                                        OCH.sub.3                                                                          NOCH.sub.3                                                                          162-166                                      I.03                                                                             H  CH.sub.3                                                                         3,5-Cl.sub.2C.sub.6 H.sub.3                                                                OCH.sub.3                                                                          NOCH.sub.3                                                                          155-159                                      I.04                                                                             H  CH.sub.3                                                                         4-CH.sub.3C.sub.6 H.sub.4                                                                  OCH.sub.3                                                                          NOCH.sub.3                                                                          129                                          I.05                                                                             H  CH.sub.3                                                                         4-C(CH.sub.3).sub.3C.sub.6 H.sub.4                                                         OCH.sub.3                                                                          NOCH.sub.3                                                                          122                                          I.06                                                                             H  CH.sub.3                                                                         C.sub.6 H.sub.5                                                                            NHCH.sub.3                                                                         NOCH.sub.3                                                                          140-143                                      I.07                                                                             H  CH.sub.3                                                                         4-ClC.sub.6 H.sub.4                                                                        NHCH.sub.3                                                                         NOCH.sub.3                                                                          145-148                                      I.08                                                                             H  CH.sub.3                                                                         3,5-Cl.sub.2C.sub.6 H.sub.3                                                                NHCH.sub.3                                                                         NOCH.sub.3                                                                          155-159                                      I.09                                                                             H  CH.sub.3                                                                         4-CH.sub.3C.sub.6 H.sub.4                                                                  NHCH.sub.3                                                                         NOCH.sub.3                                                                          182-185                                      I.10                                                                             H  CH.sub.3                                                                         4-C(CH.sub.3).sub.3C.sub.6 H.sub.4                                                         NHCH.sub.3                                                                         NOCH.sub.3                                                                          131                                          I.11                                                                             H  H  2-C(CO.sub.2 H.sub.3)NOCH.sub.3                                                            OCH.sub.3                                                                          NOCH.sub.3                                                                          207-209                                               C.sub.6 H.sub.4                                                      __________________________________________________________________________

Examples of the action against harmful fungi

The fungicidal action of the compounds of the general formula I can beshown by the following tests:

The active compounds were prepared as a 20% strength emulsion in amixture of 70% by weight of cyclohexanone, 20% by weight of Nekanil® LN(Lutensol® AP6, wetting agent with emulsifying and dispersant actionbased on ethoxylated alkylphenols) and 10% by weight of Emulphor® EL(Emulan® EL, emulsifier based on ethoxylated fatty alcohols) andappropriately diluted to the desired concentration with water.

A. Botrytis cinerea

Slices of green peppers were sprayed with the active compoundpreparation until dripping wet. After drying, the fruit slices weresprayed with a spore suspension of the fungus Botrytis cinerea (1.7×10⁶spores per ml of a 2% strength biomalt solution) and kept for 4 days at18° C. at high atmospheric humidity. Assessment was carried outvisually.

In this test, the untreated controls showed an attack of 90% while thefruit slices treated in each case with 500 ppm-containing activecompound preparation of compounds 1.01, 1.04, 1.06 and I.08 wereattacked to 15% at most.

B. Plasmopara viticola

Potted vines (variety: M uller Thurgau) were sprayed with the activecompound preparation until dripping wet. After 8 days, the plants weresprayed with a zoospore suspension of the fungus Plasmopara viticola andkept for 5 days at 20°-30° C. at high atmospheric humidity. Beforeassessment, the plants were then kept for 16 h at high atmospherichumidity. Assessment was carried out visually.

In this test, the untreated controls showed an attack of 70% while theplants treated with 63 ppm-containing active compound preparation of thecompounds I.01, I.03, I.04, I.06, I.07, I.08 and I.09 were attacked to15% at most.

Examples of the action against animal pests

It was possible to show the action of the compounds of the generalformula I against animal pests by the following tests:

The active compounds were prepared

a. as a 0.1% strength solution in acetone or

b. as a 10% strength emulsion in a mixture of 70% by weight ofcyclohexanone, 20% by weight of Nekanil® LN (Lutensol® AP6, wettingagent with emulsifying and dispersant action based on ethoxylatedalkylphenols) and 10% by weight of Emulphor® EL (Emulan® EL, emulsifierbased on ethoxylated fatty alcohols)

and appropriately diluted to the desired concentration with acetone inthe case of a. or with water in the case of b.

After conclusion of the tests, in each case the lowest concentration wasdetermined at which the compounds still produced an 80 to 100%inhibition or mortality in comparison to untreated control tests(activity threshold or minimum concentration).

We claim:
 1. A compound of the formula ##STR22## where the substituentshave the following meanings: X is hydrogen, cyano, nitro,trifluoromethyl, halogen, C₁ -C₆₋ alkyl or C₁ -C₆ -alkoxy;Y is amino,methylamino or dimethylamino; Z is CHCH₃, CHOCH₃ or NOCH₃ ; R ishydrogen or C₁ -C₆ -alkyl; A is hydrogen, C₁ -C₆ -alkyl, C₁ -C₆-haloalkyl or C₃ -C₇ -cycloalkyl; B is unsubstituted or substituted C₁-C₆ -alkyl, C₂ -C₆ -alkenyl, C₂ -C₆ -alkynyl, C₃ -C₇ -cycloalkyl, C₅ -C₇-cycloalkenyl, an unsubstituted or substituted, saturated or partiallyunsaturated heterocyclyl, unsubstituted or substituted aryl, which maybe fused, unsubstituted or substituted 5- or 6-membered heteroaryl,which may be benzo- or hetero-fused, unsubstituted or substitutedaryl-C₁ -C₆ -alkyl or heteroaryl-C₁ -C₆ -alkyl, or C(═O)W;where W ishydrogen, unsubstituted or substituted C₁ -C₆ -alkyl, C₁ -C₆ -alkoxy, C₁-C₆ -alkylthio, C₁ -C₆ -alkylamino or di-C₁ -C₆ -alkylamino,unsubstituted or substituted aryl, heteroaryl, aryloxy, arylthio,arylamino, aryl-N-(C₁ -C₆ -alkyl)amino, heteroaryloxy, heteroarylthio,heteroarylamino or heteroaryl-N-(C₁ -C₆ -alkyl)amino;or A and B,together with the C atom whose substituents they are, are anunsubstituted or substituted, saturated or unsaturated 3- to 7-memberedisocyclic ring or 5- to 7-membered heterocyclic ring, which may be fusedand which may also be quinonoid.
 2. A composition for the control ofharmful fungi, containing a solid or liquid carrier and a compound ofthe general formula I as claimed in claim
 1. 3. The compound of claim 1,wherein X is hydrogen.
 4. The compound of claim 1, wherein Y ismethylamino.
 5. The compound of claim 1, wherein Z is NOCH₃.
 6. Thecompound of claim 1, wherein R is hydrogen.
 7. The compound of claim 1,wherein A is hydrogen or methyl.
 8. The compound of claim 1, wherein Bis unsubstituted or substituted phenyl.
 9. The compound of claim 1,whereinX is hydrogen; Y is methylamino; Z is NOCH₃ ; R is hydrogen; andA is hydrogen or methyl.
 10. A process for preparing the composition ofclaim 4, comprising the step of:extending the compound with a solvent orcarrier, or mixing or joint grinding of the compound with a solidcarrier.
 11. The process of claim 10, wherein said composition comprises0.1 to 95% by weight of the compound.
 12. The method of claim 10,wherein said composition comprises 0.5 to 90% by weight of the compound.13. The compound of claim 1, wherein said heteroaryl is selected fromthe group consisting of 5-membered heteroaryls containing 1-4 nitrogenatoms or 1-3 nitrogen atoms and a sulfur or oxygen atom, benzo-fused5-membered heteroaryls containing 1-3 nitrogen atoms or a nitrogen atomand an oxygen or sulfur atom, 5-membered heteroaryls bonded vianitrogen, benzo-fused 5-membered heteroaryls bonded via nitrogen,6-membered heteroaryls containing 1-3 or 1-4 nitrogen atoms andbenzo-fused 6-membered heteroaryls containing 1-3 nitrogen atoms. 14.The compound of claim 1, wherein said heterocyclyl is selected from thegroup consisting of oxiranyl, oxetanyl, tetrahydrofuryl,tetrahydrothienyl, pyrrolidinyl, isoxazolidinyl, isothiazolidinyl,pyrazolidinyl, oxazolidinyl, thiazolidinyl, imidazolidinyl,oxadiazolidinyl, thiazolidinyl, triazolidinyl, dihydrofuryl,dihydrothienyl, dihydropyrrolyl, dihydroisoxazolyl, dihydroisothiazolyl,dihydropyrazolyl, dihydrooxazolyl, dihydrothiazolyl, dihydroimidazolyl,piperidinyl, tetrahydropyridazinyl, tetrahydropyrimidinyl,tetrahydropyrazinyl, tetrahydrotriazinyl, dihydrooxazinyl, dithianyl,tetrahydropyranyl, dioxolanyl, thiazinyl, benzothiazinyl, benzoxazinyl,dioxotetrahydrothienyl, dihydrooxazinyl, morpholinyl, anddihydroquinazolinyl.
 15. The compound of claim 1, wherein saidheteroaryl is selected from the group consisting of furyl, thienyl,pyrrolyl, isoxazolyl, isothiazolyl, pyrazolyl, oxazolyl, thiazolyl,imidazolyl, thiadiazolyl, oxadiazolyl, triazolyl, tetrazolyl, pyridyl,pyridazinyl, pyrimidinyl, pyrazinyl, triazinyl, tetrazinyl, benzofuryl,isobenzofuryl, benzothienyl, indolyl, isoindolyl, benzisoxazolyl,benzisothiazolyl, benzothiazolyl, indazolyl, benzimidazolyl,benzotriazolyl, dibenzofuryl, dibenzothienyl, carbazolyl, acridinyl,phenanthridinyl, quinolinyl, isoquinolinyl, phthalazinyl, quinazolinyl,quinoxalinyl, cinnolinyl, naphthyridinyl, pteridinyl, pyrrolopyrazinyl,pyrrolypyridazinyl, pyrrolopyrimidinyl, pyrrolopyrazinyl,pyrrolotriazinyl, furopyridinyl, furopyridazinyl, furopyrimidinyl,furopyrazinyl, thienopyridinyl, thienopyridazinyl, thienopyrimidinyl,thienopyrazinyl, imidazopyridinyl, imidazolopyridazinyl,imidazopyrimidinyl, purinyl, imidazopyrazinyl, pyrazolopyridinyl,pyrazolopyridazinyl, pyrazolopyrimidinyl, pyrazolopyrazinyl,isoxazolopyrazinyl, oxazolopyridinyl, oxazolopyrimidinyl,isothiazolopyrimidinyl, and triazolopyrimidinyl.